PT754680E - Benzoil-guanidinas substituidas em posicao 4 por fluoroalquilo processo para a sua preparacao a sua utilizacao como medicamento bem como medicamento que as contem - Google Patents

Benzoil-guanidinas substituidas em posicao 4 por fluoroalquilo processo para a sua preparacao a sua utilizacao como medicamento bem como medicamento que as contem

Info

Publication number
PT754680E
PT754680E PT96111359T PT96111359T PT754680E PT 754680 E PT754680 E PT 754680E PT 96111359 T PT96111359 T PT 96111359T PT 96111359 T PT96111359 T PT 96111359T PT 754680 E PT754680 E PT 754680E
Authority
PT
Portugal
Prior art keywords
medicinal product
fluoroalquilo
benzoyl
preparation
product containing
Prior art date
Application number
PT96111359T
Other languages
English (en)
Inventor
Albus Dr Udo
Kleemann Dr Heinz-Werner
Joachim Brendel
Jochen Lang Dr Hans
Weichert Dr Andreas
Jan-Robert Schwark
Wolfgang Scholz
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of PT754680E publication Critical patent/PT754680E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00Sulfonic acids; Halides, esters, or anhydrides thereof
    • C07C309/01Sulfonic acids
    • C07C309/28Sulfonic acids having sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C309/45Sulfonic acids having sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing nitrogen atoms, not being part of nitro or nitroso groups, bound to the carbon skeleton
    • C07C309/52Sulfonic acids having sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing nitrogen atoms, not being part of nitro or nitroso groups, bound to the carbon skeleton the carbon skeleton being further substituted by doubly-bound oxygen atoms
    • C07C309/53Sulfonic acids having sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing nitrogen atoms, not being part of nitro or nitroso groups, bound to the carbon skeleton the carbon skeleton being further substituted by doubly-bound oxygen atoms the carbon skeleton containing carbon atoms of quinone rings
    • C07C309/54Sulfonic acids having sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing nitrogen atoms, not being part of nitro or nitroso groups, bound to the carbon skeleton the carbon skeleton being further substituted by doubly-bound oxygen atoms the carbon skeleton containing carbon atoms of quinone rings at least one of the nitrogen atoms being part of any of the groups, X being a hetero atom, Y being any atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00Sulfones; Sulfoxides
    • C07C317/44Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/08Drugs for disorders of the urinary system of the prostate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P41/00Drugs used in surgical methods, e.g. surgery adjuvants for preventing adhesion or for vitreum substitution
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Emergency Medicine (AREA)
  • Surgery (AREA)
  • Vascular Medicine (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
PT96111359T 1995-07-19 1996-07-15 Benzoil-guanidinas substituidas em posicao 4 por fluoroalquilo processo para a sua preparacao a sua utilizacao como medicamento bem como medicamento que as contem PT754680E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19526381A DE19526381A1 (de) 1995-07-19 1995-07-19 4-Fluoralkyl-substituierte Benzoylguanidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament

Publications (1)

Publication Number Publication Date
PT754680E true PT754680E (pt) 2002-06-28

Family

ID=7767257

Family Applications (1)

Application Number Title Priority Date Filing Date
PT96111359T PT754680E (pt) 1995-07-19 1996-07-15 Benzoil-guanidinas substituidas em posicao 4 por fluoroalquilo processo para a sua preparacao a sua utilizacao como medicamento bem como medicamento que as contem

Country Status (28)

