GT200000090A - Nuevos derivados de equinocandina, su procedimiento de preparacion y su aplicacion como antifungicos. - Google Patents
Nuevos derivados de equinocandina, su procedimiento de preparacion y su aplicacion como antifungicos.Info
- Publication number
- GT200000090A GT200000090A GT200000090A GT200000090A GT200000090A GT 200000090 A GT200000090 A GT 200000090A GT 200000090 A GT200000090 A GT 200000090A GT 200000090 A GT200000090 A GT 200000090A GT 200000090 A GT200000090 A GT 200000090A
- Authority
- GT
- Guatemala
- Prior art keywords
- application
- preparation procedure
- equinocandina
- antifungicos
- new derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/50—Cyclic peptides containing at least one abnormal peptide link
- C07K7/54—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
- C07K7/56—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Biochemistry (AREA)
- Oncology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Communicable Diseases (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Hydrogenated Pyridines (AREA)
Abstract
LA PRESENTE INVENCION SE REFIERE A NUEVOS DERIVADOS DE EQUINOCANDINA (VER FORMULA I, EN LOS CUALES R1 = H O CH3; R2 = AMINAS PRIMARIAS, SECUNDARIAS O CICLICAS; R3 = H, CH3 O OH; R = CADENA LINEAL, RAMIFICADA O CICLICA DE HASTA 30 CARBONOS QUE INCLUYE UNO O VARIOS HETEROATOMOS; T = H, CH3, AMIDA, NITRILO O AMINA; Y = H, OH, HALOGENO, O RADICAL BISULFATO O UNA DE LAS SALES DE ESTE RADICAL; PARA LOCALIZAR LOS GRUPOS ESPECIFICOS EN UNA ESTRUCTURA DADA DEBERA CONSULTARSE EL MATERIAL ORIGINAL), EN TODAS LAS FORMAS DE ISOMEROS POSIBLES ASI COMO SUS MEZCLAS, SU PROCEDIMIENTO DE PREPARACION Y SU APLICACION COMO ANTIFUNGICOS.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9907252A FR2794747B1 (fr) | 1999-06-09 | 1999-06-09 | Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme anti-fongiques |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GT200000090A true GT200000090A (es) | 2001-11-30 |
Family
ID=9546549
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GT200000090A GT200000090A (es) | 1999-06-09 | 2000-06-08 | Nuevos derivados de equinocandina, su procedimiento de preparacion y su aplicacion como antifungicos. |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US7005417B1 (es) |
| EP (1) | EP1189932B1 (es) |
| JP (1) | JP4619592B2 (es) |
| AR (1) | AR024315A1 (es) |
| AT (1) | ATE240971T1 (es) |
| AU (1) | AU5539100A (es) |
| CA (1) | CA2376490A1 (es) |
| CO (1) | CO5200761A1 (es) |
| DE (1) | DE60002866T2 (es) |
| DK (1) | DK1189932T3 (es) |
| ES (1) | ES2194744T3 (es) |
| FR (1) | FR2794747B1 (es) |
| GT (1) | GT200000090A (es) |
| PE (1) | PE20010234A1 (es) |
| PT (1) | PT1189932E (es) |
| TN (1) | TNSN00127A1 (es) |
| UY (1) | UY26195A1 (es) |
| WO (1) | WO2000075178A1 (es) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| UA72200C2 (uk) * | 1997-12-10 | 2005-02-15 | Авентіс Фарма С.А. | Похідні ехінокандину, спосіб їх одержання, їх застосування, проміжні сполуки та фармацевтична композиція |
| FR2794746B1 (fr) * | 1999-06-09 | 2002-12-06 | Hoechst Marion Roussel Inc | Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme anti-fongiques |
| FR2833596B1 (fr) * | 2001-12-14 | 2005-02-18 | Aventis Pharma Sa | Procede de preparation de derives d'echinocandine |
| DE102004060750A1 (de) | 2004-12-15 | 2006-07-13 | Sanofi-Aventis Deutschland Gmbh | Verfahren zur Deacylierung von Lipopeptiden |
