NZ572467A - Haloaryl substituted aminopurines, compositions thereof, and methods of treatment therewith - Google Patents

Info

Publication number

NZ572467A

NZ572467A NZ572467A NZ57246707A NZ572467A NZ 572467 A NZ572467 A NZ 572467A NZ 572467 A NZ572467 A NZ 572467A NZ 57246707 A NZ57246707 A NZ 57246707A NZ 572467 A NZ572467 A NZ 572467A

Authority

NZ

New Zealand

Prior art keywords

substituted

unsubstituted

compound

aryl

kinase

Prior art date

2006-04-26

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• 239000000203 mixture Chemical class 0.000 title claims description 88
• 125000003106 haloaryl group Chemical group 0.000 title abstract 2
• 238000011282 treatment Methods 0.000 title description 29
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• -1 aminopurine compound Chemical class 0.000 claims abstract description 286
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• 150000001875 compounds Chemical class 0.000 claims description 263
• 125000002924 primary amino group Chemical group [H]N([H])* 0.000 claims description 64
• 125000003118 aryl group Chemical group 0.000 claims description 42
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• 125000002887 hydroxy group Chemical group [H]O* 0.000 claims description 23
• 125000003545 alkoxy group Chemical group 0.000 claims description 21
• 125000004183 alkoxy alkyl group Chemical group 0.000 claims description 19
• 229910052736 halogen Inorganic materials 0.000 claims description 19
• 125000002768 hydroxyalkyl group Chemical group 0.000 claims description 19
• 238000003556 assay Methods 0.000 claims description 18
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