BRPI0415725A - formulação aspergìvel transdérmica, método para administrar um agente farmaceuticamente ativo e método para formar uma pelìcula farmaceuticamente ativa - Google Patents

formulação aspergìvel transdérmica, método para administrar um agente farmaceuticamente ativo e método para formar uma pelìcula farmaceuticamente ativa

Info

Publication number
BRPI0415725A
BRPI0415725A BRPI0415725-7A BRPI0415725A BRPI0415725A BR PI0415725 A BRPI0415725 A BR PI0415725A BR PI0415725 A BRPI0415725 A BR PI0415725A BR PI0415725 A BRPI0415725 A BR PI0415725A
Authority
BR
Brazil
Prior art keywords
pharmaceutically active
active agent
administering
forming
film
Prior art date
Application number
BRPI0415725-7A
Other languages
English (en)
Inventor
Amar Lulla
Geena Malhotra
Original Assignee
Cipla Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cipla Ltd filed Critical Cipla Ltd
Publication of BRPI0415725A publication Critical patent/BRPI0415725A/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/568Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/12Aerosols; Foams
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/70Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7015Drug-containing film-forming compositions, e.g. spray-on
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Dispersion Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Cardiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Heart & Thoracic Surgery (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

"FORMULAçãO ASPERGìVEL TRANSDéRMICA, MéTODO PARA ADMINISTRAR UM AGENTE FARMACEUTICAMENTE ATIVO E MéTODO PARA FORMAR UMA PELìCULA FARMACEUTICAMENTE ATIVA". São providos formulações aspergíveis transdérmicas contendo um agente farmaceuticamente ativo e métodos para administrar as mesmas. As formulações compreendem o agente farmaceuticamente ativo, um copolímero de VP/AV e um veículo não aquoso. As formulações compreendem ainda um agente anti-nucleante para evitar a recristalização do agente farmaceuticamente ativo e um intensificador de penetração para aumentar a taxa de liberação do fármaco através da pele. Quando da aplicação da pele, a presente formulação seca para prover uma película no local de tratamento.
BRPI0415725-7A 2003-10-23 2004-10-21 formulação aspergìvel transdérmica, método para administrar um agente farmaceuticamente ativo e método para formar uma pelìcula farmaceuticamente ativa BRPI0415725A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN1122MU2003 2003-10-23
PCT/GB2004/004487 WO2005041943A1 (en) 2003-10-23 2004-10-21 Transdermal pharmaceutical spray formulations comprising a vp/va copolymer and a non-aqueous vehicle

Publications (1)

Publication Number Publication Date
BRPI0415725A true BRPI0415725A (pt) 2006-12-19

Family

ID=34531861

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0415725-7A BRPI0415725A (pt) 2003-10-23 2004-10-21 formulação aspergìvel transdérmica, método para administrar um agente farmaceuticamente ativo e método para formar uma pelìcula farmaceuticamente ativa

Country Status (23)

