LT2552920T - Nauji nk-3 receptoriaus selektyvūs antagonistų junginiai, farmacinė kompozicija ir būdai, skirti naudoti nk-3 receptoriaus sąlygotų sutrikimų gydymui - Google Patents

Nauji nk-3 receptoriaus selektyvūs antagonistų junginiai, farmacinė kompozicija ir būdai, skirti naudoti nk-3 receptoriaus sąlygotų sutrikimų gydymui

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Publication number
LT2552920T
LT2552920T LTEP11711922.2T LT11711922T LT2552920T LT 2552920 T LT2552920 T LT 2552920T LT 11711922 T LT11711922 T LT 11711922T LT 2552920 T LT2552920 T LT 2552920T
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LT
Lithuania
Prior art keywords
novel
methods
pharmaceutical composition
mediated disorders
antagonist compounds
Prior art date
Application number
LTEP11711922.2T
Other languages
English (en)
Inventor
Hamid Hoveyda
Marie-Odile Roy
Graeme Lovat Fraser
Guillaume Dutheuil
Original Assignee
Ogeda Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ogeda Sa filed Critical Ogeda Sa
Publication of LT2552920T publication Critical patent/LT2552920T/lt

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    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/4155—1,2-Diazoles non condensed and containing further heterocyclic rings
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
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    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
LTEP11711922.2T 2010-04-02 2011-04-04 Nauji nk-3 receptoriaus selektyvūs antagonistų junginiai, farmacinė kompozicija ir būdai, skirti naudoti nk-3 receptoriaus sąlygotų sutrikimų gydymui LT2552920T (lt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP10305343 2010-04-02
US37902810P 2010-09-01 2010-09-01
PCT/EP2011/055218 WO2011121137A1 (en) 2010-04-02 2011-04-04 Novel nk-3 receptor selective antagonist compounds, pharmaceutical composition and methods for use in nk-3 receptors mediated disorders

Publications (1)

Publication Number Publication Date
LT2552920T true LT2552920T (lt) 2017-06-12

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LTEP11711922.2T LT2552920T (lt) 2010-04-02 2011-04-04 Nauji nk-3 receptoriaus selektyvūs antagonistų junginiai, farmacinė kompozicija ir būdai, skirti naudoti nk-3 receptoriaus sąlygotų sutrikimų gydymui

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US (4) US8871761B2 (lt)
EP (2) EP2552920B1 (lt)
JP (1) JP5822911B2 (lt)
KR (1) KR101878888B1 (lt)
CN (1) CN102906093B (lt)
AU (1) AU2011234398B8 (lt)
BR (1) BR112012025101B1 (lt)
CA (1) CA2793313C (lt)
DK (1) DK2552920T3 (lt)
EA (1) EA023161B1 (lt)
ES (1) ES2627688T3 (lt)
HR (1) HRP20170712T1 (lt)
HU (1) HUE032770T2 (lt)
LT (1) LT2552920T (lt)
MX (1) MX342161B (lt)
PL (1) PL2552920T3 (lt)
PT (1) PT2552920T (lt)
RS (1) RS55997B1 (lt)
SI (1) SI2552920T1 (lt)
WO (1) WO2011121137A1 (lt)

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