PH23584A - Piperidine compounds and pharmaceutical compositions containing the same - Google Patents
Piperidine compounds and pharmaceutical compositions containing the sameInfo
- Publication number
- PH23584A PH23584A PH35635A PH35635A PH23584A PH 23584 A PH23584 A PH 23584A PH 35635 A PH35635 A PH 35635A PH 35635 A PH35635 A PH 35635A PH 23584 A PH23584 A PH 23584A
- Authority
- PH
- Philippines
- Prior art keywords
- piperidine compounds
- same
- pharmaceutical compositions
- compositions containing
- chem
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Cephalosporin Compounds (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DK426986A DK426986D0 (da) | 1986-09-08 | 1986-09-08 | Piperidine forbindelser, deres fremstilling og anvendelse |
DK597186A DK597186D0 (da) | 1986-12-12 | 1986-12-12 | Heterocykliske forbindelser, deres fremstilling og anvendelse |
Publications (1)
Publication Number | Publication Date |
---|---|
PH23584A true PH23584A (en) | 1989-09-11 |
Family
ID=26067417
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PH35635A PH23584A (en) | 1986-09-08 | 1987-08-06 | Piperidine compounds and pharmaceutical compositions containing the same |
Country Status (17)
Country | Link |
---|---|
US (2) | US4837241A (no) |
EP (1) | EP0259621B1 (no) |
JP (1) | JPH0662616B2 (no) |
KR (1) | KR950009366B1 (no) |
AT (1) | ATE82751T1 (no) |
AU (1) | AU603603B2 (no) |
CA (1) | CA1340937C (no) |
DE (1) | DE3782785T2 (no) |
ES (1) | ES2043624T3 (no) |
FI (1) | FI86424C (no) |
GR (1) | GR3007053T3 (no) |
IE (1) | IE62485B1 (no) |
IL (1) | IL83275A (no) |
NO (1) | NO169285C (no) |
NZ (1) | NZ221672A (no) |
PH (1) | PH23584A (no) |
PT (1) | PT85650B (no) |
Families Citing this family (41)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NZ219646A (en) * | 1986-03-27 | 1990-10-26 | Merck Sharp & Dohme | Oxadiazole derivatives of azacyclics for treating cns disorders |
GB8714789D0 (en) * | 1987-06-24 | 1987-07-29 | Lundbeck & Co As H | Heterocyclic compounds |
IE63906B1 (en) * | 1987-11-13 | 1995-06-14 | Novo Nordisk As | Azabicyclic compounds and their preparation and use |
EP0322034A3 (en) * | 1987-12-22 | 1991-01-02 | Merck Sharp & Dohme Ltd. | Methyl tetrahydropyridyl oxadiazoles |
IL88846A0 (en) * | 1988-01-08 | 1989-07-31 | Merck Sharp & Dohme | Lipophilic oxadiazoles,their preparation and pharmaceutical compositions containing them |
DK162892C (da) * | 1988-07-04 | 1992-05-11 | Novo Nordisk As | 1,2,5,6-tetrahydropyridinforbindelser, deres fremstilling og farmaceutiske praeparater indeholdende disse |
US5328925A (en) * | 1989-02-22 | 1994-07-12 | Novo Nordisk A/S | Piperidine compounds and their use |
US5043345A (en) * | 1989-02-22 | 1991-08-27 | Novo Nordisk A/S | Piperidine compounds and their preparation and use |
US5264444A (en) * | 1989-02-22 | 1993-11-23 | Novo Nordisk A/S | Piperidine compounds and use |
US5260311A (en) * | 1989-02-22 | 1993-11-09 | Novo Nordisk A/S | Piperidine compounds and their use |
EP0459568A3 (en) * | 1990-05-31 | 1992-09-30 | Merck Sharp & Dohme Ltd. | Substituted oxadiazoles and thiadiazoles for use in the treatment of glaucoma and novel compounds having such use |
MX9100517A (es) * | 1990-08-06 | 1992-04-01 | Smith Kline French Lab | Compuestos |
DK198490D0 (da) * | 1990-08-21 | 1990-08-21 | Novo Nordisk As | Heterocykliske forbindelser, deres fremstilling og anvendelse |
