PT75070B - N-oxacyclyl-alkylpiperidin-derivate verfahren zu ihrer herstellung sie enthaltende pharmazeutische praparate und deren verwendung - Google Patents
N-oxacyclyl-alkylpiperidin-derivate verfahren zu ihrer herstellung sie enthaltende pharmazeutische praparate und deren verwendungInfo
- Publication number
- PT75070B PT75070B PT75070A PT7507082A PT75070B PT 75070 B PT75070 B PT 75070B PT 75070 A PT75070 A PT 75070A PT 7507082 A PT7507082 A PT 7507082A PT 75070 B PT75070 B PT 75070B
- Authority
- PT
- Portugal
- Prior art keywords
- praparates
- oxacyclyl
- alkylpiperidin
- pharmaceutical
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D411/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Neurology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19813124366 DE3124366A1 (de) | 1981-06-20 | 1981-06-20 | N-oxacyclyl-alkylpiperidin-derivate, verfahren zu ihrer herstellung, sie enthaltende pharmazeutische praeparate und deren verwendung |
Publications (2)
Publication Number | Publication Date |
---|---|
PT75070A PT75070A (de) | 1982-07-01 |
PT75070B true PT75070B (de) | 1985-01-07 |
Family
ID=6135055
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PT75070A PT75070B (de) | 1981-06-20 | 1982-06-17 | N-oxacyclyl-alkylpiperidin-derivate verfahren zu ihrer herstellung sie enthaltende pharmazeutische praparate und deren verwendung |
Country Status (20)
Country | Link |
---|---|
US (1) | US4470989A (pt) |
EP (1) | EP0068261B1 (pt) |
JP (1) | JPS58977A (pt) |
KR (1) | KR840000540A (pt) |
AT (1) | ATE12498T1 (pt) |
AU (1) | AU551182B2 (pt) |
CA (1) | CA1175432A (pt) |
DE (2) | DE3124366A1 (pt) |
DK (1) | DK275782A (pt) |
ES (1) | ES513102A0 (pt) |
FI (1) | FI822178L (pt) |
GR (1) | GR76502B (pt) |
HU (1) | HU190989B (pt) |
IE (1) | IE53127B1 (pt) |
IL (1) | IL66084A (pt) |
NO (1) | NO822041L (pt) |
NZ (1) | NZ201006A (pt) |
PH (1) | PH18536A (pt) |
PT (1) | PT75070B (pt) |
ZA (1) | ZA824328B (pt) |
Families Citing this family (24)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3366460D1 (en) * | 1982-08-05 | 1986-10-30 | Toshiba Kk | Color picture tube and method for manufacturing the same |
US5312840A (en) * | 1986-07-10 | 1994-05-17 | State Of Oregon, Acting By And Through The Oregon State Board Of Higher Education | Substituted guanidines having high binding to the sigma receptor and the use thereof |
US5221745A (en) * | 1991-06-21 | 1993-06-22 | American Home Products Corp. | Psychotropic piperidinylmethyl benzodioxans |
US5212170A (en) * | 1991-06-21 | 1993-05-18 | American Home Products Corporation | Psychotropic piperidinylmethyl benzodioxans |
US5182292A (en) * | 1991-06-21 | 1993-01-26 | American Home Products Corporation | Psychotropic piperidinylmethyl benzodioxans |
DE4140540A1 (de) * | 1991-12-09 | 1993-06-17 | Bayer Ag | Neue azaheterocyclylmethyl-chromane |
US6096763A (en) * | 1995-02-23 | 2000-08-01 | Merck & Co., Inc. | α1a adrenergic receptor antagonists |
US5952351A (en) * | 1995-02-23 | 1999-09-14 | Merck & Co., Inc. | Alpha 1a adrenergic receptor antagonists |
GB9603457D0 (pt) * | 1996-02-19 | 1996-04-17 | Merck & Co Inc | |
US6025355A (en) * | 1997-05-19 | 2000-02-15 | Cambridge Neuroscience, Inc. | Pharmaceutically active compounds and methods of use |
US6242198B1 (en) | 1996-07-25 | 2001-06-05 | Cambridge Neuroscience, Inc. | Methods of treatment of eye trauma and disorders |
US6756389B2 (en) * | 1996-08-09 | 2004-06-29 | Cambridge Neuroscience, Inc. | Pharmaceutically active compounds and methods of use |
KR100699512B1 (ko) | 1999-06-02 | 2007-03-26 | 얀센 파마슈티카 엔.브이. | 아미노알킬 치환된 (벤조디옥산, 벤조푸란 또는 벤조피란)유도체 |
CA2374905C (en) | 1999-06-02 | 2010-02-23 | Janssen Pharmaceutica N.V. | Pyrrolidinyl, piperidinyl or homopiperidinyl-substituted benzopyran derivatives for treating impaired fundic relaxation |
JO2654B1 (en) * | 2000-09-04 | 2012-06-17 | شركة جانسين فارماسوتيكا ان. في | Multiple aryl caroxa amides are useful as lipid - lowering agents |
