RU2016149319A3 - - Google Patents

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Publication number
RU2016149319A3
RU2016149319A3 RU2016149319A RU2016149319A RU2016149319A3 RU 2016149319 A3 RU2016149319 A3 RU 2016149319A3 RU 2016149319 A RU2016149319 A RU 2016149319A RU 2016149319 A RU2016149319 A RU 2016149319A RU 2016149319 A3 RU2016149319 A3 RU 2016149319A3
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RU
Russia
Application number
RU2016149319A
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RU2016149319A (ru
RU2658008C2 (ru
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
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Publication of RU2016149319A publication Critical patent/RU2016149319A/ru
Publication of RU2016149319A3 publication Critical patent/RU2016149319A3/ru
Application granted granted Critical
Publication of RU2658008C2 publication Critical patent/RU2658008C2/ru

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D519/00Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
RU2016149319A 2014-06-24 2015-06-24 Новое пирролопиримидиновое соединение или его соль, фармацевтическая композиция, содержащая ее, в частности, агент для предотвращения и/или лечения опухолей, и тому подобное, на основе ингибиторного воздействия на nae RU2658008C2 (ru)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
JP2014-129740 2014-06-24
JP2014129740 2014-06-24
JP2015024785 2015-02-10
JP2015-024785 2015-02-10
PCT/JP2015/068218 WO2015199136A1 (ja) 2014-06-24 2015-06-24 新規ピロロピリミジン化合物又はその塩、及びこれを含有する医薬組成物、特にnae阻害作用に基づく腫瘍等の予防剤及び/又は治療剤

Publications (3)

Publication Number Publication Date
RU2016149319A RU2016149319A (ru) 2018-06-18
RU2016149319A3 true RU2016149319A3 (ru) 2018-06-18
RU2658008C2 RU2658008C2 (ru) 2018-06-19

Family

ID=54938214

Family Applications (1)

Application Number Title Priority Date Filing Date
RU2016149319A RU2658008C2 (ru) 2014-06-24 2015-06-24 Новое пирролопиримидиновое соединение или его соль, фармацевтическая композиция, содержащая ее, в частности, агент для предотвращения и/или лечения опухолей, и тому подобное, на основе ингибиторного воздействия на nae

Country Status (21)

Country Link
US (2) US9963456B2 (ru)
EP (1) EP3103802B1 (ru)
JP (1) JP6192741B2 (ru)
KR (1) KR101947289B1 (ru)
CN (1) CN106661031B (ru)
AU (1) AU2015281155B9 (ru)
BR (1) BR112016025835B1 (ru)
CA (1) CA2946833C (ru)
DK (1) DK3103802T3 (ru)
ES (1) ES2656772T3 (ru)
HU (1) HUE037266T2 (ru)
MX (1) MX2016015015A (ru)
MY (1) MY183327A (ru)
NO (1) NO3103802T3 (ru)
PH (1) PH12016502130A1 (ru)
PL (1) PL3103802T3 (ru)
PT (1) PT3103802T (ru)
RU (1) RU2658008C2 (ru)
SG (1) SG11201608441YA (ru)
TW (1) TWI605048B (ru)
WO (1) WO2015199136A1 (ru)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI623316B (zh) * 2015-12-22 2018-05-11 Taiho Pharmaceutical Co Ltd Antitumor effect enhancer derived from pyrrolopyrimidine compound
WO2018085818A1 (en) * 2016-11-07 2018-05-11 Prelude Therapeutics, Incorporated Selective inhibitors of protein arginine methyltransferase 5 (prmt5)
WO2018085833A2 (en) * 2016-11-07 2018-05-11 Prelude Therapeutics, Incorporated Selective inhibitors of protein arginine methyl transferase 5 (prmt5)
US10865208B2 (en) 2016-11-11 2020-12-15 Millennium Pharmaceuticals, Inc. ATG7 inhibitors and the uses thereof
WO2018110591A1 (ja) * 2016-12-13 2018-06-21 ヤマサ醤油株式会社 抗ウイルス活性を有する2'-デオキシ-7-デアザプリンヌクレオシド誘導体
JP7060694B2 (ja) * 2018-01-18 2022-04-26 アレイ バイオファーマ インコーポレイテッド Retキナーゼ阻害剤としての置換ピロロ[2,3-d]ピリミジン化合物
CN108640945B (zh) * 2018-06-11 2020-10-23 广东工业大学 一种酰胺类化合物及其制备方法与应用
CN108822145B (zh) * 2018-06-11 2020-10-23 广东工业大学 一种磺酰胺类化合物及其制备方法和应用
EP3820533A2 (en) * 2018-07-13 2021-05-19 IL-2RX, Inc. Compounds, compositions, methods, and uses for treating cancer and immunological disorders

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL1848718T3 (pl) * 2005-02-04 2012-12-31 Millennium Pharm Inc Inhibitory enzymów hamujących E1
EP1960518A2 (en) * 2005-12-06 2008-08-27 Regents Of The University Of Minnesota Antibacterial agents
PT1989206E (pt) 2006-02-02 2012-10-15 Millennium Pharm Inc Inibidores da enzima de ativação e1
US20120115892A1 (en) 2010-11-05 2012-05-10 Millennium Pharmaceuticals, Inc. Administration of nedd8-activating enzyme inhibitor
EP2661436B1 (en) 2011-01-07 2016-04-13 Leo Pharma A/S Novel sulfamide piperazine derivatives as protein tyrosine kinase inhibitors and pharmaceutical use thereof
WO2013016906A1 (zh) * 2011-07-29 2013-02-07 深圳光启高等理工研究院 人工复合材料和人工复合材料天线
PT2657233E (pt) 2012-01-19 2014-10-24 Taiho Pharmaceutical Co Ltd Composto de alcinil-benzeno substituído nas posições 3 e 5 e um seu sal

Also Published As

Publication number Publication date
BR112016025835B1 (pt) 2022-09-20
RU2016149319A (ru) 2018-06-18
WO2015199136A1 (ja) 2015-12-30
BR112016025835A2 (ru) 2017-08-15
US9963456B2 (en) 2018-05-08
CA2946833C (en) 2019-03-05
NO3103802T3 (ru) 2018-04-07
PH12016502130B1 (en) 2016-12-19
US20170066772A1 (en) 2017-03-09
MX2016015015A (es) 2017-02-27
JP6192741B2 (ja) 2017-09-06
TW201625629A (zh) 2016-07-16
AU2015281155A1 (en) 2016-11-03
PL3103802T3 (pl) 2018-02-28
CA2946833A1 (en) 2015-12-30
CN106661031B (zh) 2019-07-23
JPWO2015199136A1 (ja) 2017-04-27
US10174040B2 (en) 2019-01-08
AU2015281155B9 (en) 2017-11-16
SG11201608441YA (en) 2016-11-29
AU2015281155B2 (en) 2017-07-13
PT3103802T (pt) 2017-12-11
EP3103802A4 (en) 2017-03-08
RU2658008C2 (ru) 2018-06-19
KR101947289B1 (ko) 2019-02-12
KR20170016510A (ko) 2017-02-13
PH12016502130A1 (en) 2016-12-19
CN106661031A (zh) 2017-05-10
MY183327A (en) 2021-02-18
TWI605048B (zh) 2017-11-11
EP3103802B1 (en) 2017-11-08
DK3103802T3 (en) 2017-12-11
HUE037266T2 (hu) 2018-08-28
US20180162864A1 (en) 2018-06-14
EP3103802A1 (en) 2016-12-14
ES2656772T3 (es) 2018-02-28

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