RU2567044C2 - Ингибиторы 1 киназы контрольной точки клеточного цикла для усиления днк-повреждающих агентов - Google Patents
Ингибиторы 1 киназы контрольной точки клеточного цикла для усиления днк-повреждающих агентов Download PDFInfo
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- RU2567044C2 RU2567044C2 RU2011145773/15A RU2011145773A RU2567044C2 RU 2567044 C2 RU2567044 C2 RU 2567044C2 RU 2011145773/15 A RU2011145773/15 A RU 2011145773/15A RU 2011145773 A RU2011145773 A RU 2011145773A RU 2567044 C2 RU2567044 C2 RU 2567044C2
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| EP1667684A1 (en) * | 2003-09-17 | 2006-06-14 | ICOS Corporation | Use of chk1 inhibitors to control cell proliferation |
| UY29177A1 (es) * | 2004-10-25 | 2006-05-31 | Astex Therapeutics Ltd | Derivados sustituidos de purina, purinona y deazapurina, composiciones que los contienen métodos para su preparación y sus usos |
| CN101415417A (zh) * | 2006-04-04 | 2009-04-22 | 辉瑞产品公司 | (2r,z)-2-氨基-2-环己基-n-(5-(1-甲基-1h-吡唑-4-基)-1-氧代-2,6-二氢-1h-[1,2]二氮杂卓并[4,5,6-cd]吲哚-8-基)乙酰胺的组合疗法 |
| WO2008063558A2 (en) * | 2006-11-17 | 2008-05-29 | Schering Corporation | Combination of an inhibitor of dna polymerase-alpha and an inhibitor of a checkpoint kinase for proliferative disorders |
| AR071717A1 (es) * | 2008-05-13 | 2010-07-07 | Array Biopharma Inc | Pirrolo[2,3-b]piridinas inhibidoras de quinasas chk1 y chk2,composiciones farmaceuticas que las contienen,proceso para prepararlas y uso de las mismas en el tratamiento y prevencion del cancer. |
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2010
- 2010-04-09 SG SG10201404012RA patent/SG10201404012RA/en unknown
- 2010-04-09 CA CA2758300A patent/CA2758300C/en active Active
- 2010-04-09 MX MX2011010675A patent/MX341368B/es active IP Right Grant
- 2010-04-09 NZ NZ596125A patent/NZ596125A/xx not_active IP Right Cessation
- 2010-04-09 CN CN201080025806.6A patent/CN102612365B/zh not_active Expired - Fee Related
- 2010-04-09 BR BRPI1013920A patent/BRPI1013920A2/pt not_active Application Discontinuation
- 2010-04-09 KR KR1020117026769A patent/KR101676062B1/ko not_active Expired - Fee Related
- 2010-04-09 JP JP2012504909A patent/JP5805071B2/ja not_active Expired - Fee Related
- 2010-04-09 RU RU2011145773/15A patent/RU2567044C2/ru active
- 2010-04-09 SG SG2011075520A patent/SG175242A1/en unknown
- 2010-04-09 WO PCT/US2010/030634 patent/WO2010118390A1/en not_active Ceased
- 2010-04-09 SG SG10201900212QA patent/SG10201900212QA/en unknown
- 2010-04-09 AU AU2010233122A patent/AU2010233122B2/en not_active Ceased
- 2010-04-09 EP EP10721579.0A patent/EP2416773B1/en active Active
- 2010-04-09 ES ES10721579.0T patent/ES2608656T3/es active Active
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2011
- 2011-10-11 IL IL215709A patent/IL215709A/en active IP Right Grant
- 2011-11-10 ZA ZA2011/08273A patent/ZA201108273B/en unknown
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2014
- 2014-07-29 JP JP2014153687A patent/JP2014198741A/ja not_active Withdrawn
Non-Patent Citations (4)
| Title |
|---|
| MATTHEWS DJ et al. Pharmacological abrogation of S-phase check-point enhances the anti-tumor activity of gemcitabine in vivo. Cell cycle. 2007 Jan 1;6(1):104-10 [он-лайн][Найдено 2014-02-25](Найдено из Интернет: www.ncbi.nlm.nih.gov/pubmed/17245119). * |
| PARSELS LA et al.Gemcitabine sensitization by checkpoint kinase 1 inhibitorcorrelates with inhibition of Rad51 DNA damage response in pancreatic cancer cells. Mol.Cancer Ther. 2009 Jan;8(1):45-54 Реферат [он-лайн][Найдено 2014-02-25](Найдено из Интернет: www.ncbi.nlm.nih.gov/pubmed/19139112). * |
| pеферат * |
| SABLUDOFF SD et al.AZD7762, a novel checkpoint kinase inhibitor, drives checkpointabrogation and potentiates DNA-targeted therapies. Mol.Cancer Ther. 2008 Sep;7(9):2955-66 [он-лайн][Найдено 2014-02-25](Найдено из Интернет: www.ncbi.nlm.nih.gov/pubmed/18790776). * |
Also Published As
| Publication number | Publication date |
|---|---|
| JP5805071B2 (ja) | 2015-11-04 |
| SG175242A1 (en) | 2011-11-28 |
| SG10201900212QA (en) | 2019-02-27 |
| ZA201108273B (en) | 2013-07-31 |
| MX2011010675A (es) | 2012-03-16 |
| JP2014198741A (ja) | 2014-10-23 |
| CA2758300A1 (en) | 2010-10-14 |
| IL215709A (en) | 2017-06-29 |
| RU2011145773A (ru) | 2013-05-20 |
| CN102612365B (zh) | 2017-04-12 |
| ES2608656T3 (es) | 2017-04-12 |
| BRPI1013920A2 (pt) | 2016-04-05 |
| KR20120004523A (ko) | 2012-01-12 |
| JP2012523435A (ja) | 2012-10-04 |
| AU2010233122A1 (en) | 2011-11-24 |
| IL215709A0 (en) | 2012-01-31 |
| SG10201404012RA (en) | 2014-09-26 |
| KR101676062B1 (ko) | 2016-11-14 |
| AU2010233122B2 (en) | 2015-09-17 |
| MX341368B (es) | 2016-08-17 |
| CA2758300C (en) | 2017-07-25 |
| NZ596125A (en) | 2012-08-31 |
| WO2010118390A1 (en) | 2010-10-14 |
| CN102612365A (zh) | 2012-07-25 |
| EP2416773A1 (en) | 2012-02-15 |
| EP2416773B1 (en) | 2016-09-28 |
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