PT1189932E - Derivados de echinocandina processo para a sua preparacao e sua utilizacao como agentes antifungicos - Google Patents

Derivados de echinocandina processo para a sua preparacao e sua utilizacao como agentes antifungicos

Info

Publication number
PT1189932E
PT1189932E PT00940456T PT00940456T PT1189932E PT 1189932 E PT1189932 E PT 1189932E PT 00940456 T PT00940456 T PT 00940456T PT 00940456 T PT00940456 T PT 00940456T PT 1189932 E PT1189932 E PT 1189932E
Authority
PT
Portugal
Prior art keywords
antifung
echinocandin
derivatives
agents
preparation
Prior art date
Application number
PT00940456T
Other languages
English (en)
Inventor
Patrick Fauveau
Alain Corbier
Nathalie Pietre-Dischamp
Laurent Schio
Pascale Vicat
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Publication of PT1189932E publication Critical patent/PT1189932E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/50Cyclic peptides containing at least one abnormal peptide link
    • C07K7/54Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
    • C07K7/56Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
PT00940456T 1999-06-09 2000-06-08 Derivados de echinocandina processo para a sua preparacao e sua utilizacao como agentes antifungicos PT1189932E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9907252A FR2794747B1 (fr) 1999-06-09 1999-06-09 Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme anti-fongiques

Publications (1)

Publication Number Publication Date
PT1189932E true PT1189932E (pt) 2003-09-30

Family

ID=9546549

Family Applications (1)

Application Number Title Priority Date Filing Date
PT00940456T PT1189932E (pt) 1999-06-09 2000-06-08 Derivados de echinocandina processo para a sua preparacao e sua utilizacao como agentes antifungicos

Country Status (18)

Country Link
US (1) US7005417B1 (pt)
EP (1) EP1189932B1 (pt)
JP (1) JP4619592B2 (pt)
AR (1) AR024315A1 (pt)
AT (1) ATE240971T1 (pt)
AU (1) AU5539100A (pt)
CA (1) CA2376490A1 (pt)
CO (1) CO5200761A1 (pt)
DE (1) DE60002866T2 (pt)
DK (1) DK1189932T3 (pt)
ES (1) ES2194744T3 (pt)
FR (1) FR2794747B1 (pt)
GT (1) GT200000090A (pt)
PE (1) PE20010234A1 (pt)
PT (1) PT1189932E (pt)
TN (1) TNSN00127A1 (pt)
UY (1) UY26195A1 (pt)
WO (1) WO2000075178A1 (pt)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA72200C2 (uk) * 1997-12-10 2005-02-15 Авентіс Фарма С.А. Похідні ехінокандину, спосіб їх одержання, їх застосування, проміжні сполуки та фармацевтична композиція
FR2794746B1 (fr) * 1999-06-09 2002-12-06 Hoechst Marion Roussel Inc Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme anti-fongiques
FR2833596B1 (fr) * 2001-12-14 2005-02-18 Aventis Pharma Sa Procede de preparation de derives d'echinocandine
DE102004060750A1 (de) 2004-12-15 2006-07-13 Sanofi-Aventis Deutschland Gmbh Verfahren zur Deacylierung von Lipopeptiden
US8853392B2 (en) 2007-06-03 2014-10-07 Vanderbilt University Benzamide mGluR5 positive allosteric modulators and methods of making and using same
US8034806B2 (en) 2007-11-02 2011-10-11 Vanderbilt University Bicyclic mGluR5 positive allosteric modulators and methods of making and using same
HUE029720T2 (en) * 2011-09-09 2017-03-28 Sandoz Ag Preparation of micafungin intermediates
WO2016056023A2 (en) * 2014-10-07 2016-04-14 Alaparthi Lakshmi Prasad Intermediates and processes to prepare micafungin

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL109615A (en) * 1993-05-17 2000-12-06 Fujisawa Pharmaceutical Co Cyclic polypeptide derivatives processes for the preparation thereof and pharmaceutical compositions containing the same
US5516756A (en) * 1994-10-31 1996-05-14 Merck & Co., Inc. Aza cyclohexapeptide compounds
US5646111A (en) * 1995-04-07 1997-07-08 Eli Lilly And Company Cyclic peptide antifungal Agents
AUPO381496A0 (en) * 1996-11-25 1996-12-19 Fujisawa Pharmaceutical Co., Ltd. New compound
UA72200C2 (uk) * 1997-12-10 2005-02-15 Авентіс Фарма С.А. Похідні ехінокандину, спосіб їх одержання, їх застосування, проміжні сполуки та фармацевтична композиція

Also Published As

Publication number Publication date
ES2194744T3 (es) 2003-12-01
DK1189932T3 (da) 2003-09-15
AR024315A1 (es) 2002-09-25
DE60002866D1 (de) 2003-06-26
FR2794747B1 (fr) 2004-04-16
EP1189932A1 (fr) 2002-03-27
JP4619592B2 (ja) 2011-01-26
JP2003504309A (ja) 2003-02-04
UY26195A1 (es) 2001-01-31
PE20010234A1 (es) 2001-02-24
AU5539100A (en) 2000-12-28
ATE240971T1 (de) 2003-06-15
FR2794747A1 (fr) 2000-12-15
DE60002866T2 (de) 2004-03-11
GT200000090A (es) 2001-11-30
EP1189932B1 (fr) 2003-05-21
TNSN00127A1 (fr) 2005-11-10
CO5200761A1 (es) 2002-09-27
WO2000075178A1 (fr) 2000-12-14
US7005417B1 (en) 2006-02-28
CA2376490A1 (fr) 2000-12-14

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