PL362173A1 - Pochodne difenyloazetydynonu, sposób ich wytwarzania, środki lecznicze zawierające te związki oraz ich zastosowanie - Google Patents

Pochodne difenyloazetydynonu, sposób ich wytwarzania, środki lecznicze zawierające te związki oraz ich zastosowanie

Info

Publication number
PL362173A1
PL362173A1 PL01362173A PL36217301A PL362173A1 PL 362173 A1 PL362173 A1 PL 362173A1 PL 01362173 A PL01362173 A PL 01362173A PL 36217301 A PL36217301 A PL 36217301A PL 362173 A1 PL362173 A1 PL 362173A1
Authority
PL
Poland
Prior art keywords
compounds
production
medicaments containing
azetidinone derivatives
diphenyl azetidinone
Prior art date
Application number
PL01362173A
Other languages
English (en)
Inventor
Heiner Glombik
Werner Kramer
Stefanie Flohr
Wendelin Frick
Hubert Heuer
Gerhard Jaehne
Andreas Lindenschmidt
Hans-Ludwig Schaefer
Original Assignee
Aventis Pharma Deutschland Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE10064402A external-priority patent/DE10064402A1/de
Priority claimed from DE2001154520 external-priority patent/DE10154520A1/de
Application filed by Aventis Pharma Deutschland Gmbh filed Critical Aventis Pharma Deutschland Gmbh
Publication of PL362173A1 publication Critical patent/PL362173A1/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
PL01362173A 2000-12-21 2001-12-11 Pochodne difenyloazetydynonu, sposób ich wytwarzania, środki lecznicze zawierające te związki oraz ich zastosowanie PL362173A1 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE10064402A DE10064402A1 (de) 2000-12-21 2000-12-21 Diphenylazetidinonderivate, Verfahren zu deren Herstellung, diese Verbindungen enthaltende Arzneimittel und deren Verwendung
DE2001154520 DE10154520A1 (de) 2001-11-07 2001-11-07 Diphenylazetidinonderivate, Verfahren zu deren Herstellung, diese Verbindungen enthaltende Arzneimittel und deren Verwendung
PCT/EP2001/014532 WO2002050068A1 (de) 2000-12-21 2001-12-11 Diphenylazetidinonderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung

Publications (1)

Publication Number Publication Date
PL362173A1 true PL362173A1 (pl) 2004-10-18

Family

ID=26008045

Family Applications (1)

Application Number Title Priority Date Filing Date
PL01362173A PL362173A1 (pl) 2000-12-21 2001-12-11 Pochodne difenyloazetydynonu, sposób ich wytwarzania, środki lecznicze zawierające te związki oraz ich zastosowanie

Country Status (24)

Country Link
US (1) US6498156B2 (pl)
EP (1) EP1345932B1 (pl)
JP (1) JP2004516293A (pl)
KR (1) KR20030061462A (pl)
CN (1) CN1222522C (pl)
AR (1) AR034282A1 (pl)
AT (1) ATE342899T1 (pl)
AU (2) AU1917302A (pl)
BR (1) BR0116482A (pl)
CA (1) CA2431985A1 (pl)
CZ (1) CZ20031731A3 (pl)
DE (1) DE50111293D1 (pl)
EE (1) EE200300237A (pl)
HK (1) HK1059936A1 (pl)
HR (1) HRP20030499A2 (pl)
HU (1) HUP0401067A2 (pl)
IL (1) IL156552A0 (pl)
MX (1) MXPA03005018A (pl)
NO (1) NO20032733L (pl)
NZ (1) NZ526592A (pl)
PL (1) PL362173A1 (pl)
SK (1) SK7812003A3 (pl)
WO (1) WO2002050068A1 (pl)
YU (1) YU46903A (pl)

