PL2552920T3 - Nowe wybiórcze związki antagonistów receptora NK-3, farmaceutyczne kompozycje i sposoby do zastosowania w zaburzeniach pośredniczonych przez receptory NK-3 - Google Patents

Nowe wybiórcze związki antagonistów receptora NK-3, farmaceutyczne kompozycje i sposoby do zastosowania w zaburzeniach pośredniczonych przez receptory NK-3

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Publication number
PL2552920T3
PL2552920T3 PL11711922T PL11711922T PL2552920T3 PL 2552920 T3 PL2552920 T3 PL 2552920T3 PL 11711922 T PL11711922 T PL 11711922T PL 11711922 T PL11711922 T PL 11711922T PL 2552920 T3 PL2552920 T3 PL 2552920T3
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PL
Poland
Prior art keywords
novel
methods
pharmaceutical composition
mediated disorders
antagonist compounds
Prior art date
Application number
PL11711922T
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English (en)
Inventor
Hamid Hoveyda
Marie-Odile Roy
Graeme Lovat Fraser
Guillaume Dutheuil
Original Assignee
Ogeda Sa
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Publication date
Application filed by Ogeda Sa filed Critical Ogeda Sa
Publication of PL2552920T3 publication Critical patent/PL2552920T3/pl

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/4155—1,2-Diazoles non condensed and containing further heterocyclic rings
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    • A61K31/33—Heterocyclic compounds
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
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    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

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  • Diabetes (AREA)
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  • Obesity (AREA)
  • Hematology (AREA)
  • Rheumatology (AREA)
  • Pregnancy & Childbirth (AREA)
  • Oncology (AREA)
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PL11711922T 2010-04-02 2011-04-04 Nowe wybiórcze związki antagonistów receptora NK-3, farmaceutyczne kompozycje i sposoby do zastosowania w zaburzeniach pośredniczonych przez receptory NK-3 PL2552920T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP10305343 2010-04-02
US37902810P 2010-09-01 2010-09-01
EP11711922.2A EP2552920B1 (en) 2010-04-02 2011-04-04 Novel nk-3 receptor selective antagonist compounds, pharmaceutical composition and methods for use in nk-3 receptors mediated disorders

Publications (1)

Publication Number Publication Date
PL2552920T3 true PL2552920T3 (pl) 2017-08-31

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PL11711922T PL2552920T3 (pl) 2010-04-02 2011-04-04 Nowe wybiórcze związki antagonistów receptora NK-3, farmaceutyczne kompozycje i sposoby do zastosowania w zaburzeniach pośredniczonych przez receptory NK-3

Country Status (21)

Country Link
US (4) US8871761B2 (pl)
EP (2) EP2552920B1 (pl)
JP (1) JP5822911B2 (pl)
KR (1) KR101878888B1 (pl)
CN (1) CN102906093B (pl)
AU (1) AU2011234398B8 (pl)
BR (1) BR112012025101B1 (pl)
CA (1) CA2793313C (pl)
DK (1) DK2552920T3 (pl)
EA (1) EA023161B1 (pl)
ES (1) ES2627688T3 (pl)
HR (1) HRP20170712T1 (pl)
HU (1) HUE032770T2 (pl)
LT (1) LT2552920T (pl)
MX (1) MX342161B (pl)
PL (1) PL2552920T3 (pl)
PT (1) PT2552920T (pl)
RS (1) RS55997B1 (pl)
SI (1) SI2552920T1 (pl)
SM (1) SMT201700282T1 (pl)
WO (1) WO2011121137A1 (pl)

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