NZ206659A - Cephalosporin derivatives and pharmaceutical compositions - Google Patents

Cephalosporin derivatives and pharmaceutical compositions

Info

Publication number
NZ206659A
NZ206659A NZ206659A NZ20665983A NZ206659A NZ 206659 A NZ206659 A NZ 206659A NZ 206659 A NZ206659 A NZ 206659A NZ 20665983 A NZ20665983 A NZ 20665983A NZ 206659 A NZ206659 A NZ 206659A
Authority
NZ
New Zealand
Prior art keywords
group
denotes
isoquinoline
alkyl
general formula
Prior art date
Application number
NZ206659A
Other languages
English (en)
Inventor
R Lattrell
W Durckheimer
R Kirrstetter
W Schwab
N Klesel
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of NZ206659A publication Critical patent/NZ206659A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/38—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof
    • C07D501/46—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof with the 7-amino radical acylated by carboxylic acids containing hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/57—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with a further substituent in position 7, e.g. cephamycines
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Rigid Pipes And Flexible Pipes (AREA)
NZ206659A 1982-12-23 1983-12-21 Cephalosporin derivatives and pharmaceutical compositions NZ206659A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19823247614 DE3247614A1 (de) 1982-12-23 1982-12-23 Cephalosporinderivate und verfahren zu ihrer herstellung

Publications (1)

Publication Number Publication Date
NZ206659A true NZ206659A (en) 1986-11-12

Family

ID=6181485

Family Applications (1)

Application Number Title Priority Date Filing Date
NZ206659A NZ206659A (en) 1982-12-23 1983-12-21 Cephalosporin derivatives and pharmaceutical compositions

Country Status (19)

Country Link
EP (1) EP0111935B1 (enrdf_load_html_response)
JP (1) JPS59130294A (enrdf_load_html_response)
KR (1) KR840007015A (enrdf_load_html_response)
AT (1) ATE37881T1 (enrdf_load_html_response)
AU (1) AU2280983A (enrdf_load_html_response)
CS (1) CS249132B2 (enrdf_load_html_response)
DD (1) DD216026A5 (enrdf_load_html_response)
DE (2) DE3247614A1 (enrdf_load_html_response)
DK (1) DK594383A (enrdf_load_html_response)
ES (1) ES528247A0 (enrdf_load_html_response)
FI (1) FI834710A7 (enrdf_load_html_response)
GR (1) GR81360B (enrdf_load_html_response)
HU (1) HU189792B (enrdf_load_html_response)
IL (1) IL70519A0 (enrdf_load_html_response)
NO (1) NO834775L (enrdf_load_html_response)
NZ (1) NZ206659A (enrdf_load_html_response)
PH (1) PH20088A (enrdf_load_html_response)
PT (1) PT77877B (enrdf_load_html_response)
ZA (1) ZA839526B (enrdf_load_html_response)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK500285A (da) * 1984-11-02 1986-05-03 Glaxo Group Ltd Cephalosporinantibiotika
CA1267647A (en) * 1984-12-27 1990-04-10 Ryosuke Ushijima Cephalosporin derivatives
NO166283C (no) * 1985-03-01 1991-06-26 Takeda Chemical Industries Ltd Analogifremgangsmaate for fremstilling av terapeutisk aktive 7beta-(2-(5-amino-1,2,4-tiadiazol-3-yl)-2(z)-substituertoksyiminoacetamido)-3-(heterocyclylmetyl)-3-cefem-4-karboksylsyrederivater.
GB2183630A (en) * 1985-10-31 1987-06-10 Glaxo Group Ltd Cephalosporin antibiotics
EP0238060B1 (en) * 1986-03-19 1992-01-08 Banyu Pharmaceutical Co., Ltd. Cephalosporin derivatives, processes for their preparation and antibacterial agents
JPH0645631B2 (ja) * 1986-03-19 1994-06-15 萬有製薬株式会社 新規セフアロスポリン誘導体
US4814328A (en) * 1986-03-19 1989-03-21 Banyu Pharmaceutical Co., Ltd. Cephalosporin derivatives, and antibacterial agents
WO1988005776A1 (en) * 1987-02-02 1988-08-11 Teijin Limited Cephalosporin compounds or their salts, process for their preparation, and parmaceutical compositions
AU1228988A (en) * 1987-02-03 1988-08-24 Teijin Limited Cephalosporin compounds or their salts, process for their preparation, and pharmaceutical compositions
DE3910421A1 (de) * 1989-03-31 1990-10-04 Hoechst Ag Polare cephalosporinderivate und verfahren zu ihrer herstellung
TW200305422A (en) 2002-03-18 2003-11-01 Shionogi & Co Broad spectrum cefem compounds

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2715385A1 (de) * 1976-04-14 1977-11-10 Takeda Chemical Industries Ltd Cephalosporinderivate, verfahren zu ihrer herstellung und sie enthaltende arzneimittel
DE2714880A1 (de) * 1977-04-02 1978-10-26 Hoechst Ag Cephemderivate und verfahren zu ihrer herstellung
US4396619A (en) * 1981-09-08 1983-08-02 Eli Lilly And Company Cephalosporin betaines
US4396620A (en) * 1981-09-08 1983-08-02 Eli Lilly And Company Cephalosporin quinolinium betaines
US4450270A (en) * 1981-10-02 1984-05-22 Eli Lilly And Company Dioximino cephalosporin antibiotics
US4402955A (en) * 1981-10-02 1983-09-06 Eli Lilly And Company Dioximino cephalosporin antibiotics

Also Published As

Publication number Publication date
DE3378212D1 (en) 1988-11-17
ES8406494A1 (es) 1984-08-01
GR81360B (enrdf_load_html_response) 1984-12-11
NO834775L (no) 1984-06-25
EP0111935B1 (de) 1988-10-12
AU2280983A (en) 1984-06-28
DE3247614A1 (de) 1984-07-05
PT77877A (de) 1984-01-01
HU189792B (en) 1986-07-28
DK594383A (da) 1984-06-24
ATE37881T1 (de) 1988-10-15
PH20088A (en) 1986-09-24
FI834710A7 (fi) 1984-06-24
JPS59130294A (ja) 1984-07-26
CS249132B2 (en) 1987-03-12
HUT34036A (en) 1985-01-28
PT77877B (de) 1986-04-21
ES528247A0 (es) 1984-08-01
KR840007015A (ko) 1984-12-04
DD216026A5 (de) 1984-11-28
DK594383D0 (da) 1983-12-22
ZA839526B (en) 1984-08-29
IL70519A0 (en) 1984-03-30
EP0111935A2 (de) 1984-06-27
EP0111935A3 (en) 1985-07-03
FI834710A0 (fi) 1983-12-21

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