JO2409B1 (en) * | 2000-11-21 | 2007-06-17 | شركة جانسين فارماسوتيكا ان. في | Second-phenyl carboxy amides are useful as lipid-lowering agents |
CA2465328C (en) * | 2001-11-01 | 2011-06-14 | Michael Francis Gross | Piperidines |
WO2007036715A2 (en) | 2005-09-30 | 2007-04-05 | Glaxo Group Limited | Compounds which have activity at m1 receptor and their uses in medicine |
US8288413B2 (en) | 2005-09-30 | 2012-10-16 | Glaxo Group Limited | Benzimidazolones which have activity at M1 receptor |
EP1960389B1 (en) | 2005-09-30 | 2012-08-15 | Glaxo Group Limited | Compounds which have activity at m1 receptor and their uses in medicine |
GB0605784D0 (en) * | 2006-03-22 | 2006-05-03 | Glaxo Group Ltd | Compounds |
GB0718415D0 (en) | 2007-09-20 | 2007-10-31 | Glaxo Group Ltd | Compounds |
EP2194982A1 (en) | 2007-09-20 | 2010-06-16 | Glaxo Group Limited | Compounds which have activity at m1 receptor and their uses in medicine |
CN108358832A (zh) * | 2017-12-29 | 2018-08-03 | 上海艾康睿医药科技有限公司 | 一种合成4-[(2-氨基-4-氯)苯基]-氨基-n-哌啶甲酸乙酯的方法 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3910930A (en) * | 1973-01-04 | 1975-10-07 | Janssen Pharmaceutica Nv | 1-{55 1-{8 2-(1,4-Benzodioxan-2-yl)-2-hydroxyethyl{9 -4-piperidyl{56 -2-benzimidazolinones |
US4066772A (en) * | 1975-07-21 | 1978-01-03 | Janssen Pharmaceutica N.V. | 1,3-Dihydro-1-[3-(1-piperidinyl)propyl]-2H-benzimidazol-2-ones and related compounds |
GR71865B (pt) * | 1978-03-20 | 1983-07-07 | Ciba Geigy | |
US4181802A (en) * | 1978-05-11 | 1980-01-01 | Janssen Pharmaceutica N.V. | 1-(Heterocyclylalkyl)-1,3-dihydro-2-H-benzimidazole-2-ones |
US4329348A (en) * | 1979-02-26 | 1982-05-11 | Ciba-Geigy Corporation | N-Oxacyclic-alkylpiperidines as psychostimulants |
-
1981
- 1981-06-20 DE DE19813124366 patent/DE3124366A1/de not_active Withdrawn
-
1982
- 1982-06-14 AT AT82105174T patent/ATE12498T1/de active
- 1982-06-14 EP EP82105174A patent/EP0068261B1/de not_active Expired
- 1982-06-14 DE DE8282105174T patent/DE3262861D1/de not_active Expired
- 1982-06-15 ES ES513102A patent/ES513102A0/es active Granted
- 1982-06-17 PT PT75070A patent/PT75070B/pt unknown
- 1982-06-17 FI FI822178A patent/FI822178L/fi not_active Application Discontinuation
- 1982-06-18 JP JP57104048A patent/JPS58977A/ja active Pending
- 1982-06-18 DK DK275782A patent/DK275782A/da not_active Application Discontinuation
- 1982-06-18 IE IE1448/82A patent/IE53127B1/en unknown
- 1982-06-18 NZ NZ201006A patent/NZ201006A/en unknown
- 1982-06-18 HU HU821992A patent/HU190989B/hu unknown
- 1982-06-18 GR GR68474A patent/GR76502B/el unknown
- 1982-06-18 CA CA000405525A patent/CA1175432A/en not_active Expired
- 1982-06-18 PH PH27449A patent/PH18536A/en unknown
- 1982-06-18 IL IL66084A patent/IL66084A/xx unknown
- 1982-06-18 US US06/389,677 patent/US4470989A/en not_active Expired - Fee Related
- 1982-06-18 ZA ZA824328A patent/ZA824328B/xx unknown
- 1982-06-18 KR KR1019820002715A patent/KR840000540A/ko unknown
- 1982-06-18 NO NO822041A patent/NO822041L/no unknown
- 1982-06-18 AU AU84992/82A patent/AU551182B2/en not_active Ceased
Also Published As
Publication number | Publication date |
---|---|
DK275782A (da) | 1982-12-21 |
US4470989A (en) | 1984-09-11 |
IL66084A0 (en) | 1982-09-30 |
FI822178A0 (fi) | 1982-06-17 |
DE3262861D1 (en) | 1985-05-09 |
ATE12498T1 (de) | 1985-04-15 |
AU551182B2 (en) | 1986-04-17 |
CA1175432A (en) | 1984-10-02 |
PT75070A (de) | 1982-07-01 |
GR76502B (pt) | 1984-08-10 |
ZA824328B (en) | 1983-04-27 |
DE3124366A1 (de) | 1982-12-30 |
ES8304974A1 (es) | 1983-03-16 |
JPS58977A (ja) | 1983-01-06 |
AU8499282A (en) | 1983-01-06 |
NZ201006A (en) | 1985-12-13 |
PH18536A (en) | 1985-08-09 |
IL66084A (en) | 1986-07-31 |
IE53127B1 (en) | 1988-07-06 |
NO822041L (no) | 1982-12-21 |
FI822178L (fi) | 1982-12-21 |
KR840000540A (ko) | 1984-02-25 |
ES513102A0 (es) | 1983-03-16 |
EP0068261A1 (de) | 1983-01-05 |
IE821448L (en) | 1982-12-20 |
EP0068261B1 (de) | 1985-04-03 |
HU190989B (en) | 1986-12-28 |
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