RU2730506C2 - Твердые формы соединения, модулирующего киназы - Google Patents

Твердые формы соединения, модулирующего киназы Download PDF

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RU2730506C2
RU2730506C2 RU2017141035A RU2017141035A RU2730506C2 RU 2730506 C2 RU2730506 C2 RU 2730506C2 RU 2017141035 A RU2017141035 A RU 2017141035A RU 2017141035 A RU2017141035 A RU 2017141035A RU 2730506 C2 RU2730506 C2 RU 2730506C2
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compound
disease
application
crystalline
solid
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RU2017141035A3 (OSRAM
RU2017141035A (ru
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Прабха Н. Ибрахим
Гэри Конрад ВАЙЗОР
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Плексксикон Инк.
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    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
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    • A61K31/436—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having oxygen as a ring hetero atom, e.g. rapamycin
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    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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RU2017141035A 2015-05-06 2016-05-05 Твердые формы соединения, модулирующего киназы RU2730506C2 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562157902P 2015-05-06 2015-05-06
US62/157,902 2015-05-06
PCT/US2016/031027 WO2016179415A1 (en) 2015-05-06 2016-05-05 Solid forms of a compound modulating kinases

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RU2017141035A RU2017141035A (ru) 2019-06-06
RU2017141035A3 RU2017141035A3 (OSRAM) 2019-08-09
RU2730506C2 true RU2730506C2 (ru) 2020-08-24

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US (4) US9802932B2 (OSRAM)
EP (2) EP3292123B1 (OSRAM)
JP (1) JP6946194B2 (OSRAM)
KR (1) KR102630889B1 (OSRAM)
CN (1) CN107548394B (OSRAM)
AU (1) AU2016258027B2 (OSRAM)
BR (1) BR112017023490B1 (OSRAM)
CA (1) CA2984910C (OSRAM)
CO (1) CO2017011534A2 (OSRAM)
CY (1) CY1123796T1 (OSRAM)
DK (1) DK3292123T3 (OSRAM)
ES (1) ES2820827T3 (OSRAM)
HR (1) HRP20201383T1 (OSRAM)
HU (1) HUE050506T2 (OSRAM)
IL (1) IL255313A0 (OSRAM)
LT (1) LT3292123T (OSRAM)
MX (1) MX386963B (OSRAM)
MY (1) MY192352A (OSRAM)
NZ (1) NZ737616A (OSRAM)
PH (1) PH12017501995A1 (OSRAM)
PT (1) PT3292123T (OSRAM)
RS (1) RS60731B1 (OSRAM)
RU (1) RU2730506C2 (OSRAM)
SG (1) SG10201912355TA (OSRAM)
SI (1) SI3292123T1 (OSRAM)
SM (1) SMT202000535T1 (OSRAM)
TW (1) TWI727949B (OSRAM)
WO (1) WO2016179415A1 (OSRAM)
ZA (1) ZA201708007B (OSRAM)

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TWI803530B (zh) 2017-10-27 2023-06-01 美商普雷辛肯公司 調節激酶之化合物之調配物
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AU2020271836B2 (en) 2019-04-09 2025-11-13 Opna Bio SA Condensed azines for EP300 or CBP modulation and indications therefor
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