FI860287A - 3-(piperidinyl)- och 3-(pyrrolidinyl) -1h-indazoler, foerfarande foer deras framstaellning och deras anvaendning som laekemedel. - Google Patents

3-(piperidinyl)- och 3-(pyrrolidinyl) -1h-indazoler, foerfarande foer deras framstaellning och deras anvaendning som laekemedel. Download PDF

Info

Publication number
FI860287A
FI860287A FI860287A FI860287A FI860287A FI 860287 A FI860287 A FI 860287A FI 860287 A FI860287 A FI 860287A FI 860287 A FI860287 A FI 860287A FI 860287 A FI860287 A FI 860287A
Authority
FI
Finland
Prior art keywords
och
deras
indazoler
pyrrolidinyl
piperidinyl
Prior art date
Application number
FI860287A
Other languages
English (en)
Other versions
FI82243B (fi
FI860287A0 (fi
FI82243C (fi
Inventor
Joseph T Strupczewski
Original Assignee
Hoechst Roussel Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Roussel Pharma filed Critical Hoechst Roussel Pharma
Publication of FI860287A0 publication Critical patent/FI860287A0/fi
Publication of FI860287A publication Critical patent/FI860287A/fi
Publication of FI82243B publication Critical patent/FI82243B/fi
Application granted granted Critical
Publication of FI82243C publication Critical patent/FI82243C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FI860287A 1985-01-23 1986-01-21 Foerfarande foer framstaellning av terapeutiskt aktiva 3-(4-piperidinyl)-1h-indazolderivat. FI82243C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US69419885A 1985-01-23 1985-01-23
US69419885 1985-01-23

Publications (4)

Publication Number Publication Date
FI860287A0 FI860287A0 (fi) 1986-01-21
FI860287A true FI860287A (fi) 1986-07-24
FI82243B FI82243B (fi) 1990-10-31
FI82243C FI82243C (fi) 1991-02-11

Family

ID=24787823

Family Applications (1)

Application Number Title Priority Date Filing Date
FI860287A FI82243C (fi) 1985-01-23 1986-01-21 Foerfarande foer framstaellning av terapeutiskt aktiva 3-(4-piperidinyl)-1h-indazolderivat.

Country Status (18)

Country Link
EP (1) EP0192935B1 (fi)
JP (1) JPS61172875A (fi)
KR (1) KR900002243B1 (fi)
AR (1) AR241434A1 (fi)
AT (1) ATE61054T1 (fi)
AU (1) AU581726B2 (fi)
CA (1) CA1287355C (fi)
DE (1) DE3677609D1 (fi)
DK (1) DK32886A (fi)
ES (3) ES8705876A1 (fi)
FI (1) FI82243C (fi)
GR (1) GR860159B (fi)
HU (1) HU196784B (fi)
NO (1) NO164976C (fi)
NZ (1) NZ214876A (fi)
PH (1) PH22660A (fi)
PT (1) PT81886B (fi)
ZA (1) ZA86465B (fi)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5017573A (en) * 1988-07-29 1991-05-21 Dainippon Pharmaceutical Co., Ltd. Indazole-3-carboxylic acid derivatives
IL90879A0 (en) * 1988-09-02 1990-02-09 Janssen Pharmaceutica Nv 3-piperidinyl-indazole derivatives,their preparation and antihypertensive compositions containing them

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4355037A (en) * 1981-11-12 1982-10-19 Hoechst-Roussel Pharmaceuticals 3-(4-Piperidyl)-1,2-benzisoxales
US4458076A (en) * 1983-05-31 1984-07-03 Hoechst-Roussel Pharmaceuticals 3-(4-Piperidinyl)-1,2-benzisothiazoles
HU198036B (en) * 1983-08-22 1989-07-28 Hoechst Roussel Pharma Process for production of derivatives of 3-piperidil-/1h/-indasole and medical preparatives containing them

Also Published As

Publication number Publication date
HU196784B (en) 1989-01-30
AU5264086A (en) 1986-07-31
PH22660A (en) 1988-11-14
DK32886A (da) 1986-07-24
ES557044A0 (es) 1987-12-01
HUT40104A (en) 1986-11-28
ATE61054T1 (de) 1991-03-15
PT81886A (en) 1986-02-01
FI82243B (fi) 1990-10-31
ES551063A0 (es) 1987-05-16
FI860287A0 (fi) 1986-01-21
PT81886B (pt) 1988-05-27
DE3677609D1 (de) 1991-04-04
KR860005809A (ko) 1986-08-13
ZA86465B (en) 1986-09-24
CA1287355C (en) 1991-08-06
EP0192935A1 (en) 1986-09-03
ES8705876A1 (es) 1987-05-16
ES8800925A1 (es) 1987-12-01
JPS61172875A (ja) 1986-08-04
KR900002243B1 (ko) 1990-04-07
AU581726B2 (en) 1989-03-02
FI82243C (fi) 1991-02-11
NO164976C (no) 1990-12-05
NZ214876A (en) 1990-03-27
ES557043A0 (es) 1988-07-16
ES8802510A1 (es) 1988-07-16
EP0192935B1 (en) 1991-02-27
GR860159B (en) 1986-05-19
NO860227L (no) 1986-07-24
DK32886D0 (da) 1986-01-22
NO164976B (no) 1990-08-27
AR241434A1 (es) 1992-07-31

