RU2455996C2 - Новая парентеральная композиция карбамазепина - Google Patents
Новая парентеральная композиция карбамазепина Download PDFInfo
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- RU2455996C2 RU2455996C2 RU2008117161/15A RU2008117161A RU2455996C2 RU 2455996 C2 RU2455996 C2 RU 2455996C2 RU 2008117161/15 A RU2008117161/15 A RU 2008117161/15A RU 2008117161 A RU2008117161 A RU 2008117161A RU 2455996 C2 RU2455996 C2 RU 2455996C2
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- carbamazepine
- cyclodextrin
- cbz
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- C08B—POLYSACCHARIDES; DERIVATIVES THEREOF
- C08B37/00—Preparation of polysaccharides not provided for in groups C08B1/00 - C08B35/00; Derivatives thereof
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- C08B37/0009—Homoglycans, i.e. polysaccharides having a main chain consisting of one single sugar, e.g. colominic acid alpha-D-Glucans, e.g. polydextrose, alternan, glycogen; (alpha-1,4)(alpha-1,6)-D-Glucans; (alpha-1,3)(alpha-1,4)-D-Glucans, e.g. isolichenan or nigeran; (alpha-1,4)-D-Glucans; (alpha-1,3)-D-Glucans, e.g. pseudonigeran; Derivatives thereof
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| Publication number | Priority date | Publication date | Assignee | Title |
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| US20100204178A1 (en) | 2006-10-02 | 2010-08-12 | James Cloyd | Novel parenteral carbamazepine formulation |
| RU2464042C1 (ru) * | 2011-03-31 | 2012-10-20 | Общество С Ограниченной Ответственностью "Научно-Исследовательская Компания "Медбиофарм" | КЛАТРАТНЫЙ КОМПЛЕКС β-ЦИКЛОДЕКСТРИНА С ПРОИЗВОДНЫМ 5-ГИДРОКСИ-4-АМИНОМЕТИЛ-1-ЦИКЛОГЕКСИЛ(ИЛИ ЦИКЛОГЕПТИЛ)-3-АЛКОКСИКАРБОНИЛИНДОЛА, СПОСОБ ЕГО ПОЛУЧЕНИЯ (ВАРИАНТЫ), ФАРМАЦЕВТИЧЕСКАЯ КОМПОЗИЦИЯ И ЛЕКАРСТВЕННОЕ СРЕДСТВО |
| US20140178479A1 (en) | 2011-08-12 | 2014-06-26 | Perosphere, Inc. | Concentrated Felbamate Formulations for Parenteral Administration |
| US11235020B2 (en) * | 2013-03-13 | 2022-02-01 | Abraham Palmer | Methods and compositions for inhibiting glyoxalase 1 (GLO1) |
| CN105726466A (zh) * | 2014-12-10 | 2016-07-06 | 辽宁药联制药有限公司 | 一种奥卡西平注射剂及其制备方法 |
| MY200159A (en) * | 2016-12-14 | 2023-12-09 | Sk Biopharmaceuticals Co Ltd | Parenteral liquid preparation comprising carbamate compound |
| WO2020157257A1 (en) * | 2019-02-01 | 2020-08-06 | H. Lundbeck A/S | Injectable carbamazepine composition essentially free of 10-br-carbamazepine |
| US12383633B1 (en) | 2024-10-01 | 2025-08-12 | Zymeron Corporation | Injectable formulations of PARP inhibitors and uses thereof |
| CN120754274A (zh) * | 2025-07-15 | 2025-10-10 | 江苏鹏鹞药业有限公司 | 一种卡马西平的生产工艺及负载分散剂 |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5134127A (en) * | 1990-01-23 | 1992-07-28 | University Of Kansas | Derivatives of cyclodextrins exhibiting enhanced aqueous solubility and the use thereof |
| US5646131A (en) * | 1994-02-22 | 1997-07-08 | The Arab Company For Drug Industries And Medical Applicances (Acdima) | Method for solubilizing drugs using cyclodextrins and carboxylic acids |
| US6458770B1 (en) * | 1997-10-09 | 2002-10-01 | Novartis Ag | Parenteral formulations comprising carbamazepine or its derivatives |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3459731A (en) | 1966-12-16 | 1969-08-05 | Corn Products Co | Cyclodextrin polyethers and their production |