ES2113939T3 (es) * | 1990-11-29 | 1998-05-16 | Allergan Inc | Uso de derivados de piridina en el tratamiento de la hipertension ocular. |
US5175166A (en) * | 1991-08-27 | 1992-12-29 | The University Of Toledo | Muscarinic agonists |
EP0619814A1 (en) * | 1991-12-31 | 1994-10-19 | Fujisawa Pharmaceutical Co., Ltd. | Oxadiazole derivatives having acetylcholinesterase-inhibitory and muscarinic agonist activity |
US5424301A (en) * | 1993-02-01 | 1995-06-13 | Warner-Lambert Company | Starch stabilized o-substituted tetrahydropyridine oxime cholinergic agents |
DK0637586T3 (da) * | 1993-08-05 | 1999-12-06 | Hoechst Marion Roussel Inc | 2-(Piperidin-4-yl, pyridin-4-yl og tetrahydropyridin-4-yl)-benzofuran-7-carbamatderivater, deres fremstilling og anvendelse |
US5753683A (en) * | 1993-08-19 | 1998-05-19 | Novo Nordisk A/S | Antipsychotic method |
US5998404A (en) * | 1994-10-24 | 1999-12-07 | Eli Lilly And Company | Heterocyclic compounds and their use |
US5672709A (en) * | 1994-10-24 | 1997-09-30 | Eli Lilly And Company | Heterocyclic compounds and their preparation and use |
US5605908A (en) * | 1994-10-24 | 1997-02-25 | Eli Lilly And Company | Heterocyclic compounds and their use |
US5726193A (en) * | 1994-10-31 | 1998-03-10 | Eli Lilly And Company | Method for treating anxiety |
US5488056A (en) * | 1994-10-31 | 1996-01-30 | Eli Lilly And Company | Method for treating anxiety |
US5574028A (en) * | 1994-10-31 | 1996-11-12 | Eli Lilly And Company | Method for treating anxiety |
US6297262B1 (en) | 1997-05-29 | 2001-10-02 | H. Lundbeck A/S | Treatment of schizophrenia and psychosis |
AU2307899A (en) * | 1997-12-23 | 1999-07-12 | Alcon Laboratories, Inc. | Muscarinic agents and use thereof to treat glaucoma, myopia and various other conditions |
US6107313A (en) * | 1998-10-02 | 2000-08-22 | Combichem, Inc. | Dopamine receptor antagonists |
US7332508B2 (en) * | 2002-12-18 | 2008-02-19 | Novo Nordisk A/S | Substituted homopiperidine, piperidine or pyrrolidine derivatives |
RU2381226C2 (ru) * | 2004-02-18 | 2010-02-10 | Астразенека Аб | Полигетероциклические соединения и их применение в качестве антагонистов метаботропного рецептора глутамата |
EP1720874A4 (en) * | 2004-02-24 | 2010-03-03 | Bioaxone Therapeutique Inc | SUBSTITUTED PIPERIDINE DERIVATIVES IN POSITION 4 |
RU2446166C2 (ru) * | 2007-04-24 | 2012-03-27 | Солвей Фармасьютикалс Б.В. | Гетероциклические соединения, имеющие сродство к мускариновым рецепторам |
US8084473B2 (en) | 2007-04-24 | 2011-12-27 | Solvay Pharmaceuticals B.V. | Heterocyclic compounds with affinity to muscarinic receptors |
WO2009140483A1 (en) | 2008-05-15 | 2009-11-19 | University Of Toledo | Muscarinic agonists as cognitive enhancers |
US9549928B2 (en) | 2011-04-29 | 2017-01-24 | The University Of Toledo | Muscarinic agonists as enhancers of cognitive flexibility |
US10149856B2 (en) | 2015-01-26 | 2018-12-11 | BioAxone BioSciences, Inc. | Treatment of cerebral cavernous malformations and cerebral aneurysms with rho kinase inhibitors |
US10857157B2 (en) | 2015-01-26 | 2020-12-08 | BioAxone BioSciences, Inc. | Treatment of cerebral cavernous malformations and cerebral aneurysms with rho kinase inhibitors |
US10106525B2 (en) | 2015-01-26 | 2018-10-23 | BioAxone BioSciences, Inc. | Rho kinase inhibitor BA-1049 (R) and active metabolites thereof |
