PH15368A - 2(2-(2-aminothiazol-4-yl)-2-alkoxyimino)acetamido-3(4-alkyl-5-oxo-6-hydroxy-4,5-dihydro-1,2,4-triazin-3-yl)trio methyl cephalosporins - Google Patents

2(2-(2-aminothiazol-4-yl)-2-alkoxyimino)acetamido-3(4-alkyl-5-oxo-6-hydroxy-4,5-dihydro-1,2,4-triazin-3-yl)trio methyl cephalosporins

Info

Publication number
PH15368A
PH15368A PH21906A PH21906A PH15368A PH 15368 A PH15368 A PH 15368A PH 21906 A PH21906 A PH 21906A PH 21906 A PH21906 A PH 21906A PH 15368 A PH15368 A PH 15368A
Authority
PH
Philippines
Prior art keywords
aminothiazol
alkoxyimino
trio
triazin
acetamido
Prior art date
Application number
PH21906A
Other languages
English (en)
Inventor
Allen Samuel Kather
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of PH15368A publication Critical patent/PH15368A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/36—Methylene radicals, substituted by sulfur atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PH21906A 1977-12-20 1978-12-07 2(2-(2-aminothiazol-4-yl)-2-alkoxyimino)acetamido-3(4-alkyl-5-oxo-6-hydroxy-4,5-dihydro-1,2,4-triazin-3-yl)trio methyl cephalosporins PH15368A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/862,318 US4200745A (en) 1977-12-20 1977-12-20 7[2-(2-Aminothiazol-4-yl)-2-alkoxyimino]acetamido 3[4-alkyl-5-oxo-6-hydroxy-3,4 dihydro 1,2,4-triazin 3-yl]thio methyl cephalosporins

Publications (1)

Publication Number Publication Date
PH15368A true PH15368A (en) 1982-12-10

Family

ID=25338200

Family Applications (1)

Application Number Title Priority Date Filing Date
PH21906A PH15368A (en) 1977-12-20 1978-12-07 2(2-(2-aminothiazol-4-yl)-2-alkoxyimino)acetamido-3(4-alkyl-5-oxo-6-hydroxy-4,5-dihydro-1,2,4-triazin-3-yl)trio methyl cephalosporins

Country Status (33)

