RU2019122355A - Полиморфы - Google Patents
Полиморфы Download PDFInfo
- Publication number
- RU2019122355A RU2019122355A RU2019122355A RU2019122355A RU2019122355A RU 2019122355 A RU2019122355 A RU 2019122355A RU 2019122355 A RU2019122355 A RU 2019122355A RU 2019122355 A RU2019122355 A RU 2019122355A RU 2019122355 A RU2019122355 A RU 2019122355A
- Authority
- RU
- Russia
- Prior art keywords
- composition
- crystalline polymorph
- agriculture
- propagation material
- plant propagation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/10—Spiro-condensed systems
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
- A01N25/12—Powders or granules
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Claims (8)
1. Кристаллический полиморф соединения формулы I,
который характеризуется порошковой дифракционной рентгенограммой, содержащей одно значение угла 2θ, составляющее 13,7±0,2, и по меньшей мере три значения угла 2θ, выбранные из группы, состоящей из 7,7±0,2, 12,6±0,2, 13,9±0,2, 15,3±0,2, 16,0±0,2, 17,4±0,2, 23,1±0,2 и 23,8±0,2.
3. Кристаллический полиморф по п. 1 или 2, который характеризуется температурой плавления 125°С±2°С.
4. Композиция для использования в сельском хозяйстве, содержащая полиморф по любому из пп. 1-3 и по меньшей мере один приемлемый с точки зрения сельского хозяйства носитель или разбавитель.
5. Композиция по п. 4, которая содержит по меньшей мере один дополнительный инсектицид или нематоцид.
6. Способ предупреждения или осуществления контроля инфекции растений или материала для размножения растений насекомыми, включающий обработку растения или материала для размножения растений инсектицидно эффективным количеством композиции для использования в сельском хозяйстве по п. 4 или 5.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB1622007.1A GB201622007D0 (en) | 2016-12-22 | 2016-12-22 | Polymorphs |
GB1622007.1 | 2016-12-22 | ||
PCT/EP2017/082984 WO2018114649A1 (en) | 2016-12-22 | 2017-12-15 | Polymorphs |
Publications (2)
Publication Number | Publication Date |
---|---|
RU2019122355A true RU2019122355A (ru) | 2021-01-22 |
RU2019122355A3 RU2019122355A3 (ru) | 2021-04-13 |
Family
ID=58360566
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
RU2019122355A RU2019122355A (ru) | 2016-12-22 | 2017-12-15 | Полиморфы |
Country Status (29)
Country | Link |
---|---|
US (2) | US11001584B2 (ru) |
EP (1) | EP3558995B1 (ru) |
JP (1) | JP2020504116A (ru) |
KR (1) | KR102565863B1 (ru) |
CN (1) | CN110099903A (ru) |
AU (1) | AU2017379297B2 (ru) |
BR (1) | BR112019012561B1 (ru) |
CA (1) | CA3047053A1 (ru) |
CL (1) | CL2019001736A1 (ru) |
CO (1) | CO2019006673A2 (ru) |
DK (1) | DK3558995T3 (ru) |
ES (1) | ES2958516T3 (ru) |
GB (1) | GB201622007D0 (ru) |
HR (1) | HRP20231137T1 (ru) |
HU (1) | HUE063269T2 (ru) |
IL (1) | IL267530B (ru) |
LT (1) | LT3558995T (ru) |
MA (1) | MA47085B1 (ru) |
MX (1) | MX2019007336A (ru) |
PH (1) | PH12019501359A1 (ru) |
PL (1) | PL3558995T3 (ru) |
PT (1) | PT3558995T (ru) |
RS (1) | RS64684B1 (ru) |
RU (1) | RU2019122355A (ru) |
SI (1) | SI3558995T1 (ru) |
TW (1) | TWI734881B (ru) |
UA (1) | UA124166C2 (ru) |
WO (1) | WO2018114649A1 (ru) |
ZA (1) | ZA201903936B (ru) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2014187847A1 (en) * | 2013-05-23 | 2014-11-27 | Syngenta Participations Ag | Tank-mix formulations |
MA47081B1 (fr) * | 2016-12-22 | 2021-04-30 | Syngenta Participations Ag | Polymorphes |
GB201622007D0 (en) * | 2016-12-22 | 2017-02-08 | And See Cambridge Display Tech Ltd Syngenta Participations Ag | Polymorphs |
JP2022521732A (ja) | 2019-02-20 | 2022-04-12 | シンジェンタ クロップ プロテクション アクチェンゲゼルシャフト | スピロピジオンの使用 |
MA55589A (fr) | 2019-04-10 | 2022-02-16 | Syngenta Crop Protection Ag | Compositions pesticides |
