PT90689A - Processo para a preparacao de composicoes farmaceuticas contendo ibuprofen em associacao com um piperidinoalcanol - Google Patents

Processo para a preparacao de composicoes farmaceuticas contendo ibuprofen em associacao com um piperidinoalcanol

Info

Publication number
PT90689A
PT90689A PT90689A PT9068989A PT90689A PT 90689 A PT90689 A PT 90689A PT 90689 A PT90689 A PT 90689A PT 9068989 A PT9068989 A PT 9068989A PT 90689 A PT90689 A PT 90689A
Authority
PT
Portugal
Prior art keywords
piperidinoalcanol
association
preparation
pharmaceutical compositions
compositions containing
Prior art date
Application number
PT90689A
Other languages
English (en)
Other versions
PT90689B (pt
Inventor
Herbert Schock
David Francis Long
William Richard Nadler
Original Assignee
Merrell Dow Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merrell Dow Pharma filed Critical Merrell Dow Pharma
Publication of PT90689A publication Critical patent/PT90689A/pt
Publication of PT90689B publication Critical patent/PT90689B/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pain & Pain Management (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Rheumatology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PT90689A 1988-06-01 1989-05-30 Processo para a preparacao de composicoes farmaceuticas contendo ibuprofen em associacao com um piperidinoalcanol PT90689B (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US20081788A 1988-06-01 1988-06-01
US07/344,183 US4999226A (en) 1988-06-01 1989-04-27 Pharmaceutical compositions for piperidinoalkanol-ibuprofen combination

Publications (2)

Publication Number Publication Date
PT90689A true PT90689A (pt) 1989-12-29
PT90689B PT90689B (pt) 1993-12-31

Family

ID=26896133

Family Applications (1)

Application Number Title Priority Date Filing Date
PT90689A PT90689B (pt) 1988-06-01 1989-05-30 Processo para a preparacao de composicoes farmaceuticas contendo ibuprofen em associacao com um piperidinoalcanol

Country Status (17)

Country Link
US (1) US4999226A (pt)
EP (1) EP0348683B1 (pt)
JP (1) JP2757017B2 (pt)
KR (1) KR0126129B1 (pt)
CN (1) CN1038021A (pt)
AU (1) AU615751B2 (pt)
CA (1) CA1327011C (pt)
DE (1) DE68900378D1 (pt)
DK (1) DK174638B1 (pt)
ES (1) ES2037908T3 (pt)
FI (1) FI90205C (pt)
GR (1) GR3003477T3 (pt)
HU (1) HU202746B (pt)
IE (1) IE61182B1 (pt)
IL (1) IL90461A0 (pt)
NZ (1) NZ229325A (pt)
PT (1) PT90689B (pt)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5605930A (en) * 1991-10-21 1997-02-25 The United States Of America As Represented By The Department Of Health And Human Services Compositions and methods for treating and preventing pathologies including cancer
JPH069382A (ja) * 1992-04-17 1994-01-18 Takeda Chem Ind Ltd 安定化された固型製剤およびその製造方法
WO1994014476A1 (en) * 1992-12-21 1994-07-07 The Procter & Gamble Company Use of s(+) antipodes of analgesic agents for the manufacture of a composition to treat respiratory disorders
SK279684B6 (sk) * 1993-06-14 1999-02-11 Janssen Pharmaceutica N.V. Tableta a spôsob jej výroby
EP0725639B1 (en) * 1993-10-25 2000-11-15 Merrell Pharmaceuticals Inc. A stable pharmaceutical composition of terfenadine and ibuprofen
ES2148470T3 (es) * 1993-12-10 2000-10-16 Fujisawa Pharmaceutical Co Farmaco analgesico antipiretico combinado.
US5419917A (en) * 1994-02-14 1995-05-30 Andrx Pharmaceuticals, Inc. Controlled release hydrogel formulation
US5399356A (en) * 1994-03-24 1995-03-21 The Procter & Gamble Company Process for making solid dose forms containing bismuth
WO1996026726A1 (en) * 1995-02-28 1996-09-06 Hoechst Marion Roussel, Inc. Pharmaceutical composition for piperidinoalkanol compounds
US5574045A (en) * 1995-06-06 1996-11-12 Hoechst Marion Roussel, Inc. Oral pharmaceutical composition of piperidinoalkanol compounds in solution form
US6077539A (en) 1996-11-12 2000-06-20 Pozen, Inc. Treatment of migraine headache
AU725811B2 (en) * 1997-08-26 2000-10-19 Aventisub Llc Pharmaceutical composition for combination of piperidinoalkanol-decongestant
MY125516A (en) * 1999-11-16 2006-08-30 Smithkline Beecham Plc Novel composition based on thiazolidinedione and metformin and use
WO2002036077A2 (en) * 2000-11-06 2002-05-10 Andrx Pharmaceuticals, Inc. Once a day antihistamine and decongestant formulation
EP1334732B1 (en) * 2000-11-17 2010-06-02 Takeda Pharmaceutical Company Limited Pharmaceutical preparation of n-[2-(1,6,7,8-tetrahydro-2h-indeno[5,4 b]furan-8-yl)ethyl]propionamide coated with a copolyvidone-containing coating free of polyethylene glycol
BR0212951A (pt) * 2001-09-28 2004-10-26 Mcneil Ppc Inc Formas de dosagens compósitas
US20030181488A1 (en) * 2002-03-07 2003-09-25 Boehringer Ingelheim Pharma Gmbh & Co. Kg Administration form for the oral application of 3-[(2-{[4-(hexyloxycarbonylamino-imino-methyl)-phenylamino]-methyl}-1-methyl-1H-benzimidazol-5-carbonyl)-pyridin-2-yl-amino]-propionic acid ethyl ester and the salts thereof
US7807197B2 (en) * 2002-09-28 2010-10-05 Mcneil-Ppc, Inc. Composite dosage forms having an inlaid portion
US8092831B2 (en) * 2002-11-08 2012-01-10 Andrx Pharmaceuticals, Llc Antihistamine and decongestant system
US20040253311A1 (en) * 2002-12-18 2004-12-16 Roger Berlin Multi-layer tablet comprising non-steroidal anti-inflammatory drugs, decongestants and non-sedating antihist amines
US20050220877A1 (en) * 2004-03-31 2005-10-06 Patel Ashish A Bilayer tablet comprising an antihistamine and a decongestant
US7879352B2 (en) * 2004-05-21 2011-02-01 Accu-Break Technologies, Inc. Scored pharmaceutical tablets comprising a plurality of segments
CN1960713A (zh) * 2004-05-21 2007-05-09 阿库-伯雷克技术公司 含有两个或多个单元片段的药片
US8673352B2 (en) * 2005-04-15 2014-03-18 Mcneil-Ppc, Inc. Modified release dosage form
BRPI0620863A8 (pt) 2005-12-29 2018-01-16 Osmotica Kereskedelmi Es Szolgaltato Kft comprimido em camadas com combinação de liberação tripla
US8377475B2 (en) 2009-01-05 2013-02-19 Mcneil-Ppc, Inc. Tablet containing cetirizine, pseudoephedrine, and naproxen containing a barrier layer
CA2748783A1 (en) * 2009-01-05 2010-07-08 Mcneil-Ppc, Inc. Three layer tablet containing cetirizine, pseudoephedrine, and naproxen
US8252330B2 (en) 2009-01-05 2012-08-28 Mcneil-Ppc, Inc. Tablet containing coated particles of cetirizine, pseudoephedrine, and/or naproxen
US20130115250A1 (en) * 2009-05-13 2013-05-09 Wyeth Llc Burst Drug Release Compositions
US11382865B2 (en) * 2016-12-09 2022-07-12 Bayer Animal Health Gmbh Pharmaceutical preparation and method for its manufacture
CN108703828B (zh) * 2018-06-04 2021-03-30 王荣涛 下肢牵引器
CN109481272B (zh) * 2019-01-10 2020-07-24 河南省洛阳正骨医院(河南省骨科医院) 肺癌骨转移术后康复装置

