PT99435A - Processo para a preparacao de derivados de amino-sulfonil-ureia e de composicoes farmaceuticas que os contem - Google Patents
Processo para a preparacao de derivados de amino-sulfonil-ureia e de composicoes farmaceuticas que os contemInfo
- Publication number
- PT99435A PT99435A PT99435A PT9943591A PT99435A PT 99435 A PT99435 A PT 99435A PT 99435 A PT99435 A PT 99435A PT 9943591 A PT9943591 A PT 9943591A PT 99435 A PT99435 A PT 99435A
- Authority
- PT
- Portugal
- Prior art keywords
- pharmaceutical compositions
- sulfonyl
- amino
- preparation
- compositions containing
- Prior art date
Links
- OJXASOYYODXRPT-UHFFFAOYSA-N sulfamoylurea Chemical class NC(=O)NS(N)(=O)=O OJXASOYYODXRPT-UHFFFAOYSA-N 0.000 title abstract 3
- 238000000034 method Methods 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- HVYWMOMLDIMFJA-DPAQBDIFSA-N cholesterol Chemical compound C1C=C2C[C@@H](O)CC[C@]2(C)[C@@H]2[C@@H]1[C@@H]1CC[C@H]([C@H](C)CCCC(C)C)[C@@]1(C)CC2 HVYWMOMLDIMFJA-DPAQBDIFSA-N 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 239000003112 inhibitor Substances 0.000 abstract 2
- 239000008280 blood Substances 0.000 abstract 1
- 210000004369 blood Anatomy 0.000 abstract 1
- 238000009877 rendering Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/92—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with a hetero atom directly attached to the ring nitrogen atom
- C07D211/96—Sulfur atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C307/00—Amides of sulfuric acids, i.e. compounds having singly-bound oxygen atoms of sulfate groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C307/04—Diamides of sulfuric acids
- C07C307/06—Diamides of sulfuric acids having nitrogen atoms of the sulfamide groups bound to acyclic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C307/00—Amides of sulfuric acids, i.e. compounds having singly-bound oxygen atoms of sulfate groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C307/04—Diamides of sulfuric acids
- C07C307/08—Diamides of sulfuric acids having nitrogen atoms of the sulfamide groups bound to carbon atoms of rings other than six-membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C307/00—Amides of sulfuric acids, i.e. compounds having singly-bound oxygen atoms of sulfate groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C307/04—Diamides of sulfuric acids
- C07C307/10—Diamides of sulfuric acids having nitrogen atoms of the sulfamide groups bound to carbon atoms of six-membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/04—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C07D307/10—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D307/14—Radicals substituted by nitrogen atoms not forming part of a nitro radical
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
- C07C2601/14—The ring being saturated
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Vascular Medicine (AREA)
- Urology & Nephrology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyridine Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Furan Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US61028790A | 1990-11-07 | 1990-11-07 | |
| US07/747,040 US5214206A (en) | 1990-11-07 | 1991-08-19 | Aminosulfonyl urea acat inhibitors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| PT99435A true PT99435A (pt) | 1992-12-31 |
| PT99435B PT99435B (pt) | 1999-04-30 |
Family
ID=27086230
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PT99435A PT99435B (pt) | 1990-11-07 | 1991-11-06 | Processo para a preparacao de derivados de amino-sulfonil-ureia e de composicoes farmaceuticas que os contem |
Country Status (16)
| Country | Link |
|---|---|
| US (2) | US5214206A (pt) |
| EP (1) | EP0556322B1 (pt) |
| JP (2) | JP3256541B2 (pt) |
| AT (1) | ATE139226T1 (pt) |
| AU (1) | AU657928B2 (pt) |
| CA (1) | CA2094806C (pt) |
| DE (1) | DE69120287T2 (pt) |
| DK (1) | DK0556322T3 (pt) |
| ES (1) | ES2088128T3 (pt) |
| GR (1) | GR3020355T3 (pt) |
| IE (1) | IE75379B1 (pt) |
| MX (1) | MX9101958A (pt) |
| NZ (1) | NZ240481A (pt) |
| PH (1) | PH30665A (pt) |
| PT (1) | PT99435B (pt) |
| WO (1) | WO1992008694A1 (pt) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1992012144A1 (en) * | 1990-12-28 | 1992-07-23 | Teijin Limited | Condensed benzoxa ring compound, production thereof, and pharmaceutical composition containing the same |
| US5576335A (en) * | 1994-02-01 | 1996-11-19 | Nisshin Flour Milling Co., Ltd. | Urea derivatives and their use as ACAT inhibitors |
| US5491170A (en) * | 1994-12-19 | 1996-02-13 | Warner-Lambert Company | β-carboxy sulfonamide ACAT inhibitors |
| US6103733A (en) * | 1998-09-09 | 2000-08-15 | Bachmann; Kenneth A. | Method for increasing HDL cholesterol levels using heteroaromatic phenylmethanes |
