PT1234818E - Sais de calcio de derivados de 1,5-benzodiazepina, processo para producao dos sais e drogas que os contem - Google Patents

Sais de calcio de derivados de 1,5-benzodiazepina, processo para producao dos sais e drogas que os contem

Info

Publication number
PT1234818E
PT1234818E PT00979047T PT00979047T PT1234818E PT 1234818 E PT1234818 E PT 1234818E PT 00979047 T PT00979047 T PT 00979047T PT 00979047 T PT00979047 T PT 00979047T PT 1234818 E PT1234818 E PT 1234818E
Authority
PT
Portugal
Prior art keywords
salts
drugs
contain
production
benzodiazepine derivatives
Prior art date
Application number
PT00979047T
Other languages
English (en)
Inventor
Katsuo Shinozaki
Naoyoshi Miura
Kiyoto Maeda
Masakazu Murata
Taguchi Hiroaki
Kawase Nobuo
Original Assignee
Zeria Pharm Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zeria Pharm Co Ltd filed Critical Zeria Pharm Co Ltd
Publication of PT1234818E publication Critical patent/PT1234818E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/121,5-Benzodiazepines; Hydrogenated 1,5-benzodiazepines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)
PT00979047T 1999-12-02 2000-12-01 Sais de calcio de derivados de 1,5-benzodiazepina, processo para producao dos sais e drogas que os contem PT1234818E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP34279999 1999-12-02

Publications (1)

Publication Number Publication Date
PT1234818E true PT1234818E (pt) 2005-01-31

Family

ID=18356597

Family Applications (1)

Application Number Title Priority Date Filing Date
PT00979047T PT1234818E (pt) 1999-12-02 2000-12-01 Sais de calcio de derivados de 1,5-benzodiazepina, processo para producao dos sais e drogas que os contem

Country Status (13)

Country Link
US (1) US6747022B2 (pt)
EP (1) EP1234818B1 (pt)
JP (1) JP3922024B2 (pt)
KR (1) KR100753005B1 (pt)
CN (1) CN1221538C (pt)
AT (1) ATE275403T1 (pt)
AU (1) AU776283B2 (pt)
CA (1) CA2392057C (pt)
DE (1) DE60013639T2 (pt)
ES (1) ES2228633T3 (pt)
PT (1) PT1234818E (pt)
TW (1) TWI288747B (pt)
WO (1) WO2001040197A1 (pt)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN100481894C (zh) * 2000-08-28 2009-04-22 索尼电子有限公司 用于交互式电视的系统
EP1789391B1 (en) 2004-07-23 2017-06-28 Endocyte, Inc. Bivalent linkers and conjugates thereof
SI1839662T1 (sl) * 2005-01-19 2010-07-30 Zeria Pharm Co Ltd Antitumorsko sredstvo
US9877965B2 (en) 2007-06-25 2018-01-30 Endocyte, Inc. Vitamin receptor drug delivery conjugates for treating inflammation
BRPI0812970A2 (pt) 2007-06-25 2019-09-24 Endocyte Inc conjugados contendo espaçadores hidrofílicos
TWI459948B (zh) * 2008-05-15 2014-11-11 Zeria Pharm Co Ltd The use of a 1,5-benzodiazepine derivative or a pharmaceutically acceptable salt thereof for the manufacture of a pain therapeutic agent composition
CN102333763A (zh) * 2009-03-31 2012-01-25 善利亚新药工业股份有限公司 1,5-苯二氮䓬衍生物的制备方法
US10080805B2 (en) 2012-02-24 2018-09-25 Purdue Research Foundation Cholecystokinin B receptor targeting for imaging and therapy
CN104604880A (zh) * 2014-12-31 2015-05-13 江阴苏利化学股份有限公司 一种含有氮杂卓的防治甘蓝蚜虫的农药组合物
JP2019131467A (ja) * 2016-04-08 2019-08-08 ゼリア新薬工業株式会社 1,5−ベンゾジアゼピン化合物の結晶
JP2019167295A (ja) * 2016-07-04 2019-10-03 ゼリア新薬工業株式会社 1,5−ベンゾジアゼピン化合物カルシウム塩の製造法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4820834A (en) 1984-06-26 1989-04-11 Merck & Co., Inc. Benzodiazepine analogs
CA1332410C (en) 1984-06-26 1994-10-11 Roger M. Freidinger Benzodiazepine analogs
AU670597B2 (en) 1992-06-24 1996-07-25 Ferring B.V. Novel benzodiazepine derivative
EP0728748B1 (en) 1993-12-28 2002-03-06 Shionogi & Co., Ltd. Benzodiazepine derivatives
AU721081B2 (en) * 1996-12-10 2000-06-22 Zeria Pharmaceutical Co., Ltd. 1,5-benzodiazepine derivatives
JP2000026434A (ja) * 1998-06-05 2000-01-25 Zeria Pharmaceut Co Ltd 新規1,5−ベンゾジアゼピン誘導体

Also Published As

Publication number Publication date
TWI288747B (en) 2007-10-21
EP1234818A4 (en) 2002-11-06
DE60013639T2 (de) 2005-02-03
CA2392057C (en) 2009-10-27
US6747022B2 (en) 2004-06-08
KR20020058038A (ko) 2002-07-12
ATE275403T1 (de) 2004-09-15
DE60013639D1 (de) 2004-10-14
AU1650301A (en) 2001-06-12
KR100753005B1 (ko) 2007-08-30
EP1234818A1 (en) 2002-08-28
CN1409706A (zh) 2003-04-09
CN1221538C (zh) 2005-10-05
AU776283B2 (en) 2004-09-02
JP3922024B2 (ja) 2007-05-30
EP1234818B1 (en) 2004-09-08
CA2392057A1 (en) 2001-06-07
WO2001040197A1 (fr) 2001-06-07
US20030096809A1 (en) 2003-05-22
ES2228633T3 (es) 2005-04-16

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