PT81886B - Processo para a preparacao de 3-(piperidinil)- e 3-(pirrolidinil)-1h-indazois e de composicoes farmaceuticas que os contem - Google Patents

Processo para a preparacao de 3-(piperidinil)- e 3-(pirrolidinil)-1h-indazois e de composicoes farmaceuticas que os contem

Info

Publication number
PT81886B
PT81886B PT81886A PT8188686A PT81886B PT 81886 B PT81886 B PT 81886B PT 81886 A PT81886 A PT 81886A PT 8188686 A PT8188686 A PT 8188686A PT 81886 B PT81886 B PT 81886B
Authority
PT
Portugal
Prior art keywords
indazoes
pyrrolidinyl
piperidinyl
preparation
pharmaceutical compositions
Prior art date
Application number
PT81886A
Other languages
English (en)
Other versions
PT81886A (en
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of PT81886A publication Critical patent/PT81886A/pt
Publication of PT81886B publication Critical patent/PT81886B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PT81886A 1985-01-23 1986-01-22 Processo para a preparacao de 3-(piperidinil)- e 3-(pirrolidinil)-1h-indazois e de composicoes farmaceuticas que os contem PT81886B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US69419885A 1985-01-23 1985-01-23

Publications (2)

Publication Number Publication Date
PT81886A PT81886A (en) 1986-02-01
PT81886B true PT81886B (pt) 1988-05-27

Family

ID=24787823

Family Applications (1)

Application Number Title Priority Date Filing Date
PT81886A PT81886B (pt) 1985-01-23 1986-01-22 Processo para a preparacao de 3-(piperidinil)- e 3-(pirrolidinil)-1h-indazois e de composicoes farmaceuticas que os contem

Country Status (18)

Country Link
EP (1) EP0192935B1 (pt)
JP (1) JPS61172875A (pt)
KR (1) KR900002243B1 (pt)
AR (1) AR241434A1 (pt)
AT (1) ATE61054T1 (pt)
AU (1) AU581726B2 (pt)
CA (1) CA1287355C (pt)
DE (1) DE3677609D1 (pt)
DK (1) DK32886A (pt)
ES (3) ES8705876A1 (pt)
FI (1) FI82243C (pt)
GR (1) GR860159B (pt)
HU (1) HU196784B (pt)
NO (1) NO164976C (pt)
NZ (1) NZ214876A (pt)
PH (1) PH22660A (pt)
PT (1) PT81886B (pt)
ZA (1) ZA86465B (pt)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ230068A (en) * 1988-07-29 1991-07-26 Dainippon Pharmaceutical Co Indazole-3-carboxylic acid esters and amides of diaza compounds having 6,7, or 8 ring members: preparatory processes and pharmaceutical compositions
IL90879A0 (en) * 1988-09-02 1990-02-09 Janssen Pharmaceutica Nv 3-piperidinyl-indazole derivatives,their preparation and antihypertensive compositions containing them

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4355037A (en) * 1981-11-12 1982-10-19 Hoechst-Roussel Pharmaceuticals 3-(4-Piperidyl)-1,2-benzisoxales
US4458076A (en) * 1983-05-31 1984-07-03 Hoechst-Roussel Pharmaceuticals 3-(4-Piperidinyl)-1,2-benzisothiazoles
HU198036B (en) * 1983-08-22 1989-07-28 Hoechst Roussel Pharma Process for production of derivatives of 3-piperidil-/1h/-indasole and medical preparatives containing them

Also Published As

Publication number Publication date
ATE61054T1 (de) 1991-03-15
AU581726B2 (en) 1989-03-02
KR860005809A (ko) 1986-08-13
HUT40104A (en) 1986-11-28
FI82243B (fi) 1990-10-31
DK32886D0 (da) 1986-01-22
ES551063A0 (es) 1987-05-16
GR860159B (en) 1986-05-19
DK32886A (da) 1986-07-24
FI860287A0 (fi) 1986-01-21
AU5264086A (en) 1986-07-31
FI860287A (fi) 1986-07-24
ES8705876A1 (es) 1987-05-16
PT81886A (en) 1986-02-01
FI82243C (fi) 1991-02-11
ES557043A0 (es) 1988-07-16
ES8802510A1 (es) 1988-07-16
NO164976B (no) 1990-08-27
DE3677609D1 (de) 1991-04-04
PH22660A (en) 1988-11-14
AR241434A1 (es) 1992-07-31
ES557044A0 (es) 1987-12-01
ES8800925A1 (es) 1987-12-01
JPS61172875A (ja) 1986-08-04
CA1287355C (en) 1991-08-06
HU196784B (en) 1989-01-30
KR900002243B1 (ko) 1990-04-07
ZA86465B (en) 1986-09-24
NO860227L (no) 1986-07-24
NO164976C (no) 1990-12-05
EP0192935B1 (en) 1991-02-27
EP0192935A1 (en) 1986-09-03
NZ214876A (en) 1990-03-27

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MM3A Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 19930531