| CA2369967A1 (en) * | 2001-02-12 | 2002-08-12 | Joseph Anthony Cornicelli | Methods of treating nuclear factor-kappa b mediated diseases and disorders |
| EP1281399A3 (en) * | 2001-08-01 | 2004-02-11 | Warner-Lambert Company | Dual inhibitors of wax ester and cholesteryl ester synthesis for inhibiting sebum production |
| EP2640721B1 (en) * | 2010-11-16 | 2018-06-06 | Texas Heart Institute | Agonists that enhance binding of integrin-expressing cells to integrin receptors |
| CN103288749A (zh) * | 2013-03-04 | 2013-09-11 | 盐城工学院 | 可作除草剂的氨基磺酰脲类化合物 |
| WO2016053107A1 (en) * | 2014-10-03 | 2016-04-07 | Synaffix B.V. | Sulfamide linker, conjugates thereof, and methods of preparation |
| MY193765A (en) * | 2015-02-16 | 2022-10-27 | Univ Queensland | Sulfonylureas and related compounds and use of same |
| US11858922B2 (en) * | 2016-02-16 | 2024-01-02 | The University Of Queensland | Sulfonylureas and related compounds and use of same |
| HRP20220195T1 (hr) | 2017-07-07 | 2022-04-15 | Inflazome Limited | Novi spojevi sulfonamid karboksamida |
| GB201721185D0 (en) | 2017-12-18 | 2018-01-31 | Nodthera Ltd | Sulphonyl urea derivatives |
| PE20211333A1 (es) | 2018-08-15 | 2021-07-22 | Inflazome Ltd | Compuestos de sulfonamidaurea novedosos |
| SMT202400291T1 (it) | 2019-06-12 | 2024-09-16 | Nodthera Ltd The Mansion | Derivati di solfonilurea e loro usi |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2312404A (en) * | 1939-11-22 | 1943-03-02 | Haack Erich | Method of preparing n-sulphonylureas |
| CH396872A (de) | 1959-08-13 | 1965-08-15 | Ciba Geigy | Verfahren zur Herstellung neuer Harnstoffe |
| US3242174A (en) * | 1962-02-06 | 1966-03-22 | Pfizer & Co C | 1-(tertiary aminosulfonyl)-3-(hydrocarbon) ureas |
| GB990860A (en) * | 1962-02-08 | 1965-05-05 | Pfizer & Co C | N,n-disubstituted sulfamylureas and compositions thereof |
| US3245982A (en) | 1962-03-27 | 1966-04-12 | Pfizer & Co C | Sulfamylsemicarbazides |
| DE1518541A1 (de) * | 1965-03-16 | 1969-09-11 | Boehringer Mannheim Gmbh | Verfahren zur Herstellung von Sulfonylharnstoffen und Sulfonylsemicarbaziden |
| FR2339694A1 (fr) | 1976-01-30 | 1977-08-26 | Martin Usines Fonderie Arthur | Machine a laver le linge comportant un dispositif de sechage par ventilation d'air chaud |
| CH649081A5 (de) * | 1982-01-12 | 1985-04-30 | Ciba Geigy Ag | Triaza-verbindungen. |
-
1991
- 1991-08-19 US US07/747,040 patent/US5214206A/en not_active Expired - Lifetime
- 1991-11-05 ES ES92900981T patent/ES2088128T3/es not_active Expired - Lifetime
- 1991-11-05 EP EP92900981A patent/EP0556322B1/en not_active Expired - Lifetime
- 1991-11-05 CA CA002094806A patent/CA2094806C/en not_active Expired - Fee Related
- 1991-11-05 NZ NZ240481A patent/NZ240481A/xx not_active IP Right Cessation
- 1991-11-05 AU AU89597/91A patent/AU657928B2/en not_active Ceased
- 1991-11-05 AT AT92900981T patent/ATE139226T1/de not_active IP Right Cessation
- 1991-11-05 DE DE69120287T patent/DE69120287T2/de not_active Expired - Fee Related
- 1991-11-05 WO PCT/US1991/008223 patent/WO1992008694A1/en not_active Ceased
- 1991-11-05 JP JP50093292A patent/JP3256541B2/ja not_active Expired - Fee Related
- 1991-11-05 DK DK92900981.9T patent/DK0556322T3/da active
- 1991-11-06 IE IE387491A patent/IE75379B1/en not_active IP Right Cessation
- 1991-11-06 MX MX9101958A patent/MX9101958A/es not_active IP Right Cessation
- 1991-11-06 PH PH43413A patent/PH30665A/en unknown
- 1991-11-06 PT PT99435A patent/PT99435B/pt not_active IP Right Cessation
-
1993
- 1993-02-19 US US08/019,519 patent/US5288757A/en not_active Expired - Lifetime
-
1996
- 1996-06-27 GR GR960401724T patent/GR3020355T3/el unknown
-
2000
- 2000-06-14 JP JP2000177740A patent/JP2001026574A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| PT99435B (pt) | 1999-04-30 |
| US5288757A (en) | 1994-02-22 |
| GR3020355T3 (en) | 1996-09-30 |
| PH30665A (en) | 1997-09-16 |
| EP0556322A1 (en) | 1993-08-25 |
| DK0556322T3 (da) | 1996-10-14 |
| AU657928B2 (en) | 1995-03-30 |
| IE75379B1 (en) | 1997-09-10 |
| MX9101958A (es) | 1992-07-08 |
| DE69120287D1 (en) | 1996-07-18 |
| DE69120287T2 (de) | 1996-10-10 |
| JP3256541B2 (ja) | 2002-02-12 |
| NZ240481A (en) | 1994-06-27 |
| AU8959791A (en) | 1992-06-11 |
| WO1992008694A1 (en) | 1992-05-29 |
| ES2088128T3 (es) | 1996-08-01 |
| IE913874A1 (en) | 1992-05-20 |
| CA2094806C (en) | 2004-11-02 |
| ATE139226T1 (de) | 1996-06-15 |
| JP2001026574A (ja) | 2001-01-30 |
| EP0556322B1 (en) | 1996-06-12 |
| JPH06501707A (ja) | 1994-02-24 |
| US5214206A (en) | 1993-05-25 |
| CA2094806A1 (en) | 1992-05-08 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| BB1A | Laying open of patent application |
Effective date: 19920814 |
|
| FG3A | Patent granted, date of granting |
Effective date: 19990119 |
|
| MM3A | Annulment or lapse |
Effective date: 20060719 |