Country Link
US (1) US4200745A (cs)
EP (1) EP0002605B1 (cs)
JP (1) JPS5490194A (cs)
AR (1) AR220733A1 (cs)
AT (1) AT364189B (cs)
AU (1) AU518484B2 (cs)
BE (1) BE872616A (cs)
CA (1) CA1140112A (cs)
CH (1) CH635846A5 (cs)
CS (1) CS204957B2 (cs)
DD (1) DD139857A5 (cs)
DE (1) DE2861493D1 (cs)
DK (1) DK540278A (cs)
EG (1) EG13666A (cs)
ES (1) ES476154A1 (cs)
FI (1) FI67083C (cs)
FR (1) FR2412553A1 (cs)
GB (1) GB2010256B (cs)
GR (1) GR72240B (cs)
HU (1) HU181875B (cs)
IE (1) IE47696B1 (cs)
IL (1) IL56166A0 (cs)
IT (1) IT1112300B (cs)
LU (1) LU80669A1 (cs)
MX (1) MX5586E (cs)
NZ (1) NZ189121A (cs)
PH (1) PH15368A (cs)
PL (1) PL123368B1 (cs)
PT (1) PT68888A (cs)
RO (1) RO75804A (cs)
SU (1) SU793403A3 (cs)
YU (1) YU300278A (cs)
ZA (1) ZA787110B (cs)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5760345B2 (cs) * 1974-12-19 1982-12-18 Takeda Chemical Industries Ltd
CH641468A5 (de) * 1978-05-30 1984-02-29 Hoffmann La Roche Cephemderivate.
MC1259A1 (fr) * 1978-05-30 1980-01-14 Hoffmann La Roche Derives acyles
ZA806977B (en) * 1979-11-19 1981-10-28 Fujisawa Pharmaceutical Co 7-acylamino-3-vinylcephalosporanic acid derivatives and processes for the preparation thereof
FI67385C (fi) * 1979-11-21 1985-03-11 Hoffmann La Roche Foerfarande foer framstaellning av (6r 7r)-7-(2-(2-amino-4-tiazolyl)-2-(z-metoxiimino)acetamido)-3-cefem-4-karboxylsyraderivat
US4349672A (en) * 1979-11-29 1982-09-14 Hoffmann-La Roche Inc. Cephalosporin derivatives
US4409387A (en) * 1979-11-29 1983-10-11 Hoffmann-La Roche Inc. Cephalosporin derivatives
NZ196552A (en) * 1980-03-25 1984-07-06 Hoffmann La Roche Cephalosporin derivatives and pharmaceutical compositions;intermediate cephalosporins
GR75706B (cs) * 1980-06-30 1984-08-02 Sanofi Sa
DK379581A (da) * 1980-10-06 1982-04-07 Hoffmann La Roche Fremgangsmaade til fremstilling af acylderivater
FR2494278A1 (fr) * 1980-11-20 1982-05-21 Rhone Poulenc Ind Nouveaux derives de la cephalosporine, leurs preparations et les medicaments qui les contiennent
US4698338A (en) * 1986-02-19 1987-10-06 Eli Lilly And Company 7[2-(2-aminothiazol-4-yl)-2-benzyloximino]acetamido-3[4-alkyl-5-oxo-6-hydroxy-3,4-dihydro-1,2,4-triazin-3-yl]thiomethyl cephalosporins

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1100129A (en) * 1974-08-02 1981-04-28 William H.W. Lunn Cephalosporin compounds
GR63088B (en) * 1976-04-14 1979-08-09 Takeda Chemical Industries Ltd Preparation process of novel cephalosporins
NL7805715A (nl) * 1977-06-03 1978-12-05 Hoffmann La Roche Werkwijze voor het bereiden van acylderivaten.

Also Published As

Publication number Publication date
AT364189B (de) 1981-09-25
GB2010256A (en) 1979-06-27
IT7831016A0 (it) 1978-12-19
FR2412553A1 (fr) 1979-07-20
CH635846A5 (fr) 1983-04-29
ATA908378A (de) 1981-02-15
ZA787110B (en) 1980-08-27
IE782502L (en) 1979-06-20
HU181875B (en) 1983-11-28
MX5586E (es) 1983-10-28
EP0002605A1 (en) 1979-06-27
DK540278A (da) 1979-06-21
DE2861493D1 (en) 1982-02-18
LU80669A1 (fr) 1979-04-13
IE47696B1 (en) 1984-05-30
RO75804A (ro) 1981-02-28
CA1140112A (en) 1983-01-25
GR72240B (cs) 1983-10-03
IT1112300B (it) 1986-01-13
GB2010256B (en) 1982-09-08
YU300278A (en) 1982-10-31
EG13666A (en) 1983-12-31
AU518484B2 (en) 1981-10-01
FI67083C (fi) 1985-01-10
EP0002605B1 (en) 1981-12-30
PL123368B1 (en) 1982-10-30
FR2412553B1 (cs) 1982-10-15
PL211973A1 (cs) 1980-03-10
FI67083B (fi) 1984-09-28
NZ189121A (en) 1984-02-03
JPS5490194A (en) 1979-07-17
CS204957B2 (en) 1981-04-30
AU4234778A (en) 1979-06-28
SU793403A3 (ru) 1980-12-30
FI783846A (fi) 1979-06-21
ES476154A1 (es) 1980-05-16
AR220733A1 (es) 1980-11-28
BE872616A (fr) 1979-06-08
US4200745A (en) 1980-04-29
IL56166A0 (en) 1979-03-12
DD139857A5 (de) 1980-01-23
PT68888A (en) 1979-01-01

