PH12015501056A1 - 2-pyridone compound - Google Patents

2-pyridone compound

Info

Publication number
PH12015501056A1
PH12015501056A1 PH12015501056A PH12015501056A PH12015501056A1 PH 12015501056 A1 PH12015501056 A1 PH 12015501056A1 PH 12015501056 A PH12015501056 A PH 12015501056A PH 12015501056 A PH12015501056 A PH 12015501056A PH 12015501056 A1 PH12015501056 A1 PH 12015501056A1
Authority
PH
Philippines
Prior art keywords
compound
pyridone compound
tautomer
pyridone
solvate
Prior art date
Application number
PH12015501056A
Other languages
English (en)
Other versions
PH12015501056B1 (en
Inventor
Kuroda Shoichi
Imai Yudai
Kawaguchi Takanori
Fusegi Keiko
Bohno Masahiro
Asanuma Hajime
Chonan Tomomichi
Sato Nagaaki
Monma Souichi
Sasako Shigetada
Mizutani Marie
Itoh Shin
Okada Takumi
Ota Hirofumi
Ishiyama Seishi
Original Assignee
Taisho Pharmaceutical Co Ltd
Nissan Chemical Ind Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Taisho Pharmaceutical Co Ltd, Nissan Chemical Ind Ltd filed Critical Taisho Pharmaceutical Co Ltd
Publication of PH12015501056A1 publication Critical patent/PH12015501056A1/en
Publication of PH12015501056B1 publication Critical patent/PH12015501056B1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Child & Adolescent Psychology (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
PH12015501056A 2012-11-13 2015-05-12 2-pyridone compound PH12015501056B1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2012249792 2012-11-13
PCT/JP2013/080517 WO2014077235A1 (ja) 2012-11-13 2013-11-12 2-ピリドン化合物

Publications (2)

Publication Number Publication Date
PH12015501056A1 true PH12015501056A1 (en) 2015-07-27
PH12015501056B1 PH12015501056B1 (en) 2015-07-27

Family

ID=50731146

Family Applications (1)

Application Number Title Priority Date Filing Date
PH12015501056A PH12015501056B1 (en) 2012-11-13 2015-05-12 2-pyridone compound

Country Status (25)

Country Link
US (1) US9695148B2 (enExample)
EP (1) EP2921489B1 (enExample)
JP (1) JP5963025B2 (enExample)
KR (1) KR102160841B1 (enExample)
CN (1) CN104768944B (enExample)
AU (1) AU2013345930B2 (enExample)
BR (1) BR112015010823A2 (enExample)
CA (1) CA2891406C (enExample)
DK (1) DK2921489T3 (enExample)
ES (1) ES2641469T3 (enExample)
HU (1) HUE034557T2 (enExample)
IL (1) IL238701B (enExample)
IN (1) IN2015DN03869A (enExample)
MX (1) MX361479B (enExample)
MY (1) MY173812A (enExample)
NO (1) NO2921489T3 (enExample)
NZ (1) NZ707832A (enExample)
PH (1) PH12015501056B1 (enExample)
PL (1) PL2921489T3 (enExample)
PT (1) PT2921489T (enExample)
RU (1) RU2662157C2 (enExample)
SG (1) SG11201503716RA (enExample)
TW (1) TWI591064B (enExample)
WO (1) WO2014077235A1 (enExample)
ZA (1) ZA201503323B (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP6048533B2 (ja) * 2014-05-12 2016-12-21 日産化学工業株式会社 2−ピリドン化合物を含有する医薬
CN106573909A (zh) * 2014-05-13 2017-04-19 日产化学工业株式会社 2‑吡啶酮化合物的制造方法
CA3101832A1 (en) * 2018-05-31 2019-12-05 Hua Medicine (Shanghai) Ltd. Pharmaceutical combination, composition and formulation containing glucokinase activator and a-glucosidase inhibitor, preparation methods and uses thereof

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4275069A (en) 1979-01-22 1981-06-23 The Upjohn Company Anti-diabetic 1,2-dihydro-2-oxo-6-alkyl-nicotinic acids
MXPA01009814A (es) 1999-03-29 2002-04-24 Hoffmann La Roche Activadores de la glucoquinasa.
US6353111B1 (en) 1999-12-15 2002-03-05 Hoffmann-La Roche Inc. Trans olefinic glucokinase activators
PL2076502T3 (pl) 2006-06-08 2011-09-30 Lilly Co Eli Podstawione karboksyamidy jako antagoniści receptorów metabotropowych grupy I
WO2008079787A2 (en) 2006-12-20 2008-07-03 Takeda San Diego, Inc. Glucokinase activators
TW200904440A (en) * 2007-07-17 2009-02-01 Bristol Myers Squibb Co Method for modulating GPR119 G protein-coupled receptor and selected compounds
JP2011529483A (ja) 2008-07-29 2011-12-08 ファイザー・インク フッ素化ヘテロアリール
RU2551847C2 (ru) 2009-12-04 2015-05-27 Тайсо Фармасьютикал Ко., Лтд. Производные 2-пиридона
JP2013010750A (ja) * 2011-06-02 2013-01-17 Taisho Pharmaceutical Co Ltd 2−ピリドン化合物を含有する医薬

Also Published As

Publication number Publication date
CA2891406C (en) 2021-03-16
MX361479B (es) 2018-12-06
WO2014077235A1 (ja) 2014-05-22
EP2921489A1 (en) 2015-09-23
CA2891406A1 (en) 2014-05-22
PT2921489T (pt) 2017-12-01
TWI591064B (zh) 2017-07-11
NO2921489T3 (enExample) 2018-02-03
IN2015DN03869A (enExample) 2015-10-02
PL2921489T3 (pl) 2018-01-31
NZ707832A (en) 2019-03-29
HUE034557T2 (en) 2018-02-28
US20160289208A1 (en) 2016-10-06
TW201434826A (zh) 2014-09-16
MY173812A (en) 2020-02-24
HK1207856A1 (en) 2016-02-12
US9695148B2 (en) 2017-07-04
IL238701B (en) 2018-10-31
AU2013345930B2 (en) 2017-08-24
AU2013345930A1 (en) 2015-06-04
EP2921489B1 (en) 2017-09-06
MX2015005884A (es) 2015-12-09
SG11201503716RA (en) 2015-06-29
JPWO2014077235A1 (ja) 2017-01-05
ES2641469T3 (es) 2017-11-10
KR20150082301A (ko) 2015-07-15
DK2921489T3 (en) 2017-10-16
RU2662157C2 (ru) 2018-07-24
KR102160841B1 (ko) 2020-09-28
ZA201503323B (en) 2016-08-31
RU2015122717A (ru) 2017-01-10
JP5963025B2 (ja) 2016-08-03
BR112015010823A2 (pt) 2017-07-11
CN104768944B (zh) 2017-03-29
IL238701A0 (en) 2015-06-30
CN104768944A (zh) 2015-07-08
PH12015501056B1 (en) 2015-07-27
EP2921489A4 (en) 2016-04-06

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