PT1858877E - Ureias substituídas 1,3 diarilo, moduladoras da atividade de quinase - Google Patents

Ureias substituídas 1,3 diarilo, moduladoras da atividade de quinase Download PDF

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Publication number
PT1858877E
PT1858877E PT67183582T PT06718358T PT1858877E PT 1858877 E PT1858877 E PT 1858877E PT 67183582 T PT67183582 T PT 67183582T PT 06718358 T PT06718358 T PT 06718358T PT 1858877 E PT1858877 E PT 1858877E
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PT
Portugal
Prior art keywords
modulators
kinase activity
substituted diaryl
diaryl ureas
ureas
Prior art date
Application number
PT67183582T
Other languages
English (en)
Inventor
Scott A Mitchell
Mihaela Diana Danca
Peter A Blomgren
Robert W Desimone
Douglas A I Pippin
Original Assignee
Gilead Connecticut Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gilead Connecticut Inc filed Critical Gilead Connecticut Inc
Publication of PT1858877E publication Critical patent/PT1858877E/pt

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
PT67183582T 2005-01-14 2006-01-13 Ureias substituídas 1,3 diarilo, moduladoras da atividade de quinase PT1858877E (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US64385605P 2005-01-14 2005-01-14
US73311605P 2005-11-02 2005-11-02

Publications (1)

Publication Number Publication Date
PT1858877E true PT1858877E (pt) 2014-06-05

Family

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Family Applications (1)

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PT67183582T PT1858877E (pt) 2005-01-14 2006-01-13 Ureias substituídas 1,3 diarilo, moduladoras da atividade de quinase

Country Status (6)

Country Link
US (1) US7625931B2 (pt)
EP (1) EP1858877B1 (pt)
ES (1) ES2465469T3 (pt)
PL (1) PL1858877T3 (pt)
PT (1) PT1858877E (pt)
WO (1) WO2006076592A1 (pt)

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Also Published As

Publication number Publication date
EP1858877A1 (en) 2007-11-28
PL1858877T3 (pl) 2014-08-29
US20060211738A1 (en) 2006-09-21
WO2006076592A1 (en) 2006-07-20
EP1858877B1 (en) 2014-03-12
US7625931B2 (en) 2009-12-01
ES2465469T3 (es) 2014-06-05

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