RS20050384A - Estri karbaminske kiseline sa antiholinergičkim dejstvom - Google Patents
Estri karbaminske kiseline sa antiholinergičkim dejstvomInfo
- Publication number
- RS20050384A RS20050384A YUP-2005/0384A YUP20050384A RS20050384A RS 20050384 A RS20050384 A RS 20050384A YU P20050384 A YUP20050384 A YU P20050384A RS 20050384 A RS20050384 A RS 20050384A
- Authority
- RS
- Serbia
- Prior art keywords
- acid esters
- carbamic acid
- anticholinergic action
- pharmaceutical compositions
- anticholinergic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
- C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
- C07D451/06—Oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Pulmonology (AREA)
- Urology & Nephrology (AREA)
- Heart & Thoracic Surgery (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Cardiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Predmetni pronalazak se odnosi na nove estre karbaminske kiseline opšte formule 1 u kojoj X- i grupe A, R1, R2, R3 i R4 mogu imati značenja koja su navedena u patentnim zahtevima i opisu pronalaska, na postupke za njihovo dobijanje, kao i na njihovu primenu u farmaceutskim kompozicijama, a naročito farmaceutskim kompozicijama sa antiholinergičkim dejstvom.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10255040A DE10255040A1 (de) | 2002-11-26 | 2002-11-26 | Neue Carbaminsäureester mit anticholinerger Wirksamkeit |
| PCT/EP2003/012912 WO2004048373A1 (de) | 2002-11-26 | 2003-11-19 | Carbaminsäureester mit anticholinerger wirksamkeit |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| RS20050384A true RS20050384A (sr) | 2007-12-31 |
Family
ID=32240420
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| YUP-2005/0384A RS20050384A (sr) | 2002-11-26 | 2003-11-19 | Estri karbaminske kiseline sa antiholinergičkim dejstvom |
Country Status (20)
| Country | Link |
|---|---|
| EP (1) | EP1567526B1 (sr) |
| JP (1) | JP4754829B2 (sr) |
| KR (1) | KR20050086821A (sr) |
| CN (1) | CN1717408A (sr) |
| AT (1) | ATE392424T1 (sr) |
| AU (1) | AU2003289880A1 (sr) |
| BR (1) | BR0316549A (sr) |
| CA (1) | CA2507110C (sr) |
| DE (2) | DE10255040A1 (sr) |
| EA (1) | EA200500775A1 (sr) |
| EC (1) | ECSP055803A (sr) |
| ES (1) | ES2304538T3 (sr) |
| HR (1) | HRP20050465A2 (sr) |
| MX (1) | MXPA05005443A (sr) |
| NO (1) | NO20053089L (sr) |
| PL (1) | PL376638A1 (sr) |
| RS (1) | RS20050384A (sr) |
| UA (1) | UA81649C2 (sr) |
| WO (1) | WO2004048373A1 (sr) |
| ZA (1) | ZA200502946B (sr) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE602004021921D1 (de) | 2003-05-28 | 2009-08-20 | Theravance Inc | Azabicycloalkanverbindungen als muscarinrezeptor antagonisten |
| TW200534855A (en) * | 2004-01-13 | 2005-11-01 | Glaxo Group Ltd | Muscarinic acetylcholine receptor antagonists |
| EP1765339A4 (en) * | 2004-06-30 | 2009-09-02 | Glaxo Group Ltd | ANTAGONISTS OF MUSCARIN ACETYLCHOLIN RECEPTOR |
| US20090142279A1 (en) * | 2004-11-15 | 2009-06-04 | Budzik Brian W | Novel m3 muscarinic acetylcholine receptor antagonists |
| WO2007007282A2 (en) * | 2005-07-11 | 2007-01-18 | Ranbaxy Laboratories Limited | Azabicyclo derivatives as muscarinic receptor antagonists |
| US20090182033A1 (en) * | 2005-12-16 | 2009-07-16 | Argenta Discovery Ltd. | Cyclic Amine Derivatives and Their Uses |
| KR20090107567A (ko) | 2007-02-09 | 2009-10-13 | 아스텔라스세이야쿠 가부시키가이샤 | 아자 가교환 화합물 |
| US10342786B2 (en) | 2017-10-05 | 2019-07-09 | Fulcrum Therapeutics, Inc. | P38 kinase inhibitors reduce DUX4 and downstream gene expression for the treatment of FSHD |
| CA3128468A1 (en) | 2017-10-05 | 2019-04-11 | Fulcrum Therapeutics, Inc. | P38 kinase inhibitors reduce dux4 and downstream gene expression for the treatment of fshd |
| EP3710483A4 (en) | 2017-11-16 | 2021-10-20 | XL-protein GmbH | PASYLATED VEGFR / PDGFR FUSION PROTEINS AND THEIR USE IN THERAPY |
