RO74502B - Procedeu pentru prepararea unor delta15-steroide - Google Patents
Procedeu pentru prepararea unor delta15-steroideInfo
- Publication number
- RO74502B RO74502B RO87931A RO8793176A RO74502B RO 74502 B RO74502 B RO 74502B RO 87931 A RO87931 A RO 87931A RO 8793176 A RO8793176 A RO 8793176A RO 74502 B RO74502 B RO 74502B
- Authority
- RO
- Romania
- Prior art keywords
- group
- steroids
- delta
- general formula
- hydrogen atom
- Prior art date
Links
- 238000004519 manufacturing process Methods 0.000 title 1
- 125000002252 acyl group Chemical group 0.000 abstract 3
- 125000004435 hydrogen atom Chemical class [H]* 0.000 abstract 3
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000002603 chloroethyl group Chemical group [H]C([*])([H])C([H])([H])Cl 0.000 abstract 1
- 125000002534 ethynyl group Chemical group [H]C#C* 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 125000000468 ketone group Chemical group 0.000 abstract 1
- 125000004430 oxygen atom Chemical group O* 0.000 abstract 1
- 125000002568 propynyl group Chemical group [*]C#CC([H])([H])[H] 0.000 abstract 1
- 150000003431 steroids Chemical class 0.000 abstract 1
- 125000001412 tetrahydropyranyl group Chemical group 0.000 abstract 1
- 125000004665 trialkylsilyl group Chemical group 0.000 abstract 1
Landscapes
- Steroid Compounds (AREA)
Abstract
Procedeu pentru prepararea unor delta la 15 steroide cu formula generala I: (vezi formula) în care R1 reprezinta hidrogen, o grupa trialchil silil sau o grupa acil, R2 reprezinta o grupa etinil, cloretinil sau propinil, X reprezinta un atom de oxigen sau o grupa aleasa dintre: (vezi formula) în care R3 reprezinta un atom de hidrogen, o grupa acil, R4 reprezinta un atom de hidrogen, o grupa acil, alchil sau tetrahidropiranil, caracterizat prin aceea ca se aduce în reactie un 17-oxo-steroid cu formula generala II: (vezi formula) în care Y reprezinta o grupa ceto libera sau protejata ca cetal...
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19752546062 DE2546062A1 (de) | 1975-10-10 | 1975-10-10 | Delta hoch 15 -steroide |
| DE19762636404 DE2636404C2 (de) | 1976-08-12 | 1976-08-12 | Δ↑1↑↑5↑-17α-Äthinylsteroide der Östranreihe, Verfahren zu ihrer Herstellung sowie diese enthaltende pharmazeutische Präparate |
| DE19762636405 DE2636405C2 (de) | 1976-08-12 | 1976-08-12 | Δ↑1↑↑5↑-17α-Chloräthinyl- und -Propinylsteroide der Östranreihe, Verfahren zu ihrer Herstellung sowie diese enthaltende pharmazeutische Präparate |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| RO74502B true RO74502B (ro) | 1983-01-30 |
| RO74502A RO74502A (ro) | 1983-02-01 |
Family
ID=27186580
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RO7687931A RO74502A (ro) | 1975-10-10 | 1976-10-06 | Procedeu de preparare a 17alfa-etinil17beta-hidroxi-18-metil-14,15-oestradien-3-onei |
Country Status (1)
| Country | Link |
|---|---|
| RO (1) | RO74502A (ro) |
-
1976
- 1976-10-06 RO RO7687931A patent/RO74502A/ro unknown
Also Published As
| Publication number | Publication date |
|---|---|
| RO74502A (ro) | 1983-02-01 |
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