US11198680B2 (en) | 2016-12-21 | 2021-12-14 | BioAxone BioSciences, Inc. | Rho kinase inhibitor BA-1049 (R) and active metabolites thereof |
WO2019014322A1 (en) | 2017-07-11 | 2019-01-17 | BioAxone BioSciences, Inc. | KINASE INHIBITORS FOR THE TREATMENT OF DISEASES |
US20220152005A1 (en) * | 2019-04-04 | 2022-05-19 | Andrew Coop | Methods of using muscarinic antagonists in the treatment of depression |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3966748A (en) * | 1975-05-08 | 1976-06-29 | American Cyanamid Company | Para-fluorophenyl-N-heterocyclic substituted butanes |
US4518601A (en) * | 1982-06-16 | 1985-05-21 | Ciba Geigy Corporation | 2-(3-Pyridyl)-1,3,4-oxadiazoles and use thereof in pest control |
NZ219646A (en) * | 1986-03-27 | 1990-10-26 | Merck Sharp & Dohme | Oxadiazole derivatives of azacyclics for treating cns disorders |
-
1987
- 1987-07-21 IL IL8327587A patent/IL83275A/en unknown
- 1987-08-06 PH PH35635A patent/PH23584A/en unknown
- 1987-08-07 ES ES87111470T patent/ES2043624T3/es not_active Expired - Lifetime
- 1987-08-07 AT AT87111470T patent/ATE82751T1/de not_active IP Right Cessation
- 1987-08-07 DE DE8787111470T patent/DE3782785T2/de not_active Expired - Fee Related
- 1987-08-07 EP EP87111470A patent/EP0259621B1/en not_active Expired - Lifetime
- 1987-08-14 IE IE217387A patent/IE62485B1/en not_active IP Right Cessation
- 1987-08-26 US US07/089,747 patent/US4837241A/en not_active Expired - Lifetime
- 1987-09-02 FI FI873809A patent/FI86424C/fi not_active IP Right Cessation
- 1987-09-03 PT PT85650A patent/PT85650B/pt not_active IP Right Cessation
- 1987-09-04 NZ NZ221672A patent/NZ221672A/xx unknown
- 1987-09-07 NO NO873731A patent/NO169285C/no not_active IP Right Cessation
- 1987-09-08 KR KR1019870009915A patent/KR950009366B1/ko not_active IP Right Cessation
- 1987-09-08 CA CA000546359A patent/CA1340937C/en not_active Expired - Fee Related
- 1987-09-08 JP JP62223199A patent/JPH0662616B2/ja not_active Expired - Lifetime
- 1987-09-08 AU AU78165/87A patent/AU603603B2/en not_active Ceased
-
1988
- 1988-08-25 US US07/236,550 patent/US4933353A/en not_active Expired - Fee Related
-
1993
- 1993-02-11 GR GR930400285T patent/GR3007053T3/el unknown
Also Published As
Publication number | Publication date |
---|---|
NZ221672A (en) | 1990-09-26 |
NO873731L (no) | 1988-03-09 |
GR3007053T3 (no) | 1993-07-30 |
AU603603B2 (en) | 1990-11-22 |
DE3782785T2 (de) | 1993-04-01 |
US4933353A (en) | 1990-06-12 |
FI873809A0 (fi) | 1987-09-02 |
IE62485B1 (en) | 1995-02-08 |
FI86424B (fi) | 1992-05-15 |
NO169285B (no) | 1992-02-24 |
JPH0662616B2 (ja) | 1994-08-17 |
EP0259621A2 (en) | 1988-03-16 |
EP0259621A3 (en) | 1988-10-12 |
NO169285C (no) | 1992-06-03 |
EP0259621B1 (en) | 1992-11-25 |
KR950009366B1 (ko) | 1995-08-21 |
US4837241A (en) | 1989-06-06 |
PT85650A (en) | 1987-10-01 |
AU7816587A (en) | 1988-03-31 |
IL83275A0 (en) | 1987-12-31 |
ES2043624T3 (es) | 1994-01-01 |
CA1340937C (en) | 2000-03-28 |
IE872173L (en) | 1989-03-08 |
NO873731D0 (no) | 1987-09-07 |
ATE82751T1 (de) | 1992-12-15 |
DE3782785D1 (de) | 1993-01-07 |
FI873809A (fi) | 1988-03-09 |
PT85650B (pt) | 1990-05-31 |
FI86424C (fi) | 1992-08-25 |
IL83275A (en) | 1994-02-27 |
JPS6377877A (ja) | 1988-04-08 |
KR880003939A (ko) | 1988-06-01 |
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