PL122152B1 - Process for preparing derivatives of 3-/thiomethyl/ cephalosporinsnov - Google Patents

Process for preparing derivatives of 3-/thiomethyl/ cephalosporinsnov Download PDF

Info

Publication number
PL122152B1
PL122152B1 PL1978205135A PL20513578A PL122152B1 PL 122152 B1 PL122152 B1 PL 122152B1 PL 1978205135 A PL1978205135 A PL 1978205135A PL 20513578 A PL20513578 A PL 20513578A PL 122152 B1 PL122152 B1 PL 122152B1
Authority
PL
Poland
Prior art keywords
methyl
acid
product
acetamido
group
Prior art date
Application number
PL1978205135A
Other languages
English (en)
Polish (pl)
Other versions
PL205135A1 (pl
Inventor
Deii Hatsutofuiirudo Rooeru
Original Assignee
Eli Lilly And Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/862,871 external-priority patent/US4144391A/en
Application filed by Eli Lilly And Co filed Critical Eli Lilly And Co
Publication of PL205135A1 publication Critical patent/PL205135A1/xx
Publication of PL122152B1 publication Critical patent/PL122152B1/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/36—Methylene radicals, substituted by sulfur atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PL1978205135A 1977-03-07 1978-03-07 Process for preparing derivatives of 3-/thiomethyl/ cephalosporinsnov PL122152B1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US77501877A 1977-03-07 1977-03-07
US05/862,871 US4144391A (en) 1977-03-07 1977-12-27 Cephalosporin displacement reaction

Publications (2)

Publication Number Publication Date
PL205135A1 PL205135A1 (pl) 1979-06-04
PL122152B1 true PL122152B1 (en) 1982-06-30

Family

ID=27118982

Family Applications (1)

Application Number Title Priority Date Filing Date
PL1978205135A PL122152B1 (en) 1977-03-07 1978-03-07 Process for preparing derivatives of 3-/thiomethyl/ cephalosporinsnov

Country Status (30)

Country Link
JP (1) JPS53130689A (en, 2012)
AT (1) AT366696B (en, 2012)
AU (1) AU515428B2 (en, 2012)
BG (1) BG31379A3 (en, 2012)
CA (1) CA1083141A (en, 2012)
CH (1) CH637964A5 (en, 2012)
CS (1) CS205115B2 (en, 2012)
CY (1) CY1196A (en, 2012)
DD (1) DD137356A5 (en, 2012)
DE (1) DE2809058A1 (en, 2012)
DK (1) DK97378A (en, 2012)
EG (1) EG13454A (en, 2012)
ES (1) ES467637A1 (en, 2012)
FI (1) FI69309C (en, 2012)
FR (1) FR2383189A1 (en, 2012)
GB (1) GB1597036A (en, 2012)
GR (1) GR68893B (en, 2012)
HK (1) HK49083A (en, 2012)
HU (1) HU179967B (en, 2012)
IE (1) IE46437B1 (en, 2012)
IL (1) IL54181A (en, 2012)
IT (1) IT1093504B (en, 2012)
MX (1) MX5142E (en, 2012)
NL (1) NL190703C (en, 2012)
NZ (1) NZ186610A (en, 2012)
PH (1) PH14596A (en, 2012)
PL (1) PL122152B1 (en, 2012)
PT (1) PT67732A (en, 2012)
SE (1) SE437991B (en, 2012)
YU (1) YU51478A (en, 2012)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5543043A (en) * 1978-09-22 1980-03-26 Sankyo Co Ltd Preparation of 3-substituted thiomethylcephalosporin derivative
US4576937A (en) * 1984-02-29 1986-03-18 Smithkline Beckman Corporation 7-D-Mandelamido-3(1-sulfomethyltetrazol-5-yl)thiomethyl-3-cephem-4-carboxylic acid monosodium salt
GB8519606D0 (en) * 1985-08-05 1985-09-11 Fujisawa Pharmaceutical Co 3 7-d substituted-3-cephem compounds
JP2503500B2 (ja) * 1986-04-14 1996-06-05 萬有製薬株式会社 新規セフアロスポリン誘導体及びその製造法
JPS62281881A (ja) * 1986-09-08 1987-12-07 Sankyo Co Ltd ３−置換チオメチルセフアロスポリン誘導体の製法
US20120329770A1 (en) * 2010-02-26 2012-12-27 Gary Igor Dmitrienko Cephalosporin derivatives useful as beta-lactamase inhibitors and compositions and methods of use thereof
GB201818410D0 (en) * 2018-11-12 2018-12-26 Imperial Innovations Ltd Compounds
CN114728008A (zh) * 2019-08-29 2022-07-08 加利福尼亚大学董事会 鉴定β-内酰胺酶的化合物及其使用方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3641021A (en) * 1969-04-18 1972-02-08 Lilly Co Eli 3 7-(ring-substituted) cephalosporin compounds
JPS5116436B1 (en, 2012) * 1971-05-31 1976-05-24
JPS5143785A (en) * 1974-10-11 1976-04-14 Yamanouchi Pharma Co Ltd Shinsefuarosuhorinkanrenkagobutsuno goseiho
JPS612674B2 (en, 2012) * 1974-06-20 1986-01-27 Meiji Seika Co
CA1100129A (en) * 1974-08-02 1981-04-28 William H.W. Lunn Cephalosporin compounds
FI761035A7 (en, 2012) * 1975-04-21 1976-10-22 Erba Carlo Spa

Also Published As

Publication number Publication date
BG31379A3 (bg) 1981-12-15
FI69309C (fi) 1986-01-10
CS205115B2 (en) 1981-04-30
CY1196A (en) 1983-12-31
FR2383189B1 (en, 2012) 1981-06-26
DK97378A (da) 1978-09-08
ATA150778A (de) 1981-09-15
YU51478A (en) 1982-10-31
CA1083141A (en) 1980-08-05
PH14596A (en) 1981-10-02
AT366696B (de) 1982-04-26
JPH025758B2 (en, 2012) 1990-02-05
IE46437B1 (en) 1983-06-15
FI69309B (fi) 1985-09-30
IT1093504B (it) 1985-07-19
PT67732A (en) 1978-04-01
DE2809058C2 (en, 2012) 1989-02-09
HU179967B (en) 1983-01-28
FI780716A7 (fi) 1978-09-08
AU3382878A (en) 1979-09-06
IL54181A0 (en) 1978-06-15
IT7820912A0 (it) 1978-03-06
ES467637A1 (es) 1980-04-01
MX5142E (es) 1983-03-30
AU515428B2 (en) 1981-04-02
JPS53130689A (en) 1978-11-14
IL54181A (en) 1981-03-31
DE2809058A1 (de) 1978-09-14
NL190703C (nl) 1994-07-01
SE437991B (sv) 1985-03-25
FR2383189A1 (fr) 1978-10-06
IE780453L (en) 1978-09-07
PL205135A1 (pl) 1979-06-04
GB1597036A (en) 1981-09-03
HK49083A (en) 1983-11-04
CH637964A5 (en) 1983-08-31
NL190703B (nl) 1994-02-01
NL7802376A (nl) 1978-09-11
GR68893B (en, 2012) 1982-03-15
DD137356A5 (de) 1979-08-29
SE7802530L (sv) 1978-09-08
EG13454A (en) 1981-12-31
NZ186610A (en) 1979-11-01

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