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL70071A (en) * 1982-11-01 1987-12-31 Merrell Dow Pharma Multilayered sustained release pharmaceutical tablets having non-uniform distribution of active ingredient
US4882167A (en) * 1983-05-31 1989-11-21 Jang Choong Gook Dry direct compression compositions for controlled release dosage forms
US4783465A (en) * 1984-04-09 1988-11-08 Analgesic Associates Cough/cold mixtures comprising non-sedating antihistamine drugs
US4552899A (en) * 1984-04-09 1985-11-12 Analgesic Associates Cough/cold mixtures comprising non-steroidal anti-inflammatory drugs
US4806359A (en) * 1987-04-22 1989-02-21 Mcneilab, Inc. Iburprofen sustained release matrix and process
US4808413A (en) * 1987-04-28 1989-02-28 E. R. Squibb & Sons, Inc. Pharmaceutical compositions in the form of beadlets and method

Also Published As

Publication number Publication date
ES2037908T3 (es) 1993-07-01
DK174638B1 (da) 2003-08-04
JP2757017B2 (ja) 1998-05-25
AU615751B2 (en) 1991-10-10
FI892640A (fi) 1989-12-02
NZ229325A (en) 1990-10-26
FI90205C (fi) 1994-01-10
CA1327011C (en) 1994-02-15
EP0348683A1 (en) 1990-01-03
PT90689B (pt) 1993-12-31
FI90205B (fi) 1993-09-30
AU3580089A (en) 1989-12-07
KR900017573A (ko) 1990-12-19
US4999226A (en) 1991-03-12
DK265489D0 (da) 1989-05-31
JPH0228111A (ja) 1990-01-30
DE68900378D1 (de) 1991-12-05
IL90461A0 (en) 1990-01-18
CN1038021A (zh) 1989-12-20
IE61182B1 (en) 1994-10-05
HU202746B (en) 1991-04-29
GR3003477T3 (en) 1993-02-17
DK265489A (da) 1989-12-02
FI892640A0 (fi) 1989-05-31
EP0348683B1 (en) 1991-10-30
IE891795L (en) 1989-12-01
KR0126129B1 (ko) 1997-12-24
HUT52367A (en) 1990-07-28

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Legal Events

Date Code Title Description
FG3A Patent granted, date of granting

Effective date: 19930622

MM4A Annulment/lapse due to non-payment of fees, searched and examined patent

Free format text: MAXIMUM VALIDITY LIMIT REACHED

Effective date: 20090530