PE20110069A1 - Compuestos de tetraciclina sustituidos - Google Patents

Compuestos de tetraciclina sustituidos

Info

Publication number
PE20110069A1
PE20110069A1 PE2010000229A PE2010000229A PE20110069A1 PE 20110069 A1 PE20110069 A1 PE 20110069A1 PE 2010000229 A PE2010000229 A PE 2010000229A PE 2010000229 A PE2010000229 A PE 2010000229A PE 20110069 A1 PE20110069 A1 PE 20110069A1
Authority
PE
Peru
Prior art keywords
alkenyl
alkyl
tetracycline compounds
substituted tetracycline
dimethylamine
Prior art date
Application number
PE2010000229A
Other languages
English (en)
Spanish (es)
Inventor
Joel Berniac
Todd Bowser
Original Assignee
Paratek Pharm Innc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Paratek Pharm Innc filed Critical Paratek Pharm Innc
Publication of PE20110069A1 publication Critical patent/PE20110069A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/65—Tetracyclines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Hydrogenated Pyridines (AREA)
PE2010000229A 2008-04-14 2010-04-14 Compuestos de tetraciclina sustituidos PE20110069A1 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US4477308P 2008-04-14 2008-04-14
PCT/US2009/002344 WO2009128913A1 (en) 2008-04-14 2009-04-14 Substituted tetracycline compounds
US12/423,718 US20100022483A1 (en) 2008-04-14 2009-04-14 Substituted Tetracycline Compounds

Publications (1)

Publication Number Publication Date
PE20110069A1 true PE20110069A1 (es) 2011-01-31

Family

ID=41199392

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2010000229A PE20110069A1 (es) 2008-04-14 2010-04-14 Compuestos de tetraciclina sustituidos

Country Status (7)

Country Link
US (1) US20100022483A1 (https=)
EP (1) EP2276342A4 (https=)
JP (1) JP2011517697A (https=)
AU (1) AU2009236631A1 (https=)
CA (1) CA2721399A1 (https=)
PE (1) PE20110069A1 (https=)
WO (1) WO2009128913A1 (https=)

Families Citing this family (11)

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CN103040773A (zh) 2003-07-25 2013-04-17 沃纳奇尔科特有限责任公司 多西环素金属络合物固体剂型
AU2006206359B2 (en) * 2005-01-21 2011-03-31 Allergan Pharmaceuticals International Limited A tetracycline metal complex in a solid dosage form
CA2717703A1 (en) 2008-03-05 2009-09-11 Paratek Pharmaceuticals, Inc. Minocycline compounds and methods of use thereof
PT2323972E (pt) 2008-08-08 2013-10-09 Tetraphase Pharmaceuticals Inc Compostos de tetraciclina substituídos com c7-flúor
EP2427425B1 (en) 2009-05-08 2017-03-08 Tetraphase Pharmaceuticals, Inc. Tetracycline compounds
IN2012DN02502A (https=) 2009-08-28 2015-08-28 Tetraphase Pharmaceuticals Inc
CA2874640A1 (en) * 2012-05-30 2013-12-05 Paratek Pharmaceuticals, Inc. 7-disubstituted-phenyl tetracycline derivatives
BR112015004523B1 (pt) 2012-08-31 2020-08-04 Tetraphase Pharmaceuticals, Inc Compostos de tetraciclina, composições farmacêuticas e seus usos
CN110582486B (zh) 2016-10-19 2024-01-12 四相制药公司 艾若威四环素的结晶形式
BR112019008897A2 (pt) 2016-11-01 2019-08-13 Paratek Pharm Innc método para tratar pneumonia bacteriana adquirida na comunidade.
US20230113011A1 (en) * 2020-03-13 2023-04-13 Cmtx Biotech Inc. Methods of treating illnesses caused by coronavirus, swine flu and avian flu

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Also Published As

Publication number Publication date
WO2009128913A1 (en) 2009-10-22
EP2276342A4 (en) 2012-02-22
CA2721399A1 (en) 2009-10-22
EP2276342A1 (en) 2011-01-26
JP2011517697A (ja) 2011-06-16
AU2009236631A1 (en) 2009-10-22
US20100022483A1 (en) 2010-01-28

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