RS51260B - Transdermalni sistem za dostavu gestodena - Google Patents

Transdermalni sistem za dostavu gestodena

Info

Publication number
RS51260B
RS51260B RSP-2010/0202A RSP20100202A RS51260B RS 51260 B RS51260 B RS 51260B RS P20100202 A RSP20100202 A RS P20100202A RS 51260 B RS51260 B RS 51260B
Authority
RS
Serbia
Prior art keywords
gestodene
drug
containing layer
transdermal delivery
delivery system
Prior art date
Application number
RSP-2010/0202A
Other languages
English (en)
Inventor
Thomas Langguth
Stefan Dr. Bracht
Michael Prof. Dr. Dittgen
Petra Huber
Drik Schenk
Original Assignee
Bayer Schering Pharma Aktiengesellschaft
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34924031&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=RS51260(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Schering Pharma Aktiengesellschaft filed Critical Bayer Schering Pharma Aktiengesellschaft
Publication of RS51260B publication Critical patent/RS51260B/sr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/567Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in position 17 alpha, e.g. mestranol, norethandrolone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/70Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7038Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
    • A61K9/7046Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
    • A61K9/7053Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/70Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7038Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
    • A61K9/7046Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
    • A61K9/7053Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
    • A61K9/7061Polyacrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/70Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7038Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
    • A61K9/7076Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising ingredients of undetermined constitution or reaction products thereof, e.g. rosin or other plant resins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18Feminine contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Dermatology (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Endocrinology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Reproductive Health (AREA)
  • Diabetes (AREA)
  • Botany (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Steroid Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Kompozicija za transdermalnu dostavu, naznačena time, da obuhvata sloj koji sadrži lek, a koji obuhvata Gestoden ili neki njegov ester i kerijer koji je izabran iz grupe koja se sastoji od poliizobutilena, polibutena, poliizoprena, polistirena, stiren izopren stiren blok polimera, stiren butadien stiren blok polimera i njihovih mešavina, a gde sloj koji sadrži lek poseduje rastvorivost za pomenuti Gestoden od ne više od 3% težine samoga sloja koji sadrži lek i gde Gestoden ili neki njegov ester je prisutan u količini koja se kreće u rasponu među 0.5 i 3% težine samoga sloja koji sadrži lek.Prijava sadrži još 21 patentni zahtev.
RSP-2010/0202A 2003-12-12 2004-12-10 Transdermalni sistem za dostavu gestodena RS51260B (sr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP03078881 2003-12-12
EP04078365A EP1541137B1 (en) 2003-12-12 2004-12-10 Transdermal delivery system of gestodene

Publications (1)

Publication Number Publication Date
RS51260B true RS51260B (sr) 2010-12-31

Family

ID=34924031

Family Applications (2)

Application Number Title Priority Date Filing Date
YU20140050A RS53182B (sr) 2003-12-12 2004-12-10 Transdermalni sistem dostave hormona bez upotrebe pojačivača penetracije
RSP-2010/0202A RS51260B (sr) 2003-12-12 2004-12-10 Transdermalni sistem za dostavu gestodena

Family Applications Before (1)

Application Number Title Priority Date Filing Date
YU20140050A RS53182B (sr) 2003-12-12 2004-12-10 Transdermalni sistem dostave hormona bez upotrebe pojačivača penetracije

Country Status (24)

Country Link
EP (2) EP2138169B1 (sr)
CN (1) CN101843603B (sr)
AR (1) AR046762A1 (sr)
AT (1) ATE457168T1 (sr)
CR (1) CR8465A (sr)
CY (2) CY1110637T1 (sr)
DE (1) DE602004025444D1 (sr)
DK (2) DK2138169T3 (sr)
ES (2) ES2340925T3 (sr)
GT (1) GT200400262A (sr)
HK (2) HK1074801A1 (sr)
HN (1) HN2004000526A (sr)
HR (2) HRP20100254T1 (sr)
JO (1) JO2606B1 (sr)
ME (1) ME01069B (sr)
MY (2) MY144053A (sr)
PE (1) PE20051035A1 (sr)
PL (2) PL2138169T3 (sr)
PT (2) PT2138169E (sr)
RS (2) RS53182B (sr)
SI (2) SI1541137T1 (sr)
SV (1) SV2006001970A (sr)
TW (1) TWI257299B (sr)
UA (1) UA89766C2 (sr)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT1594483E (pt) 2003-02-21 2006-12-29 Schering Ag Penso transdérmico estável aos uv
US8668925B2 (en) 2003-12-12 2014-03-11 Bayer Intellectual Property Gmbh Transdermal delivery of hormones without the need of penetration enhancers
US8962013B2 (en) 2005-05-02 2015-02-24 Bayer Intellectual Property Gmbh Multi-layered transdermal system with triazine UV absorber
DE102005050729A1 (de) * 2005-10-19 2007-04-26 Schering Ag Verfahren zur präventiven bedarfsweisen hormonalen Kontrazeption
ES2795455T3 (es) 2008-10-08 2020-11-23 Agile Therapeutics Inc Suministro transdérmico
WO2010042607A1 (en) 2008-10-08 2010-04-15 Agile Therapeutics, Inc Transdermal delivery
WO2010042610A1 (en) 2008-10-08 2010-04-15 Agile Therapeutics, Inc. Transdermal delivery
EP2410859A4 (en) 2009-03-27 2013-03-13 Agile Therapeutics Inc TRANSDERMAL ADMINISTRATION
AU2015203180B2 (en) * 2010-09-06 2016-06-30 Bayer Intellectual Property Gmbh Transdermal therapeutic systems with crystallization-inhibiting protective film (release liner)
HUE031326T2 (hu) 2010-09-06 2017-07-28 Bayer Ip Gmbh Alacsony dózisú transzdermális tapaszok magas hatóanyagleadással
DE102010040299A1 (de) * 2010-09-06 2012-03-08 Bayer Schering Pharma Aktiengesellschaft Transdermale therapeutische Systeme mit kristallisationsinhibierender Schutzfolie (Release Liner)
MX2014008693A (es) * 2012-01-27 2014-08-27 Agile Therapeutics Inc Administracion transdermica de hormonas.

