PT900227E - Processo melhorado para a sintese de diesteres de ester 2,5-dioxo-4,4-difenil-imidazolidin-1-ilmetilico do acido fosforicoo - Google Patents

Processo melhorado para a sintese de diesteres de ester 2,5-dioxo-4,4-difenil-imidazolidin-1-ilmetilico do acido fosforicoo

Info

Publication number
PT900227E
PT900227E PT97917765T PT97917765T PT900227E PT 900227 E PT900227 E PT 900227E PT 97917765 T PT97917765 T PT 97917765T PT 97917765 T PT97917765 T PT 97917765T PT 900227 E PT900227 E PT 900227E
Authority
PT
Portugal
Prior art keywords
diphenyl
imidazolidin
dioxo
phosphoric acid
pct
Prior art date
Application number
PT97917765T
Other languages
English (en)
Inventor
Edward Mark Davis
James E Ellis
David A Katonak
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of PT900227E publication Critical patent/PT900227E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic System
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/645Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having two nitrogen atoms as the only ring hetero atoms
    • C07F9/6503Five-membered rings
    • C07F9/6506Five-membered rings having the nitrogen atoms in positions 1 and 3
PT97917765T 1996-04-30 1997-04-01 Processo melhorado para a sintese de diesteres de ester 2,5-dioxo-4,4-difenil-imidazolidin-1-ilmetilico do acido fosforicoo PT900227E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US1651596P 1996-04-30 1996-04-30

Publications (1)

Publication Number Publication Date
PT900227E true PT900227E (pt) 2002-05-31

Family

ID=21777523

Family Applications (1)

Application Number Title Priority Date Filing Date
PT97917765T PT900227E (pt) 1996-04-30 1997-04-01 Processo melhorado para a sintese de diesteres de ester 2,5-dioxo-4,4-difenil-imidazolidin-1-ilmetilico do acido fosforicoo

Country Status (15)

Country Link
US (2) US6022975A (pt)
EP (1) EP0900227B1 (pt)
JP (1) JP4035642B2 (pt)
KR (1) KR100453867B1 (pt)
AT (1) ATE210670T1 (pt)
AU (1) AU708127B2 (pt)
BR (1) BR9709198B1 (pt)
DE (1) DE69709091T2 (pt)
DK (1) DK0900227T3 (pt)
ES (1) ES2169375T3 (pt)
NZ (1) NZ332115A (pt)
PT (1) PT900227E (pt)
SI (1) SI0900227T1 (pt)
WO (1) WO1997041132A1 (pt)
ZA (1) ZA973713B (pt)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2169375T3 (es) 1996-04-30 2002-07-01 Warner Lambert Co Proceso mejorado para la sintesis de diesteres del ester 2,5-dioxo-4,4-difenil-imidazolidin-1-ilmetilico de acido fosforico.
US20070219378A1 (en) * 2004-02-05 2007-09-20 Hartmut Zinser Method for Producing Sodium Fosphenytoin
CH696765A5 (de) 2004-06-02 2007-11-30 Cilag Ltd Verfahren zur Herstellung von Natrium-fosphenytoin.
DE102004046356A1 (de) * 2004-09-24 2006-03-30 Clariant Gmbh Verfahren zur Herstellung von Alk(en)ylphosphorsäureestersalzen
JP5732453B2 (ja) * 2009-06-25 2015-06-10 アルカーメス ファーマ アイルランド リミテッド Nh酸性化合物のプロドラッグ
FI2445502T4 (fi) 2009-06-25 2023-01-13 Heterosyklisiä yhdisteitä neurologisten ja psykologisten häiriöiden hoitamiseksi
US8969337B2 (en) 2011-12-15 2015-03-03 Alkermes Pharma Ireland Limited Prodrugs of secondary amine compounds
JP6861430B2 (ja) * 2016-09-29 2021-04-21 ノーベルファーマ株式会社 ホスフェニトインナトリウム水和物及びその合成中間体の製法
AU2019230014A1 (en) 2018-03-05 2020-09-17 Alkermes Pharma Ireland Limited Aripiprazole dosing strategy

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE489216A (pt) * 1948-06-05 1900-01-01
US3741978A (en) * 1971-04-21 1973-06-26 Hercules Inc Certain o,o-di (c1 and c2 alkyl) phosphorodithioate and phosphorothioate esters useful as insecticides and acaricides
US3925406A (en) * 1972-04-04 1975-12-09 Ciba Geigy Corp Dialkoxyphosphonomethyl derivatives of hydantoins
US3980647A (en) * 1972-08-10 1976-09-14 Ciba-Geigy Corporation Adducts of polyglycidyl compounds and dialkoxyphosphono-methyl derivatives of cyclic ureides
CH573948A5 (pt) * 1972-12-12 1976-03-31 Ciba Geigy Ag
US4260769A (en) * 1977-04-22 1981-04-07 Interx Research Corporation 5,5-Diphenylhydantoins
DE3126390A1 (de) * 1981-07-03 1983-01-13 Bayer Ag, 5090 Leverkusen S-azolyl-methyl-di(tri)-thiophosphorsaeureester, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
US4925860A (en) * 1987-08-05 1990-05-15 E. I. Du Pont De Nemours And Company Stable pharmaceutical composition of 3-(hydroxymethyl)-5,5-diphenylhydantoin disodium phosphate ester
ES2169375T3 (es) 1996-04-30 2002-07-01 Warner Lambert Co Proceso mejorado para la sintesis de diesteres del ester 2,5-dioxo-4,4-difenil-imidazolidin-1-ilmetilico de acido fosforico.

Also Published As

Publication number Publication date
AU708127B2 (en) 1999-07-29
EP0900227B1 (en) 2001-12-12
NZ332115A (en) 2000-05-26
JP2000509071A (ja) 2000-07-18
KR20000065111A (ko) 2000-11-06
KR100453867B1 (ko) 2005-01-15
BR9709198A (pt) 1999-08-10
WO1997041132A1 (en) 1997-11-06
DE69709091D1 (de) 2002-01-24
EP0900227A1 (en) 1999-03-10
ATE210670T1 (de) 2001-12-15
DK0900227T3 (da) 2002-04-08
DE69709091T2 (de) 2002-06-20
JP4035642B2 (ja) 2008-01-23
BR9709198B1 (pt) 2008-11-18
AU2600997A (en) 1997-11-19
US6022975A (en) 2000-02-08
ZA973713B (en) 1997-12-01
US6255492B1 (en) 2001-07-03
SI0900227T1 (en) 2002-04-30
ES2169375T3 (es) 2002-07-01

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