PA8777601A1 - Combinación de antagonista del receptor de progesterona con un agonista y un antagonista de la hormona liberadora de hormona luteinizante para usar en enfermedades mediadas por brca - Google Patents

Combinación de antagonista del receptor de progesterona con un agonista y un antagonista de la hormona liberadora de hormona luteinizante para usar en enfermedades mediadas por brca

Info

Publication number
PA8777601A1
PA8777601A1 PA20088777601A PA8777601A PA8777601A1 PA 8777601 A1 PA8777601 A1 PA 8777601A1 PA 20088777601 A PA20088777601 A PA 20088777601A PA 8777601 A PA8777601 A PA 8777601A PA 8777601 A1 PA8777601 A1 PA 8777601A1
Authority
PA
Panama
Prior art keywords
antagonist
agonist
diseases
combination
mediumed
Prior art date
Application number
PA20088777601A
Other languages
English (en)
Inventor
Hoffmann Jens
Korr Daniel
Original Assignee
Bayer Schering Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39872872&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PA8777601(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Schering Pharma Ag filed Critical Bayer Schering Pharma Ag
Publication of PA8777601A1 publication Critical patent/PA8777601A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/08Peptides having 5 to 11 amino acids
    • A61K38/09Luteinising hormone-releasing hormone [LHRH], i.e. Gonadotropin-releasing hormone [GnRH]; Related peptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/36Antigestagens
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/06Antianaemics

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Reproductive Health (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)

Abstract

COMBINACION DEL ANTAGONISTA DEL RECEPTOR DE PROGESTERONA 11ß-(4-ACETILFENIL)-17ß-HIDROXI-17ALFA-(1,1,2,2,2,-PENTAFLUOROETIL)-ESTRA-4,9-DIEN-3-ONA, O UN DERIVADO O UN ANALOGO DE ESTE ACEPTABLE PARA USO FARMACEUTICO, AL MENOS UN AGONISTA O UN ANTAGONISTA DE LA HORMONA LIBERADORA DE HORMONA LUTEINIZANTE, Y USO DE DICHA COMBINACION PARA LA PROFILAXIS Y EL TRATAMIENTO DE ENFERMEDADES MEDIADAS POR BRCAI O BRCA2. LOS AGONISTAS Y LOS ANTAGONISTAS DE LA HORMONA LIBERADORA DE HORMONA LUTEINIZANTE QUE PUEDEN COMBINARSE CON EL COMPUESTO 11ß-(4-ACETILFENIL)-17ß-HIDROXI-17ALFA -(1,1,2,2,2, PENTAFLUOROETIL) -ESTRA-4,9-DIEN-3-ONASON, POR EJEMPLO, GONADORELINA, GOSERELINA, TRIPTORELINA, BUSERELINA, NAFARELINA, DESLORELINA, HISTRELINA, ANTIDA, RAMORELIX, CETRORELIX, ANTARELIX, ORG30850, ABARELIX, GANIRELIX Y LEUPROLINA.
PA20088777601A 2007-04-23 2008-04-22 Combinación de antagonista del receptor de progesterona con un agonista y un antagonista de la hormona liberadora de hormona luteinizante para usar en enfermedades mediadas por brca PA8777601A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP07090084 2007-04-23
US91438307P 2007-04-27 2007-04-27

Publications (1)

Publication Number Publication Date
PA8777601A1 true PA8777601A1 (es) 2008-11-19

Family

ID=39872872

Family Applications (1)

Application Number Title Priority Date Filing Date
PA20088777601A PA8777601A1 (es) 2007-04-23 2008-04-22 Combinación de antagonista del receptor de progesterona con un agonista y un antagonista de la hormona liberadora de hormona luteinizante para usar en enfermedades mediadas por brca

Country Status (11)

Country Link
US (1) US20080261933A1 (es)
EP (1) EP2148682A1 (es)
JP (1) JP2010524996A (es)
AR (1) AR066233A1 (es)
CA (1) CA2683517A1 (es)
CL (1) CL2008001149A1 (es)
PA (1) PA8777601A1 (es)
PE (1) PE20090075A1 (es)
TW (1) TW200902029A (es)
UY (1) UY31042A1 (es)
WO (1) WO2008128786A1 (es)

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5372996A (en) * 1989-03-10 1994-12-13 Endorecherche, Inc. Method of treatment of androgen-related diseases
TW274552B (es) * 1992-05-26 1996-04-21 Hoechst Ag
JP3860841B2 (ja) * 1996-08-30 2006-12-20 ペプテック リミテッド 持続性ペプチド放出製剤
US8052982B2 (en) * 1998-07-20 2011-11-08 Peptech Animal Health Pty Limited Bioimplant formulation comprising lecithin and stearin
ES2389627T3 (es) * 1998-07-20 2012-10-29 Virbac (Australia) Pty Ltd Formulación para bioimplantes
DK1326617T3 (da) * 2000-10-18 2006-12-18 Schering Ag Anvendelse af 11beta- (acetylphenyl) -17beta-hydroxy-17alfa- (1,1,2,2-pentafluorethyl) estra-4,9-dien-3-on til fremstilling af et medikament til behandling af brystcancer, ovariecancer, endometrisk caner, myeloma og meningeom
UY26966A1 (es) * 2000-10-18 2002-06-20 Schering Ag Uso de antiprogestinas para la inducción de apoptosis en una célula
DE10051609A1 (de) * 2000-10-18 2002-05-02 Schering Ag Hemmung der Wachstumsfaktorabhängigkeit von Tumorzellen
CA2428249A1 (en) * 2000-11-16 2002-05-23 Pharmacia & Upjohn Company Combination therapy for estrogen-dependent disorders
US20030013694A1 (en) * 2001-05-25 2003-01-16 Jens Hoffmann Use and compositions of antiprogestins for treatment of prostate diseases
US20040043938A1 (en) * 2001-11-06 2004-03-04 Dinesh Purandare Combination therapy for estrogen-dependent disorders
GB0307777D0 (en) * 2003-04-04 2003-05-07 Medical Res Council Conjugate compounds

Also Published As

Publication number Publication date
TW200902029A (en) 2009-01-16
UY31042A1 (es) 2009-01-30
JP2010524996A (ja) 2010-07-22
AR066233A1 (es) 2009-08-05
CA2683517A1 (en) 2008-10-30
US20080261933A1 (en) 2008-10-23
EP2148682A1 (en) 2010-02-03
CL2008001149A1 (es) 2008-11-03
PE20090075A1 (es) 2009-04-24
WO2008128786A1 (en) 2008-10-30

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