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4081537A (en) 1975-10-10 1978-03-28 Schering Aktiengesellschaft Δ15 -Steroids and pharmaceutical compositions thereof
EP0394429B1 (de) * 1988-10-27 1996-01-10 Schering Aktiengesellschaft Mittel zur transdermalen applikation enthaltend gestoden
US5512292A (en) * 1990-10-29 1996-04-30 Alza Corporation Transdermal contraceptive formulations methods and devices
MX9101787A (es) * 1990-10-29 1992-06-05 Alza Corp Formulaciones,metodos y dispositivos anticonceptivos transdermicos
DE4336557C2 (de) 1993-05-06 1997-07-17 Lohmann Therapie Syst Lts Estradiolhaltiges transdermales therapeutisches System, Verfahren zu seiner Herstellung und seine Verwendung
DE4329242A1 (de) 1993-08-26 1995-03-02 Schering Ag Mittel zur transdermalen Applikation enthaltend Gestodenester
DE4405898A1 (de) * 1994-02-18 1995-08-24 Schering Ag Transdermale therapeutische Systeme enthaltend Sexualsteroide
US5762956A (en) 1996-04-24 1998-06-09 Rutgers, The State University Of New Jersey Transdermal contraceptive delivery system and process
DE19906152B4 (de) * 1999-02-10 2005-02-10 Jenapharm Gmbh & Co. Kg Wirkstoffhaltige Laminate für Transdermalsysteme
ES2338860T3 (es) 1999-11-24 2010-05-13 Agile Therapeutics, Inc. Sistema y procedimiento de administracion de anticonceptivos transdermica mejorado.
DE10053375C1 (de) * 2000-10-27 2002-01-24 Lohmann Therapie Syst Lts Transdermale therapeutische Systeme mit lichtempfindlichen Wirkstoffen
WO2002045701A2 (en) * 2000-12-05 2002-06-13 Noven Pharmaceuticals, Inc. Crystallization inhibition of drugs in transdermal drug delivery systems

Also Published As

Publication number Publication date
PL1541137T3 (pl) 2010-07-30
ATE457168T1 (de) 2010-02-15
EP1541137A3 (en) 2005-11-16
PT1541137E (pt) 2010-05-17
MY144053A (en) 2011-08-15
ES2340925T3 (es) 2010-06-11
EP2138169A3 (en) 2011-04-06
CN101843603B (zh) 2012-06-27
EP1541137B1 (en) 2010-02-10
PT2138169E (pt) 2014-02-17
MY152750A (en) 2014-11-28
ME01069B (me) 2012-10-20
ES2445690T3 (es) 2014-03-04
DK2138169T3 (da) 2013-11-18
CY1110637T1 (el) 2015-04-29
SI2138169T1 (sl) 2014-03-31
SV2006001970A (es) 2006-02-16
HRP20100254T1 (hr) 2010-06-30
PE20051035A1 (es) 2006-02-08
HK1074801A1 (en) 2005-11-25
JO2606B1 (en) 2011-11-01
RS53182B (sr) 2014-06-30
SI1541137T1 (sl) 2010-06-30
DE602004025444D1 (de) 2010-03-25
DK1541137T3 (da) 2010-04-26
EP2138169B1 (en) 2013-11-06
HN2004000526A (es) 2010-02-01
AR046762A1 (es) 2005-12-21
TW200528073A (en) 2005-09-01
UA89766C2 (en) 2010-03-10
CR8465A (es) 2007-06-06
EP2138169A2 (en) 2009-12-30
CY1115064T1 (el) 2016-12-14
GT200400262A (es) 2005-10-31
EP1541137A2 (en) 2005-06-15
PL2138169T3 (pl) 2014-04-30
HRP20140077T1 (hr) 2014-02-28
CN101843603A (zh) 2010-09-29
TWI257299B (en) 2006-07-01
HK1132682A1 (en) 2010-03-05

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