| JP2021505569A (ja) * | 2017-12-04 | 2021-02-18 | フリードリヒ−アレクサンダー−ウニヴェルシテート エアランゲン−ニュルンベルク | M2よりもm3に対して選択性を有するフルオロフェニル置換ムスカリン受容体リガンド |
| KR20220001259A (ko) | 2020-06-29 | 2022-01-05 | (주)아모레퍼시픽 | 표면처리된 무기입자, 이의 제조방법, 이의 분산액 및 이를 포함하는 화장료 조성물 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BE759460A (fr) * | 1969-11-26 | 1971-05-26 | Knoll Ag | Nouveaux carbamates et leur procede de preparation |
| GB8600978D0 (en) * | 1986-01-16 | 1986-02-19 | Beecham Group Plc | Compounds |
| IT1228293B (it) * | 1989-02-06 | 1991-06-07 | Angeli Inst Spa | Benzoderivati di composti eterociclici contenenti azoto. |
| DE4108393A1 (de) * | 1991-03-15 | 1992-09-17 | Boehringer Ingelheim Kg | Neue ester bi- und tricyclischer aminoalkohole, ihre herstellung und ihre verwendung in arzneimitteln |
| WO1995006635A1 (fr) * | 1993-09-02 | 1995-03-09 | Yamanouchi Pharmaceutical Co., Ltd. | Derive de carbamate et medicament le contenant |
| KR970701174A (ko) * | 1994-02-10 | 1997-03-17 | 오노다 마사요시 | 신규한 카바메이트 유도체 및 이의 의약 조성물(Novel carbamate derivative and medicinal composition containing the same) |
| ES2342990T3 (es) * | 1996-03-20 | 2010-07-20 | Wake Forest University Health Sciences | Receptores sigma-2 como biomarcadores de proliferacion de celulas tumorales. |
-
2002
- 2002-11-26 DE DE10255040A patent/DE10255040A1/de not_active Withdrawn
-
2003
- 2003-11-19 HR HR20050465A patent/HRP20050465A2/xx not_active Application Discontinuation
- 2003-11-19 AT AT03782212T patent/ATE392424T1/de active
- 2003-11-19 AU AU2003289880A patent/AU2003289880A1/en not_active Abandoned
- 2003-11-19 WO PCT/EP2003/012912 patent/WO2004048373A1/de active IP Right Grant
- 2003-11-19 JP JP2004554385A patent/JP4754829B2/ja not_active Expired - Lifetime
- 2003-11-19 ES ES03782212T patent/ES2304538T3/es not_active Expired - Lifetime
- 2003-11-19 EA EA200500775A patent/EA200500775A1/ru unknown
- 2003-11-19 CN CNA2003801042073A patent/CN1717408A/zh active Pending
- 2003-11-19 MX MXPA05005443A patent/MXPA05005443A/es active IP Right Grant
- 2003-11-19 EP EP03782212A patent/EP1567526B1/de not_active Expired - Lifetime
- 2003-11-19 PL PL376638A patent/PL376638A1/pl not_active Application Discontinuation
- 2003-11-19 KR KR1020057009429A patent/KR20050086821A/ko not_active Withdrawn
- 2003-11-19 RS YUP-2005/0384A patent/RS20050384A/sr unknown
- 2003-11-19 DE DE50309655T patent/DE50309655D1/de not_active Expired - Lifetime
- 2003-11-19 CA CA2507110A patent/CA2507110C/en not_active Expired - Fee Related
- 2003-11-19 BR BR0316549-3A patent/BR0316549A/pt not_active IP Right Cessation
- 2003-11-19 UA UAA200506234A patent/UA81649C2/ru unknown
-
2005
- 2005-04-12 ZA ZA200502946A patent/ZA200502946B/en unknown
- 2005-05-19 EC EC2005005803A patent/ECSP055803A/es unknown
- 2005-06-23 NO NO20053089A patent/NO20053089L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| MXPA05005443A (es) | 2005-08-03 |
| CA2507110A1 (en) | 2004-06-10 |
| JP2006514010A (ja) | 2006-04-27 |
| ATE392424T1 (de) | 2008-05-15 |
| JP4754829B2 (ja) | 2011-08-24 |
| HRP20050465A2 (en) | 2006-10-31 |
| DE50309655D1 (de) | 2008-05-29 |
| AU2003289880A1 (en) | 2004-06-18 |
| CN1717408A (zh) | 2006-01-04 |
| EP1567526A1 (de) | 2005-08-31 |
| ES2304538T3 (es) | 2008-10-16 |
| PL376638A1 (pl) | 2006-01-09 |
| EP1567526B1 (de) | 2008-04-16 |
| NO20053089D0 (no) | 2005-06-23 |
| KR20050086821A (ko) | 2005-08-30 |
| CA2507110C (en) | 2012-07-10 |
| UA81649C2 (ru) | 2008-01-25 |
| BR0316549A (pt) | 2005-10-04 |
| ECSP055803A (es) | 2005-08-11 |
| EA200500775A1 (ru) | 2005-12-29 |
| DE10255040A1 (de) | 2004-06-03 |
| NO20053089L (no) | 2005-06-23 |
| WO2004048373A1 (de) | 2004-06-10 |
| ZA200502946B (en) | 2005-11-23 |
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