RS59110B1 - Heteroarilni sik inhibitori - Google Patents

Heteroarilni sik inhibitori

Info

Publication number
RS59110B1
RS59110B1 RS20191047A RSP20191047A RS59110B1 RS 59110 B1 RS59110 B1 RS 59110B1 RS 20191047 A RS20191047 A RS 20191047A RS P20191047 A RSP20191047 A RS P20191047A RS 59110 B1 RS59110 B1 RS 59110B1
Authority
RS
Serbia
Prior art keywords
group
alkyl
het
formula
oxo
Prior art date
Application number
RS20191047A
Other languages
English (en)
Serbian (sr)
Inventor
Georg Dahmann
Matthias Hoffmann
Jasna Klicic
David James Lamb
Clive Mccarthy
Spencer Napier
Karen Parrish
John Scott
Fitzgerald Jennifer L Swantek
Edward Walker
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of RS59110B1 publication Critical patent/RS59110B1/sr

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/4162—1,2-Diazoles condensed with heterocyclic ring systems
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
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CN110713489B (zh) 2022-05-31
UA119667C2 (uk) 2019-07-25
PH12016501796A1 (en) 2016-11-21
AP2016009373A0 (en) 2016-08-31
UY36037A (es) 2015-09-30
JP2017511805A (ja) 2017-04-27
HUE046061T2 (hu) 2020-02-28
CN106255689A (zh) 2016-12-21
EP3119766B1 (en) 2019-05-22
JP2017512778A (ja) 2017-05-25
JP6416275B2 (ja) 2018-10-31
US10947243B2 (en) 2021-03-16

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