Similar Documents

Publication Publication Date Title
AU539519B2 (en) 7(2-(2-aminothiazol-4-yl)-2(2-carboxyprop-2-oxyimino) acteamido)-3-(1-pyridiniumethyl)ceph 3-em-4-carboxylate
ZA834467B (en) 2-(4-pyridyl)-thiazole derivatives
PH23284A (en) 7-/2-(2-aminothiazol-4-yl)-2-(syn)-methoxyimino acetamido/ cephalosporin derivative
DE59100424D1 (de) Massen der allgemeinen formel mo12pavbx1cx2dx3esbfregshon.
IL73293A (en) Methyl 2-(alkanamidoalkylsulfonic)ethylthiophosphonate derivatives
DE3382601D1 (en) 2-(2-substituierte benzoyl)-1,3 cyclohexandione.
JPS5791980A (en) 2,4-disubstituted thiazole derivatives
JPS6425768A (en) 2-(2-amino-4-thiazolyl)-2-methoxyiminoacetic acid derivative and manufacture
IL70045A0 (en) Fused,5,6,5-membered heterocyclic electroactive polymers
PH15368A (en) 2(2-(2-aminothiazol-4-yl)-2-alkoxyimino)acetamido-3(4-alkyl-5-oxo-6-hydroxy-4,5-dihydro-1,2,4-triazin-3-yl)trio methyl cephalosporins
AU535320B2 (en) 2-(2-(1,4-benzodioxanyl))-2-imidazoling derivatives
FI880371A0 (fi) Foerfarande foer framstaellning av 4-aryl-n-/2-(dialkylamino- och heterocykliska -amino) alkyl/-1-piperazin-karboxaminer.
GB2083461B (en) 7-beta-(alpha-syn-methoxyimino-alpha-(2-aminothiazol-4-yl)-acetamido)-3-((1,2,3-thiadiazol-5-ylthio)methyl)-3-cephem-4-carboxylic acid and c1-c6 alkyl derivatives thereof
EP0131006A4 (en) ESTER MADE OF 3- (3-SUBSTITUTED AMINO-2-HYDROXYPROPOXY) -4-SUBSTITUTED 2,5-THIADIAZOLE COMBEDS.
ES503562A0 (es) Procedimiento de preparacion de 3-(1,2,4-hidroxitriazinil) tiometil cefalosporinas
AU522242B2 (en) 3-(TETRAZOL-5-yl)-1 AZAXANTHONES
GB2058051B (en) 4,5-substituted o-aminophenol compounds
GR64418B (en) Method for the preparation of new 2,5-dihydro-1,2-thiazono(5,6-b)indal-3-carboxamid-1,1-dioxide
GB8804454D0 (en) 3-(2-haloalkyl)-1 4-oxathiins & 2-(2-haloalkyl)-1 4-dithins
PH15598A (en) 5-(optionally substituted phenyl)-6h-1,3,4-thiadiazine-2-amines
AU3464378A (en) Preparation of 2-(2',2',2'-trihalocendethyl)-4-halogenocyclobutan-1-ones
ZA804555B (en) 5-(optionally substituted phenyl)-6h-1,3,4-thiadiazine-2-amines
FI800106A (fi) Foerfarande foer separering av d,1 2-(6-metoxi-2-naftyl)propionsyra
FI833056A0 (fi) Foerfarande foer framstaellning av kristallina former av syra-additionssalter av syn-isomer-e-formeav 7-/2-(2-amino-4-tiazolyl)-2-metoxi-imino/asetamido/-2-karboxy-3-/5,6-dioxo-4-formylmetyl-1,4,5,6-tetrahydro-1,2,4-triazin-3-yl)-2-tiovinyl/-8-oxo-5-tia-1-azab icyklo/4.2.0
PT68627A (en) Process for the preparation of 2-(2-furoyl)-1,4-dimethyl-pyridinium iodide