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US20030119808A1 (en) * 2001-09-21 2003-06-26 Schering Corporation Methods of treating or preventing cardiovascular conditions while preventing or minimizing muscular degeneration side effects
US7056906B2 (en) 2001-09-21 2006-06-06 Schering Corporation Combinations of hormone replacement therapy composition(s) and sterol absorption inhibitor(s) and treatments for vascular conditions in post-menopausal women
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DE60216300T2 (de) * 2001-09-21 2007-06-28 Schering Corp. Behandlung von xanthom mittels azetidinon-derivate als hemmer der sterol absorption
US7176193B2 (en) 2002-06-19 2007-02-13 Sanofi-Aventis Deutschland Gmbh Acid-group-substituted diphenylazetidinones, process for their preparation, medicaments comprising these compounds, and their use
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WO2004100885A2 (en) * 2003-05-09 2004-11-25 The Trustees Of The University Of Pennsylvania Compositions and methods for treating cancer
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US8987322B2 (en) * 2003-11-04 2015-03-24 Circ Pharma Research And Development Limited Pharmaceutical formulations for carrier-mediated transport statins and uses thereof
EP1918000A2 (en) 2003-11-05 2008-05-07 Schering Corporation Combinations of lipid modulating agents and substituted azetidinones and treatments for vascular conditions
ATE485267T1 (de) 2003-12-23 2010-11-15 Astrazeneca Ab Diphenylazetidinonderivate mit die cholesterinabsorption hemmender wirkung
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EP1725234B2 (en) * 2004-03-05 2016-02-24 The Trustees of The University of Pennsylvania Methods for treating disorders or diseases associated with hyperlipidemia and hypercholesterolemia while minimizing side-effects
WO2006039334A1 (en) * 2004-09-29 2006-04-13 Schering Corporation Combinations of substituted azetidonones and cb1 antagonists
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CN101222950A (zh) * 2005-05-25 2008-07-16 迈克罗比亚公司 制备4-(联苯基)氮杂环丁-2-酮膦酸的方法
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CA2626461A1 (en) * 2005-10-18 2007-04-26 Aegerion Pharmaceuticals Compositions for lowering serum cholesterol and/or triglycerides
PE20071320A1 (es) 2006-01-18 2007-12-29 Schering Corp Moduladores de receptores cannabinoides
AR060623A1 (es) 2006-04-27 2008-07-02 Astrazeneca Ab Compuestos derivados de 2-azetidinona y un metodo de preparacion
RU2009108280A (ru) 2006-08-08 2010-09-20 Санофи-Авентис (Fr) Ариламиноарилалкилзамещенные имидазолидин-2,4-дионы, способы их получения, содержащие эти соединения лекарственные средства и их применение
JP2010502702A (ja) * 2006-09-05 2010-01-28 シェーリング コーポレイション 脂質管理およびアテローム性動脈硬化症および脂肪肝の治療治療において使用される医薬組成物
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Also Published As

Publication number Publication date
AR034282A1 (es) 2004-02-18
MXPA03005018A (es) 2003-09-25
NZ526592A (en) 2004-11-26
AU1917302A (en) 2002-07-01
CZ20031731A3 (cs) 2003-09-17
HUP0401067A2 (hu) 2004-09-28
NO20032733D0 (no) 2003-06-16
KR20030061462A (ko) 2003-07-18
BR0116482A (pt) 2004-02-03
SK7812003A3 (en) 2004-01-08
AU2002219173B2 (en) 2006-06-22
HK1059936A1 (en) 2004-07-23
HRP20030499A2 (en) 2005-04-30
CN1222522C (zh) 2005-10-12
CA2431985A1 (en) 2002-06-27
IL156552A0 (en) 2004-01-04
US20020128252A1 (en) 2002-09-12
ATE342899T1 (de) 2006-11-15
JP2004516293A (ja) 2004-06-03
YU46903A (sh) 2006-05-25
EP1345932A1 (de) 2003-09-24
EP1345932B1 (de) 2006-10-18
DE50111293D1 (de) 2006-11-30
US6498156B2 (en) 2002-12-24
NO20032733L (no) 2003-08-14
EE200300237A (et) 2003-08-15
CN1481381A (zh) 2004-03-10
WO2002050068A1 (de) 2002-06-27

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