| US5231098A (en) * | 1987-06-26 | 1993-07-27 | Nihon Bayer Agrochem K.K. | Insecticidal nitro-substituted heterocyclic compounds |
| US5376645A (en) | 1990-01-23 | 1994-12-27 | University Of Kansas | Derivatives of cyclodextrins exhibiting enhanced aqueous solubility and the use thereof |
| US6546131B1 (en) | 1990-12-19 | 2003-04-08 | Canon Kabushiki Kaisha | Image processing method and apparatus for achieving tone reproduction suited to the image |
| US5231089A (en) * | 1991-12-02 | 1993-07-27 | University Of Florida | Method of improving oral bioavailability of carbamazepine |
| FR2713934B1 (fr) | 1993-12-22 | 1996-01-12 | Commissariat Energie Atomique | Utilisation de cyclodextrines aminées pour la solubilisation aqueuse de composés hydrophobes, en particulier de molécules pharmaceutiquement actives. |
| US6046177A (en) * | 1997-05-05 | 2000-04-04 | Cydex, Inc. | Sulfoalkyl ether cyclodextrin based controlled release solid pharmaceutical formulations |
| AU772204B2 (en) | 1999-01-21 | 2004-04-22 | Bristol-Myers Squibb Company | Complex of ras-farnesyltransferase inhibitor and sulfobutylether-7-beta-cyclodextrin or 2-hydroxypropyl-beta-cyclodextrin and method |
| KR20030041577A (ko) * | 2001-11-20 | 2003-05-27 | 디디에스텍주식회사 | 난용성 약물과 치환된 시클로덱스트린을 함유하는고체분산체 및 이를 함유하는 약제학적 조성물 |
| JP2006509788A (ja) | 2002-11-27 | 2006-03-23 | ファルマシア・コーポレーション | バルデコキシブの濃縮液体組成物 |
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Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5134127A (en) * | 1990-01-23 | 1992-07-28 | University Of Kansas | Derivatives of cyclodextrins exhibiting enhanced aqueous solubility and the use thereof |
| US5646131A (en) * | 1994-02-22 | 1997-07-08 | The Arab Company For Drug Industries And Medical Applicances (Acdima) | Method for solubilizing drugs using cyclodextrins and carboxylic acids |
| US6458770B1 (en) * | 1997-10-09 | 2002-10-01 | Novartis Ag | Parenteral formulations comprising carbamazepine or its derivatives |
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| Title |
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| Справочник «Видаль», 1998, с.Б-288. РЛС Аптекарь, 2003, с.512-514. * |
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| WO2007041524A3 (en) | 2007-09-13 |
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| CA2624463A1 (en) | 2007-04-12 |
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| ZA200803332B (en) | 2011-05-25 |
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| JP5284096B2 (ja) | 2013-09-11 |
| US20240165125A1 (en) | 2024-05-23 |
| CY1115517T1 (el) | 2017-01-04 |
| ES2475157T3 (es) | 2014-07-10 |
| EP1928464A2 (en) | 2008-06-11 |
| RU2008117161A (ru) | 2009-11-10 |
| SI1928464T1 (sl) | 2014-09-30 |
| NZ567290A (en) | 2011-08-26 |
| BRPI0616447A2 (pt) | 2011-06-21 |
| AU2006299501B2 (en) | 2012-11-29 |
| CA2624463C (en) | 2017-02-14 |
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| EP2444090B1 (en) | 2018-12-12 |
| JP2009510123A (ja) | 2009-03-12 |
| MX2008004287A (es) | 2008-10-23 |
| PT1928464E (pt) | 2014-07-10 |
| EP1928464A4 (en) | 2009-10-21 |
| CN101309691A (zh) | 2008-11-19 |
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