TW202231187A (zh) | 2020-11-27 | 2022-08-16 | 瑞士商先正達農作物保護公司 | 殺有害生物組成物 |
AR125089A1 (es) | 2021-03-19 | 2023-06-07 | Syngenta Crop Protection Ag | Composiciones plaguicidas |
CN117794372A (zh) | 2021-08-20 | 2024-03-29 | 先正达农作物保护股份公司 | 控制茶树上的有害生物的方法 |
WO2023094286A1 (en) | 2021-11-25 | 2023-06-01 | Syngenta Crop Protection Ag | Pesticidal compositions |
WO2023222723A1 (en) | 2022-05-20 | 2023-11-23 | Syngenta Crop Protection Ag | Pesticidal compositions |
Family Cites Families (36)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6627646B2 (en) * | 2001-07-17 | 2003-09-30 | Sepracor Inc. | Norastemizole polymorphs |
ES2388548T3 (es) | 2005-04-08 | 2012-10-16 | Bayer Cropscience Nv | Suceso de élite A2704-12 y métodos y estuches para identificar a dicho suceso en muestras biológicas |
DK1871901T3 (da) | 2005-04-11 | 2011-10-17 | Bayer Bioscience Nv | Elitebegivenhed A5547-127 samt fremgangsmåder og sæt til identifikation af en sådan begivenhed i biologiske prøver |
AP2693A (en) | 2005-05-27 | 2013-07-16 | Monsanto Technology Llc | Soybean event MON89788 and methods for detection thereof |
KR20080077650A (ko) * | 2005-12-14 | 2008-08-25 | 마켓심 케미칼 웍스 리미티드 | 5-아미노-1-[2,6-디클로로-4-(트리플루오로메틸)페닐]-4-[(트리플루오로메틸)설피닐]-1h-피라졸-s-카르보니트릴의다형체 및 무정형 |
US7951995B2 (en) | 2006-06-28 | 2011-05-31 | Pioneer Hi-Bred International, Inc. | Soybean event 3560.4.3.5 and compositions and methods for the identification and detection thereof |
BRPI0716347B8 (pt) | 2006-10-31 | 2022-12-06 | Du Pont | Polinuleotídeo isolado, métodos para identificar se uma amostra biológica compreende um polinucleotídeo, para detectar a presença de um polinucleotídeo, para detectar a presença de uma sequência, para selecionar sementes e para produzir um vegetal tolerante ao inibidor de als, pares de primers de dna e construção de um dna de expressão |
AU2008321220A1 (en) | 2007-11-15 | 2009-05-22 | Monsanto Technology Llc | Soybean plant and seed corresponding to transgenic event MON87701 and methods for detection thereof |
CN102245028B (zh) | 2008-12-12 | 2014-12-31 | 先正达参股股份有限公司 | 用作农药的螺杂环n-氧基哌啶 |
CA2748973A1 (en) | 2009-01-07 | 2010-07-15 | Basf Agrochemical Products B.V. | Soybean event 127 and methods related thereto |
CA2771543C (en) | 2009-08-19 | 2018-05-15 | Dow Agrosciences Llc | Control of aad-1 monocot volunteers in fields of dicot crops |
AU2010284286B2 (en) | 2009-08-19 | 2015-08-20 | Dow Agrosciences Llc | Detection of AAD-1 event DAS-40278-9 |
JP2013526832A (ja) | 2009-08-19 | 2013-06-27 | ダウ アグロサイエンシィズ エルエルシー | Aad−1イベントdas−40278−9、関連するトランスジェニックトウモロコシ系統およびそのイベント特異的同定 |
ES2866126T3 (es) | 2009-09-17 | 2021-10-19 | Monsanto Technology Llc | Evento transgénico de soja MON 87708 y procedimientos de uso del mismo |
KR20130080485A (ko) * | 2010-05-31 | 2013-07-12 | 신젠타 파티서페이션즈 아게 | 작물 강화 방법 |
ES2642789T3 (es) * | 2010-05-31 | 2017-11-20 | Syngenta Participations Ag | Método de control de hemípteros resistentes a neonicotinoides usando derivados de pirrolidindiona espiroheterocíclicos |
TW201208573A (en) * | 2010-05-31 | 2012-03-01 | Syngenta Participations Ag | Pesticidal compositions |
CA2798320A1 (en) | 2010-05-31 | 2011-12-08 | Syngenta Participations Ag | Pesticidal compositions |
TWI667347B (zh) | 2010-12-15 | 2019-08-01 | 瑞士商先正達合夥公司 | 大豆品種syht0h2及偵測其之組合物及方法 |
BR102012019436B8 (pt) | 2011-07-26 | 2022-10-11 | Dow Agrosciences Llc | Método de detecção do evento de soja pdab9582.814.19.1 |
KR20140064849A (ko) | 2011-08-12 | 2014-05-28 | 바스프 에스이 | 아닐린 유형 화합물 |
TWI572282B (zh) | 2011-11-30 | 2017-03-01 | 先正達合夥公司 | 含有螺雜環吡咯啶二酮的殺有害生物混合物 |
