NZ579372A - Substituted phenoxy thiazolidinediones as estrogen related receptor-alpha modulators - Google Patents

Info

Publication number

NZ579372A

NZ579372A NZ579372A NZ57937208A NZ579372A NZ 579372 A NZ579372 A NZ 579372A NZ 579372 A NZ579372 A NZ 579372A NZ 57937208 A NZ57937208 A NZ 57937208A NZ 579372 A NZ579372 A NZ 579372A

Authority

NZ

New Zealand

Prior art keywords

compound

disease

phenoxy

arthritis

methyl

Prior art date

2007-03-07

Links

• Espacenet
• Global Dossier
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• RPJOCUODRFHWDQ-UHFFFAOYSA-N 3-phenoxy-1,3-thiazolidine-2,4-dione Chemical class O=C1CSC(=O)N1OC1=CC=CC=C1 RPJOCUODRFHWDQ-UHFFFAOYSA-N 0.000 title abstract 2
• 102100036832 Steroid hormone receptor ERR1 Human genes 0.000 title description 58
• 108091008559 estrogen-related receptor alpha Proteins 0.000 title description 52
• 150000001875 compounds Chemical class 0.000 claims abstract description 152
• 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 claims abstract description 64
• WQZGKKKJIJFFOK-GASJEMHNSA-N Glucose Natural products OC[C@H]1OC(O)[C@H](O)[C@@H](O)[C@@H]1O WQZGKKKJIJFFOK-GASJEMHNSA-N 0.000 claims abstract description 63
• 239000008103 glucose Substances 0.000 claims abstract description 61
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• UNAANXDKBXWMLN-UHFFFAOYSA-N sibutramine Chemical compound C=1C=C(Cl)C=CC=1C1(C(N(C)C)CC(C)C)CCC1 UNAANXDKBXWMLN-UHFFFAOYSA-N 0.000 claims description 8
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