Country Link
US (1) US6156800A (pt)
EP (1) EP0754680B1 (pt)
JP (1) JPH0931045A (pt)
KR (1) KR970006282A (pt)
CN (1) CN1072644C (pt)
AR (1) AR003461A1 (pt)
AT (1) ATE211463T1 (pt)
AU (1) AU704649B2 (pt)
BR (1) BR9603112A (pt)
CA (1) CA2181515A1 (pt)
CZ (1) CZ291240B6 (pt)
DE (2) DE19526381A1 (pt)
DK (1) DK0754680T3 (pt)
ES (1) ES2170183T3 (pt)
HR (1) HRP960343B1 (pt)
HU (1) HUP9601976A3 (pt)
IL (1) IL118887A (pt)
MX (1) MX9602841A (pt)
NO (1) NO306612B1 (pt)
NZ (1) NZ299015A (pt)
PL (1) PL183906B1 (pt)
PT (1) PT754680E (pt)
RU (1) RU2165412C2 (pt)
SI (1) SI0754680T1 (pt)
SK (1) SK281604B6 (pt)
TR (1) TR199600588A2 (pt)
TW (1) TW462960B (pt)
ZA (1) ZA966106B (pt)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19526381A1 (de) * 1995-07-19 1997-01-23 Hoechst Ag 4-Fluoralkyl-substituierte Benzoylguanidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament
CA2337087C (en) * 2000-03-08 2006-06-06 Canon Kabushiki Kaisha Magnetic toner, process for production thereof, and image forming method, apparatus and process cartridge using the toner
DE10222192A1 (de) * 2002-05-18 2003-11-27 Aventis Pharma Gmbh Pentafluorsulfuranyl-benzoylguanidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament
US7375138B2 (en) 2002-05-18 2008-05-20 Sanofi-Aventis Deutschland Gmbh Pentafluorosulfanylbenzoylguanidines, processes for their preparation, their use as medicaments or diagnostic aids, and medicaments comprising them
OA13285A (en) * 2003-11-13 2007-01-31 Sanofi Aventis Deutschland Pentafluorosulfanyl benzoylguanidines, method for their production, their use as medicaments or diagnostic agents and medicament containing the same.
US20050124666A1 (en) * 2003-11-13 2005-06-09 Aventis Pharma Deutschland Gmbh Pentafluorosulfanylbenzoylguanidines, process for their preparation, use as a medicament or diagnostic aid, and medicament comprising same
US20220291223A1 (en) 2019-08-07 2022-09-15 Abbott Laboratories Chemiluminescent compounds for multiplexing

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3780027A (en) * 1970-04-29 1973-12-18 Merck & Co Inc Anthranilic acid derivatives
DE3929582A1 (de) * 1989-09-06 1991-03-07 Hoechst Ag Benzoylguanidine, verfahren zu ihrer herstellung, ihre verwendung als medikament sowie sie enthaltendes medikament
DK0556674T3 (da) * 1992-02-15 1996-10-14 Hoechst Ag 3,5-Substituerede benzoylguanidiner med antiarytmisk virkning og inhiberende virkning på celleproliferation
DE59403818D1 (de) * 1993-02-20 1997-10-02 Hoechst Ag Substituierte Benzoylguanidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament, als Inhibitoren des zellulären Na+/H+-Austauschs oder als Diagnostikum sowie sie enthaltendes Medikament
DE4328869A1 (de) * 1993-08-27 1995-03-02 Hoechst Ag Ortho-substituierte Benzoylguanidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament
DE19526381A1 (de) * 1995-07-19 1997-01-23 Hoechst Ag 4-Fluoralkyl-substituierte Benzoylguanidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament

Also Published As

Publication number Publication date
CZ212096A3 (en) 1997-04-16
EP0754680A1 (de) 1997-01-22
HUP9601976A3 (en) 1998-07-28
SI0754680T1 (en) 2002-04-30
DE59608533D1 (de) 2002-02-07
EP0754680B1 (de) 2002-01-02
NO306612B1 (no) 1999-11-29
PL183906B1 (pl) 2002-07-31
KR970006282A (ko) 1997-02-19
MX9602841A (es) 1997-01-31
ZA966106B (en) 1997-02-03
CN1072644C (zh) 2001-10-10
SK93896A3 (en) 1997-05-07
NZ299015A (en) 1997-08-22
JPH0931045A (ja) 1997-02-04
IL118887A (en) 2002-07-25
TR199600588A2 (tr) 1997-03-21
CZ291240B6 (cs) 2003-01-15
ATE211463T1 (de) 2002-01-15
DE19526381A1 (de) 1997-01-23
US6156800A (en) 2000-12-05
CA2181515A1 (en) 1997-01-20
BR9603112A (pt) 1998-05-05
AU6056396A (en) 1997-01-23
TW462960B (en) 2001-11-11
HUP9601976A2 (en) 1997-09-29
DK0754680T3 (da) 2002-04-15
NO962999L (no) 1997-01-20
CN1143076A (zh) 1997-02-19
HRP960343B1 (en) 2002-02-28
NO962999D0 (no) 1996-07-18
SK281604B6 (sk) 2001-05-10
PL314278A1 (en) 1997-01-20
HRP960343A2 (en) 1998-02-28
AU704649B2 (en) 1999-04-29
AR003461A1 (es) 1998-08-05
IL118887A0 (en) 1996-10-31
ES2170183T3 (es) 2002-08-01
RU2165412C2 (ru) 2001-04-20
HU9601976D0 (en) 1996-09-30

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