Similar Documents

Publication Publication Date Title
FI853152L (fi) Polysackaridderivat med aldehydgrupper, deras framstaellning fraon motsvarande acetaler och deras anvaendning som papperstillsatsmedel.
FI904419A0 (fi) 3-(1-substituerade-4-piperazinyl)- 1h-indazoler, foerfarande foer deras framstaellning och deras anvaendning som laekemedel.
FI864678A (fi) Haolprofila skumplastplattor- och stycken, deras framstaellning och anvaendning som isolerings- och/eller torkningsplattor.
FI873002A (fi) Substituerade hydrazoner, foerfaranden foer deras framstaellning och deras anvaendning som bekaempningsmedel foer skadedjur.
FI863630A0 (fi) Linshaollare, speciellt haollare foer glasoegonlinser som skall renas och daerefter belaeggas.
FI874768A0 (fi) Estrar av hexahydro-8-hydroxy-2,6 -metano-2h-kinolizin-3(4h)- och beslaektade foereningar.
FI862059A (fi) Aminomalonylalanfoereningar och deras anvaendning som dietetiska soetningsmedel.
FI854071L (fi) Metallsalicylater, deras framstaellning och anvaendning som faergframkallare i tryck- eller vaermekaensliga uppteckningsmaterial.
FI854919A (fi) Aminoacylabdaner, foerfarande och mellanprodukter foer deras framstaellning och deras anvaendning som laekemedel.
FI861623A (fi) Aktivt vaete innehaollande komposition, som innehaoller tertiaert dialkanolamin och framstaellningsfoerfarande foer polyuretanskum.
FI864920A0 (fi) N-(pyrrol-1-yl)pyridinamider, foerfarande foer deras framstaellning och deras anvaendning som laekemedel.
FI862642A0 (fi) 3-(substituerade) propenylaminotiazol-yl-kefalosporansyror och deras estrar.
FI875055A0 (fi) Optiskt aktiva gyras-inhibitorer, deras framstaellning och deras anvaendning som antibiotika.
FI863537A (fi) Dihydropyridin-2-hydroxyaminer, foerfarande foer deras framstaellning och deras anvaendning som laekemedel.
FI863550A (fi) Ksantinderivator, foerfarande foer deras framstaellning och deras anvaendning som laekemedel.
FI853854L (fi) Jodtriaminobenzenfoereningar, foerfarande foer deras framstaellning och deras anvaendning som kontrastmedel foer roentgenstraolar.
FI882443A0 (fi) Substituerade vinylkefalosporiner, foerfarande foer deras framstaellning och deras anvaendning som laekemedel,
FI872774A0 (fi) Bensimidazoler, deras framstaellning, formulering och anvaendning som inhibitorer foer magsyraavsoendring.
FI860287A (fi) 3-(piperidinyl)- och 3-(pyrrolidinyl) -1h-indazoler, foerfarande foer deras framstaellning och deras anvaendning som laekemedel.
FI881873A (fi) Kondenserade heteroalkylenkinolinaminer, foerfarande och mellanprodukter foer deras framstaellning och deras anvaendning som laekemedel.
FI860980A (fi) Heterocykliska disulfider och deras anvaendning som immunmodulatorer.
FI843199A0 (fi) Foerfarande, anordning och stycke som skall fastsvetsas foer unfoerande av en svetsfog under vatten maskinellt.
FI874514A (fi) Halogensyklopropyl-foereningar, deras framstaellning och anvaendning som herbicida aemnen.
FI850801L (fi) Nitrodiarylsulfoxidderivat, foerfaranden foer deras framstaellning och dessa som aktiv bestaondsdel innehaollande laekemedels- och skadedjursgiftkompositioner.
FI872783A (fi) Cytorodin s-derivat, foerfarande foer deras framstaellning och deras anvaendning som laekemedel.

Legal Events

Date Code Title Description
MM Patent lapsed
MM Patent lapsed

Owner name: HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED