PT81029B - Processo para a preparacao de derivados de flavanona com efeito antialergico e aplicacao dos mesmos para a preparacao de composicoes farmaceuticas com efeito antialergico - Google Patents

Processo para a preparacao de derivados de flavanona com efeito antialergico e aplicacao dos mesmos para a preparacao de composicoes farmaceuticas com efeito antialergico

Info

Publication number
PT81029B
PT81029B PT81029A PT8102985A PT81029B PT 81029 B PT81029 B PT 81029B PT 81029 A PT81029 A PT 81029A PT 8102985 A PT8102985 A PT 8102985A PT 81029 B PT81029 B PT 81029B
Authority
PT
Portugal
Prior art keywords
antialergic
preparation
effect
application
pharmaceutical compositions
Prior art date
Application number
PT81029A
Other languages
English (en)
Other versions
PT81029A (en
Inventor
Rolf Gericke
Helmut Wahlig
Elvira Dingeldein
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of PT81029A publication Critical patent/PT81029A/pt
Publication of PT81029B publication Critical patent/PT81029B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D311/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/22Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 4
    • C07D311/26Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 4 with aromatic rings attached in position 2 or 3
    • C07D311/28Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 4 with aromatic rings attached in position 2 or 3 with aromatic rings attached in position 2 only
    • C07D311/322,3-Dihydro derivatives, e.g. flavanones
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/207Cyclohexane rings not substituted by nitrogen atoms, e.g. kasugamycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D311/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/22Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 4
    • C07D311/26Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 4 with aromatic rings attached in position 2 or 3
    • C07D311/28Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 4 with aromatic rings attached in position 2 or 3 with aromatic rings attached in position 2 only
    • C07D311/30Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 4 with aromatic rings attached in position 2 or 3 with aromatic rings attached in position 2 only not hydrogenated in the hetero ring, e.g. flavones
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/655Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having oxygen atoms, with or without sulfur, selenium, or tellurium atoms, as the only ring hetero atoms
    • C07F9/6552Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having oxygen atoms, with or without sulfur, selenium, or tellurium atoms, as the only ring hetero atoms the oxygen atom being part of a six-membered ring
    • C07F9/65522Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having oxygen atoms, with or without sulfur, selenium, or tellurium atoms, as the only ring hetero atoms the oxygen atom being part of a six-membered ring condensed with carbocyclic rings or carbocyclic ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/22Cyclohexane rings, substituted by nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Immunology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrane Compounds (AREA)
  • Saccharide Compounds (AREA)
PT81029A 1984-08-28 1985-08-26 Processo para a preparacao de derivados de flavanona com efeito antialergico e aplicacao dos mesmos para a preparacao de composicoes farmaceuticas com efeito antialergico PT81029B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19843431534 DE3431534A1 (de) 1984-08-28 1984-08-28 Flavanonderivate

Publications (2)

Publication Number Publication Date
PT81029A PT81029A (en) 1985-09-01
PT81029B true PT81029B (pt) 1987-12-30

Family

ID=6244043

Family Applications (1)

Application Number Title Priority Date Filing Date
PT81029A PT81029B (pt) 1984-08-28 1985-08-26 Processo para a preparacao de derivados de flavanona com efeito antialergico e aplicacao dos mesmos para a preparacao de composicoes farmaceuticas com efeito antialergico

Country Status (19)

Country Link
US (1) US4937257A (pt)
EP (1) EP0173186B1 (pt)
JP (1) JPH0674259B2 (pt)
KR (1) KR930002101B1 (pt)
AR (1) AR241246A1 (pt)
AT (1) ATE39351T1 (pt)
AU (1) AU586827B2 (pt)
CA (1) CA1270484A (pt)
DD (1) DD236313A5 (pt)
DE (2) DE3431534A1 (pt)
DK (1) DK389985A (pt)
ES (1) ES8609299A1 (pt)
FI (1) FI84061C (pt)
HU (1) HU194901B (pt)
IE (1) IE58202B1 (pt)
IL (1) IL76188A (pt)
NZ (1) NZ213236A (pt)
PT (1) PT81029B (pt)
ZA (1) ZA856521B (pt)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0518750U (ja) * 1991-08-23 1993-03-09 新東工業株式会社 鋳造品取り出し装置
DE4314871A1 (de) * 1993-05-05 1994-11-10 Merck Patent Gmbh Lösungsmittel für ein schwerlösliches Gentamicin-Salz
DE19521642C2 (de) * 1995-06-14 2000-11-09 Aesculap Ag & Co Kg Implantat, seine Verwendung in der Chirurgie und Verfahren zu seiner Herstellung
DE19856668A1 (de) * 1998-12-09 2000-06-15 Aesculap Ag & Co Kg Wirkstoffmatrix in Form eines biologisch resorbierbaren porösen Vlieses, Verfahren zu ihrer Herstellung und Verwendung
ES2707787T3 (es) * 2005-12-02 2019-04-05 Ionis Pharmaceuticals Inc Análogos antibacterianos de aminoglucósido 4,5-sustituidos que tienen sustituyentes múltiples
KR101504115B1 (ko) 2007-03-12 2015-03-19 삼성전자 주식회사 매크로 명령 동작 장치와 매크로 명령 입력 장치 및 방법
EP2148884A1 (en) * 2007-04-10 2010-02-03 Achaogen, Inc. Antibacterial 1,4,5-substituted aminoglycoside analogs
JP5315572B2 (ja) * 2007-08-30 2013-10-16 国立大学法人 千葉大学 フラボノイドの製造方法
WO2010030704A2 (en) 2008-09-10 2010-03-18 Achaogen, Inc. Antibacterial aminoglycoside analogs
WO2010030690A1 (en) 2008-09-10 2010-03-18 Isis Pharmaceuticals, Inc. Antibacterial 4,6-substituted 6', 6" and 1 modified aminoglycoside analogs
WO2010042850A1 (en) 2008-10-09 2010-04-15 Achaogen, Inc. Antibacterial aminoglycoside analogs
WO2010042851A1 (en) 2008-10-09 2010-04-15 Achaogen, Inc. Antibacterial aminoglycoside analogs
CA2777107A1 (en) 2009-10-09 2011-04-14 Achaogen, Inc. Antibacterial aminoglycoside analogs
CN103282370A (zh) 2010-11-17 2013-09-04 尔察祯有限公司 抗菌氨基糖苷类类似物
CA2906184A1 (en) * 2013-03-15 2014-09-18 Api Genesis, Llc Polyphenol/flavonoid compositions and methods of formulating oral hygienic products
DE102015214603B4 (de) * 2015-07-31 2019-01-24 Mathys Ag Bettlach Phosphorhaltige Aminoglycosid-Salze
CN115160280B (zh) * 2022-06-07 2023-08-04 贵州农业职业学院 一种黄烷酮类化合物的合成方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3678044A (en) * 1970-10-22 1972-07-18 Chevron Res Substituted flavanones
US4241069A (en) * 1979-09-04 1980-12-23 Miles Laboratories, Inc. 3-Methylene flavanones and 3-methylene chromanones
GB2122987B (en) * 1982-06-01 1985-09-25 Zyma Sa (+)-cyanidan-3-ol derivatives and pharmaceutical preparations thereof
GB8323291D0 (en) * 1983-08-31 1983-10-05 Zyma Sa Flavanone and thioflavanone derivatives

Also Published As

Publication number Publication date
HUT40096A (en) 1986-11-28
AU4664885A (en) 1986-03-06
DK389985D0 (da) 1985-08-27
CA1270484A (en) 1990-06-19
ZA856521B (en) 1986-04-30
AU586827B2 (en) 1989-07-27
IE852120L (en) 1986-02-28
DK389985A (da) 1986-03-01
ATE39351T1 (de) 1989-01-15
EP0173186B1 (de) 1988-12-21
IE58202B1 (en) 1993-07-28
ES8609299A1 (es) 1986-07-16
KR860001798A (ko) 1986-03-22
KR930002101B1 (ko) 1993-03-26
NZ213236A (en) 1988-05-30
ES546493A0 (es) 1986-07-16
DE3431534A1 (de) 1986-03-13
JPS6160677A (ja) 1986-03-28
IL76188A0 (en) 1985-12-31
DD236313A5 (de) 1986-06-04
IL76188A (en) 1990-11-29
FI84061C (fi) 1991-10-10
FI853277A0 (fi) 1985-08-27
HU194901B (en) 1988-03-28
JPH0674259B2 (ja) 1994-09-21
AR241246A1 (es) 1992-03-31
PT81029A (en) 1985-09-01
FI853277L (fi) 1986-03-01
DE3566887D1 (de) 1989-01-26
US4937257A (en) 1990-06-26
FI84061B (fi) 1991-06-28
EP0173186A1 (de) 1986-03-05

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