Country Link
US (1) US20070219171A1 (pt)
EP (1) EP1686969A1 (pt)
JP (1) JP2007509122A (pt)
CN (1) CN100431531C (pt)
AP (1) AP2006003628A0 (pt)
AR (1) AR046146A1 (pt)
AU (1) AU2004285335B2 (pt)
BR (1) BRPI0415725A (pt)
CA (1) CA2543245A1 (pt)
HK (1) HK1098351A1 (pt)
IL (1) IL175094A0 (pt)
MA (1) MA28167A1 (pt)
MX (1) MXPA06004460A (pt)
NO (1) NO20062234L (pt)
NZ (1) NZ547376A (pt)
PA (1) PA8615501A1 (pt)
PE (1) PE20050443A1 (pt)
RU (1) RU2006117527A (pt)
SM (1) SM200400022A (pt)
SV (1) SV2006001916A (pt)
TW (1) TW200524635A (pt)
WO (1) WO2005041943A1 (pt)
ZA (1) ZA200604036B (pt)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0518769D0 (en) * 2005-09-14 2005-10-19 Medpharm Ltd Topical formulations
CA2719512A1 (en) * 2010-11-01 2012-05-01 Stiefel Research Australia Pty Ltd Polymeric topical compositions
CN102018671B (zh) * 2011-01-05 2012-07-25 浙江大学 一种雌二醇透皮喷雾剂及其制备方法
US20150065449A1 (en) * 2011-08-12 2015-03-05 Florida State University Research Foundation, Inc. Treating Amyloidoses With A Vitamin B12 Composition Including Melatonin, Resveratrol, and EGCG
GB201200062D0 (en) * 2012-01-04 2012-02-15 Innotesto Bvba Estradiol oromucosal liquid compositions
TWI516281B (zh) * 2014-07-16 2016-01-11 健維生技有限公司 改良之睪固酮製劑製法及所得之睪固酮製劑
US20170296485A1 (en) * 2015-11-23 2017-10-19 Grace Therapeutics Llc Topical Film-Forming Spray
EP3737374B1 (en) * 2018-01-10 2024-04-03 Celista Pharmaceuticals Llc Testosterone transdermal spray with film
EP3817731A4 (en) * 2018-07-05 2022-04-06 Celista Pharmaceuticals Llc TRANSDERMAL TESTOSTERONE AND ESTRADIOL SPRAY
CN112206222A (zh) * 2018-11-09 2021-01-12 北京德默高科医药技术有限公司 含有布洛芬结构类似物的多层经皮给药系统
CN115154661A (zh) * 2022-07-29 2022-10-11 广州莱度品牌管理有限公司 一种仿生角质膜的制备方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH01503281A (ja) * 1987-05-27 1989-11-09 ブルグハルト,クルト 経皮治療に有効な医薬包帯剤およびこれを施用するためのデバイス
FR2732223B1 (fr) * 1995-03-30 1997-06-13 Sanofi Sa Composition pharmaceutique pour administration transdermique
FR2739031B1 (fr) * 1995-09-27 1997-11-21 Lhd Lab Hygiene Dietetique Systeme matriciel transdermique d'administration d'un oestrogene et/ou d'un progestatif a base de copolymere styrene-isoprene-styrene, procede de preparation et utilisation en therapeutique
IT1299566B1 (it) * 1998-07-17 2000-03-16 Ifi Istituto Farmacoterapico I Cerotto transdermico e composizioni farmaceutiche comprendenti r (-)- norapropilapomorfina cloridrato e/o s (+) - norapropilapomorfina
ES2209812T3 (es) * 1999-02-05 2004-07-01 Cipla Ltd. Pulverizaciones topicas que contienen una composicion filmogena.
US6962691B1 (en) * 1999-05-20 2005-11-08 U & I Pharmaceuticals Ltd. Topical spray compositions
US6274167B1 (en) * 2000-09-14 2001-08-14 Vincent Margiotta Topical anesthetic patch
US6528040B1 (en) * 2001-01-18 2003-03-04 Maurine Pearson EMU oil-based formulations for use as an analgesic, anesthetic and antipruritic
DE10211832A1 (de) * 2002-03-16 2003-10-02 Lohmann Therapie Syst Lts Hormonhaltiges transdermales therapeutisches System mit einem Wirkstoffreservoir auf der Basis von Vinylacetat-Vinylpyrrolidon-Copolymer mit verbesserter Kohäsion

Also Published As

Publication number Publication date
AU2004285335B2 (en) 2011-02-10
MXPA06004460A (es) 2006-06-27
SM200400022B (it) 2005-08-24
CN100431531C (zh) 2008-11-12
TW200524635A (en) 2005-08-01
SM200400022A (it) 2005-08-24
PE20050443A1 (es) 2005-06-14
CA2543245A1 (en) 2005-05-12
AP2006003628A0 (en) 2006-06-30
MA28167A1 (fr) 2006-09-01
EP1686969A1 (en) 2006-08-09
RU2006117527A (ru) 2007-12-10
IL175094A0 (en) 2006-08-20
KR20070000397A (ko) 2007-01-02
CN1897927A (zh) 2007-01-17
US20070219171A1 (en) 2007-09-20
JP2007509122A (ja) 2007-04-12
SV2006001916A (es) 2006-03-16
AR046146A1 (es) 2005-11-23
AU2004285335A1 (en) 2005-05-12
ZA200604036B (en) 2007-09-26
NO20062234L (no) 2006-06-30
PA8615501A1 (es) 2005-10-25
WO2005041943A1 (en) 2005-05-12
HK1098351A1 (en) 2007-07-20
NZ547376A (en) 2009-07-31

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Legal Events

Date Code Title Description
B11A Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing
B11Y Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette]