RS56570B1 - Kompozicije i metode za prevladavanje otpornosti na tramadol - Google Patents

Kompozicije i metode za prevladavanje otpornosti na tramadol

Info

Publication number
RS56570B1
RS56570B1 RS20171178A RSP20171178A RS56570B1 RS 56570 B1 RS56570 B1 RS 56570B1 RS 20171178 A RS20171178 A RS 20171178A RS P20171178 A RSP20171178 A RS P20171178A RS 56570 B1 RS56570 B1 RS 56570B1
Authority
RS
Serbia
Prior art keywords
tramadol
compositions
methods
overcoming resistance
overcoming
Prior art date
Application number
RS20171178A
Other languages
English (en)
Inventor
John A Zebala
Original Assignee
Syntrix Biosystems Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syntrix Biosystems Inc filed Critical Syntrix Biosystems Inc
Publication of RS56570B1 publication Critical patent/RS56570B1/sr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Child & Adolescent Psychology (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
RS20171178A 2011-07-09 2012-07-09 Kompozicije i metode za prevladavanje otpornosti na tramadol RS56570B1 (sr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161506092P 2011-07-09 2011-07-09
EP12810860.2A EP2729134B1 (en) 2011-07-09 2012-07-09 Compositions and methods for overcoming resistance to tramadol
PCT/US2012/045885 WO2013009666A1 (en) 2011-07-09 2012-07-09 Compositions and methods for overcoming resistance to tramadol

Publications (1)

Publication Number Publication Date
RS56570B1 true RS56570B1 (sr) 2018-02-28

Family

ID=47438792

Family Applications (1)

Application Number Title Priority Date Filing Date
RS20171178A RS56570B1 (sr) 2011-07-09 2012-07-09 Kompozicije i metode za prevladavanje otpornosti na tramadol

Country Status (14)

Country Link
US (6) US10702485B2 (sr)
EP (2) EP2729134B1 (sr)
CY (1) CY1119597T1 (sr)
DK (1) DK2729134T3 (sr)
ES (1) ES2650368T3 (sr)
HR (1) HRP20171743T1 (sr)
HU (1) HUE037341T2 (sr)
LT (1) LT2729134T (sr)
NO (1) NO2833973T3 (sr)
PL (1) PL2729134T3 (sr)
PT (1) PT2729134T (sr)
RS (1) RS56570B1 (sr)
SI (1) SI2729134T1 (sr)
WO (1) WO2013009666A1 (sr)

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US10702485B2 (en) * 2011-07-09 2020-07-07 Syntrix Biosystems Inc. Compositions and methods for overcoming resistance to tramadol
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DE102013009114A1 (de) * 2013-05-29 2014-12-04 Franz Gerstheimer Pharmazeutische Zusammensetzung zur Überwindung von Metabolisierungsproblemen
US9561232B2 (en) 2014-02-18 2017-02-07 Demerx, Inc. Low dose noribogaine for treating nicotine addiction and preventing relapse of nicotine use
US9591978B2 (en) 2014-03-13 2017-03-14 Demerx, Inc. Methods and compositions for pre-screening patients for treatment with noribogaine
EP2922348A1 (en) * 2014-03-21 2015-09-23 Alcatel Lucent Network configuration
US9549935B2 (en) 2014-07-14 2017-01-24 Demerx, Inc. Methods and compositions for treating migraines using noribogaine
EP3223906B1 (en) 2014-11-26 2021-01-06 DemeRx, Inc. Methods and compositions for potentiating the action of opioid analgesics using iboga alkaloids
CA3024081A1 (en) * 2015-05-11 2016-11-17 Demerx, Inc. Methods for treatment of opioid dependency and withdrawal using noribogaine
US11000488B2 (en) 2019-03-22 2021-05-11 Syntrix Biosystems Inc. Treating pain using desmetramadol
CN113861048A (zh) * 2020-06-30 2021-12-31 南京诺瑞特医药科技有限公司 去甲曲马多的盐及其用途

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Also Published As

Publication number Publication date
PT2729134T (pt) 2017-11-24
US20130011444A1 (en) 2013-01-10
US20170319510A1 (en) 2017-11-09
HRP20171743T1 (hr) 2017-12-29
US10702485B2 (en) 2020-07-07
ES2650368T3 (es) 2018-01-18
US20160220514A1 (en) 2016-08-04
LT2729134T (lt) 2017-10-10
PL2729134T3 (pl) 2018-01-31
CY1119597T1 (el) 2018-04-04
HUE037341T2 (hu) 2018-08-28
WO2013009666A1 (en) 2013-01-17
US9717700B2 (en) 2017-08-01
SI2729134T1 (sl) 2017-12-29
EP2729134B1 (en) 2017-08-23
US20160074341A1 (en) 2016-03-17
EP2729134A4 (en) 2015-03-04
EP2729134A1 (en) 2014-05-14
NO2833973T3 (sr) 2018-02-10
US9717701B2 (en) 2017-08-01
US20170319511A1 (en) 2017-11-09
DK2729134T3 (en) 2017-10-09
US20150342905A1 (en) 2015-12-03
US9808432B2 (en) 2017-11-07
EP3272339A1 (en) 2018-01-24

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