| US8853392B2 (en) | 2007-06-03 | 2014-10-07 | Vanderbilt University | Benzamide mGluR5 positive allosteric modulators and methods of making and using same |
| US8034806B2 (en) | 2007-11-02 | 2011-10-11 | Vanderbilt University | Bicyclic mGluR5 positive allosteric modulators and methods of making and using same |
| KR20140069097A (ko) * | 2011-09-09 | 2014-06-09 | 산도즈 아게 | 미카펀진 중간체의 제조 |
| EP3226885A4 (en) * | 2014-10-07 | 2018-07-18 | Alaparthi, Lakshmi Prasad | Intermediates and processes to prepare micafungin |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL109615A (en) * | 1993-05-17 | 2000-12-06 | Fujisawa Pharmaceutical Co | Cyclic polypeptide derivatives processes for the preparation thereof and pharmaceutical compositions containing the same |
| US5516756A (en) * | 1994-10-31 | 1996-05-14 | Merck & Co., Inc. | Aza cyclohexapeptide compounds |
| US5646111A (en) * | 1995-04-07 | 1997-07-08 | Eli Lilly And Company | Cyclic peptide antifungal Agents |
| AUPO381496A0 (en) * | 1996-11-25 | 1996-12-19 | Fujisawa Pharmaceutical Co., Ltd. | New compound |
| UA72200C2 (uk) * | 1997-12-10 | 2005-02-15 | Авентіс Фарма С.А. | Похідні ехінокандину, спосіб їх одержання, їх застосування, проміжні сполуки та фармацевтична композиція |
-
1999
- 1999-06-09 FR FR9907252A patent/FR2794747B1/fr not_active Expired - Fee Related
-
2000
- 2000-06-06 TN TNTNSN00127A patent/TNSN00127A1/fr unknown
- 2000-06-07 AR ARP000102834A patent/AR024315A1/es unknown
- 2000-06-07 PE PE2000000567A patent/PE20010234A1/es not_active Application Discontinuation
- 2000-06-07 UY UY26195A patent/UY26195A1/es not_active Application Discontinuation
- 2000-06-08 GT GT200000090A patent/GT200000090A/es unknown
- 2000-06-08 WO PCT/FR2000/001569 patent/WO2000075178A1/fr active IP Right Grant
- 2000-06-08 JP JP2001502459A patent/JP4619592B2/ja not_active Expired - Fee Related
- 2000-06-08 US US10/009,407 patent/US7005417B1/en not_active Expired - Fee Related
- 2000-06-08 AU AU55391/00A patent/AU5539100A/en not_active Abandoned
- 2000-06-08 ES ES00940456T patent/ES2194744T3/es not_active Expired - Lifetime
- 2000-06-08 CA CA002376490A patent/CA2376490A1/fr not_active Abandoned
- 2000-06-08 AT AT00940456T patent/ATE240971T1/de not_active IP Right Cessation
- 2000-06-08 EP EP00940456A patent/EP1189932B1/fr not_active Expired - Lifetime
- 2000-06-08 PT PT00940456T patent/PT1189932E/pt unknown
- 2000-06-08 DE DE60002866T patent/DE60002866T2/de not_active Expired - Lifetime
- 2000-06-08 DK DK00940456T patent/DK1189932T3/da active
- 2000-06-09 CO CO00042902A patent/CO5200761A1/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| FR2794747A1 (fr) | 2000-12-15 |
| AR024315A1 (es) | 2002-09-25 |
| UY26195A1 (es) | 2001-01-31 |
| PT1189932E (pt) | 2003-09-30 |
| DK1189932T3 (da) | 2003-09-15 |
| US7005417B1 (en) | 2006-02-28 |
| FR2794747B1 (fr) | 2004-04-16 |
| DE60002866D1 (de) | 2003-06-26 |
| ES2194744T3 (es) | 2003-12-01 |
| WO2000075178A1 (fr) | 2000-12-14 |
| CA2376490A1 (fr) | 2000-12-14 |
| PE20010234A1 (es) | 2001-02-24 |
| TNSN00127A1 (fr) | 2005-11-10 |
| JP2003504309A (ja) | 2003-02-04 |
| AU5539100A (en) | 2000-12-28 |
| DE60002866T2 (de) | 2004-03-11 |
| EP1189932B1 (fr) | 2003-05-21 |
| EP1189932A1 (fr) | 2002-03-27 |
| JP4619592B2 (ja) | 2011-01-26 |
| CO5200761A1 (es) | 2002-09-27 |
| ATE240971T1 (de) | 2003-06-15 |
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