EP3476219B1 (en) | 2012-01-17 | 2023-08-30 | Syngenta Participations AG | Pesticidal mixtures including spiroheterocyclic pyrrolidine diones |
IN2014DN05859A (ru) | 2012-01-17 | 2015-05-22 | Syngenta Participations Ag | |
WO2013107794A2 (en) | 2012-01-17 | 2013-07-25 | Syngenta Participations Ag | Pesticidal mixtures including spiroheterocyclic pyrrolidine diones |
DK3222144T3 (da) | 2012-01-17 | 2019-09-30 | Syngenta Participations Ag | Pesticidblandinger, der indbefatter spiroheterocykliske pyrrolidindioner |
GB201202393D0 (en) * | 2012-02-09 | 2012-03-28 | Syngenta Ltd | Polymorphs |
JPWO2014126208A1 (ja) * | 2013-02-14 | 2017-02-02 | 日産化学工業株式会社 | イソキサゾリン置換ベンズアミド化合物の結晶性多形体及びその製造方法 |
WO2014170327A1 (en) | 2013-04-19 | 2014-10-23 | Bayer Cropscience Ag | Method for combating pests |
CN105228448B (zh) * | 2013-05-23 | 2019-03-01 | 先正达参股股份有限公司 | 桶混配制品 |
WO2014187847A1 (en) | 2013-05-23 | 2014-11-27 | Syngenta Participations Ag | Tank-mix formulations |
WO2014191271A1 (en) | 2013-05-28 | 2014-12-04 | Syngenta Participations Ag | Use of tetramic acid derivatives as nematicides |
EA036941B1 (ru) | 2013-06-14 | 2021-01-18 | Монсанто Текнолоджи Ллс | Трансгенный объект сои mon87751 и способы его определения и применения |
JP2015028006A (ja) * | 2013-06-27 | 2015-02-12 | 日産化学工業株式会社 | イソキサゾリン化合物の結晶性多形体およびその製造方法 |
BR112016001001B1 (pt) | 2013-07-19 | 2020-11-17 | Syngenta Participations Ag | processo para a preparação de pirrolidinas dionas espiroheterocíclicas, processo para preparação de composto e composto |
GB201622007D0 (en) * | 2016-12-22 | 2017-02-08 | And See Cambridge Display Tech Ltd Syngenta Participations Ag | Polymorphs |
-
2016
- 2016-12-22 GB GBGB1622007.1A patent/GB201622007D0/en not_active Ceased
-
2017
- 2017-12-15 DK DK17828694.4T patent/DK3558995T3/da active
- 2017-12-15 RU RU2019122355A patent/RU2019122355A/ru unknown
- 2017-12-15 CA CA3047053A patent/CA3047053A1/en active Pending
- 2017-12-15 RS RS20230824A patent/RS64684B1/sr unknown
- 2017-12-15 LT LTEPPCT/EP2017/082984T patent/LT3558995T/lt unknown
- 2017-12-15 WO PCT/EP2017/082984 patent/WO2018114649A1/en active Application Filing
- 2017-12-15 PL PL17828694.4T patent/PL3558995T3/pl unknown
- 2017-12-15 JP JP2019534394A patent/JP2020504116A/ja active Pending
- 2017-12-15 EP EP17828694.4A patent/EP3558995B1/en active Active
- 2017-12-15 BR BR112019012561-2A patent/BR112019012561B1/pt active IP Right Grant
- 2017-12-15 US US16/472,608 patent/US11001584B2/en active Active
- 2017-12-15 UA UAA201908008A patent/UA124166C2/uk unknown
- 2017-12-15 MX MX2019007336A patent/MX2019007336A/es unknown
- 2017-12-15 AU AU2017379297A patent/AU2017379297B2/en active Active
- 2017-12-15 ES ES17828694T patent/ES2958516T3/es active Active
- 2017-12-15 PT PT178286944T patent/PT3558995T/pt unknown
- 2017-12-15 KR KR1020197019609A patent/KR102565863B1/ko active IP Right Grant
- 2017-12-15 CN CN201780079579.7A patent/CN110099903A/zh active Pending
- 2017-12-15 SI SI201731417T patent/SI3558995T1/sl unknown
- 2017-12-15 HR HRP20231137TT patent/HRP20231137T1/hr unknown
- 2017-12-15 HU HUE17828694A patent/HUE063269T2/hu unknown
- 2017-12-15 MA MA47085A patent/MA47085B1/fr unknown
- 2017-12-21 TW TW106145068A patent/TWI734881B/zh active
-
2019
- 2019-06-14 PH PH12019501359A patent/PH12019501359A1/en unknown
- 2019-06-18 ZA ZA2019/03936A patent/ZA201903936B/en unknown
- 2019-06-19 IL IL267530A patent/IL267530B/en unknown
- 2019-06-20 CL CL2019001736A patent/CL2019001736A1/es unknown
- 2019-06-21 CO CONC2019/0006673A patent/CO2019006673A2/es unknown
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2021
- 2021-05-10 US US17/315,538 patent/US20210261550A1/en active Pending
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