RU2549899C2 - Кристаллические формы гидрохлорида финголимода - Google Patents
Кристаллические формы гидрохлорида финголимода Download PDFInfo
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- RU2549899C2 RU2549899C2 RU2011123371/04A RU2011123371A RU2549899C2 RU 2549899 C2 RU2549899 C2 RU 2549899C2 RU 2011123371/04 A RU2011123371/04 A RU 2011123371/04A RU 2011123371 A RU2011123371 A RU 2011123371A RU 2549899 C2 RU2549899 C2 RU 2549899C2
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Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2627691C1 (ru) * | 2016-07-06 | 2017-08-10 | Олег Ростиславович Михайлов | Кристаллическая η-модификация 2-амино-2-(2-(4-октилфенил)этил)пропан-1,3-диол гидрохлорида, способ её получения и фармацевтическая композиция на её основе |
| RU2663833C2 (ru) * | 2013-03-05 | 2018-08-10 | Биокон Лимитед | Способ получения соединений 2-амино-1,3-пропандиола и их солей |
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| WO2012041358A1 (en) | 2010-10-01 | 2012-04-05 | Synthon B.V. | Process for making fingolimod hydrochloride crystals |
| ES2697605T3 (es) | 2010-10-28 | 2019-01-25 | Mapi Pharma Ltd | Compuesto intermedios y proceso para la preparación de fingolimod |
| WO2012071524A1 (en) | 2010-11-24 | 2012-05-31 | Ratiopharm Gmbh | Arylsulfonate salts of fingolimod and processes for preparation thereof |
| US9266816B2 (en) | 2010-11-25 | 2016-02-23 | Shilpa Medicare Limited | Fingolimod polymorphs and their processes |
| WO2012089238A1 (en) | 2010-12-28 | 2012-07-05 | Synthon Bv | Process for making fingolimod hydrochloride crystals |
| WO2012097330A2 (en) * | 2011-01-14 | 2012-07-19 | University Of Washington | Compositions and methods for treating degenerative muscle conditions |
| US9216943B2 (en) | 2011-04-29 | 2015-12-22 | Dr. Reddy's Laboratories Ltd. | Preparation of fingolimod and its salts |
| EP2809648B1 (en) | 2011-05-26 | 2019-04-03 | GRI Bio, Inc. | Oxygenated amino- or ammonium-containing sulfonic acid derivatives and their medical use |
| US9850265B2 (en) | 2011-05-26 | 2017-12-26 | Gri Bio, Inc. | Amino- or ammonium-containing sulfonic acid, phosphonic acid and carboxylic acid derivatives and their medical use |
| CA2887385C (en) | 2011-05-26 | 2017-01-10 | Glycoregimmune, Inc. Carrying On Business As Gri Bio, Inc. | Hydroxy-substituted amino and ammonium derivatives and their medical use |
| EA028950B1 (ru) | 2011-08-01 | 2018-01-31 | Тева Фармасьютикал Индастриз Лтд. | Способ получения фармацевтических композиций, содержащих финголимод |
| WO2013091704A1 (en) * | 2011-12-22 | 2013-06-27 | Synthon Bv | Pharmaceutical composition comprising fingolimod |
| CN102887829B (zh) * | 2012-09-05 | 2014-07-02 | 中国科学院上海药物研究所 | 芬戈莫德粘酸盐及其晶体的制备方法和用途 |
| AU2014206588A1 (en) * | 2013-01-17 | 2015-07-23 | Shilpa Medicare Limited | Process for preparation of Fingolimod and its salts |
| CA2920758A1 (en) | 2013-07-29 | 2015-02-05 | Aizant Drug Research Solutions Pvt Ltd | Pharmaceutical compositions of fingolimod |
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| RU2663833C2 (ru) * | 2013-03-05 | 2018-08-10 | Биокон Лимитед | Способ получения соединений 2-амино-1,3-пропандиола и их солей |
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Also Published As
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|---|---|
| RU2011123371A (ru) | 2012-12-20 |
| KR20110069156A (ko) | 2011-06-22 |
| JP2018035160A (ja) | 2018-03-08 |
| US20110229501A1 (en) | 2011-09-22 |
| CN102209705A (zh) | 2011-10-05 |
| RU2015111229A3 (enExample) | 2018-11-08 |
| WO2010055028A3 (en) | 2010-07-08 |
| EP2356090B1 (en) | 2017-07-05 |
| PL2356090T3 (pl) | 2017-12-29 |
| PT2356090T (pt) | 2017-10-16 |
| US20140051766A1 (en) | 2014-02-20 |
| JP2016028056A (ja) | 2016-02-25 |
| KR20130109254A (ko) | 2013-10-07 |
| BRPI0921826A2 (pt) | 2016-01-12 |
| RU2015111229A (ru) | 2015-11-20 |
| MX2011004962A (es) | 2011-05-30 |
| AU2009315736B2 (en) | 2013-08-29 |
| EP2356090A2 (en) | 2011-08-17 |
| KR101393994B1 (ko) | 2014-05-14 |
| JP2012508216A (ja) | 2012-04-05 |
| WO2010055028A2 (en) | 2010-05-20 |
| CA2743232C (en) | 2015-12-29 |
| ES2643161T3 (es) | 2017-11-21 |
| CN107233336A (zh) | 2017-10-10 |
| US8530522B2 (en) | 2013-09-10 |
| CA2743232A1 (en) | 2010-05-20 |
| CN104788325A (zh) | 2015-07-22 |
| AU2009315736A1 (en) | 2010-05-20 |
| JP2014139179A (ja) | 2014-07-31 |
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