NO980129D0 - Heterocyklylkarboksamid-derivater og deres anvendelse som terapautiske midler - Google Patents

Heterocyklylkarboksamid-derivater og deres anvendelse som terapautiske midler

Info

Publication number
NO980129D0
NO980129D0 NO980129A NO980129A NO980129D0 NO 980129 D0 NO980129 D0 NO 980129D0 NO 980129 A NO980129 A NO 980129A NO 980129 A NO980129 A NO 980129A NO 980129 D0 NO980129 D0 NO 980129D0
Authority
NO
Norway
Prior art keywords
disorders
pct
date jan
methylene
sec
Prior art date
Application number
NO980129A
Other languages
English (en)
Norwegian (no)
Other versions
NO980129L (no
Inventor
Alan Martin Birch
David John Heal
Frank Kerrigan
Keith Frank Martin
Patricia Lesley Needham
Bruce Jeremy Sargent
Original Assignee
Knoll Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Knoll Ag filed Critical Knoll Ag
Publication of NO980129L publication Critical patent/NO980129L/no
Publication of NO980129D0 publication Critical patent/NO980129D0/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Endocrinology (AREA)
  • Psychiatry (AREA)
  • Cardiology (AREA)
  • Reproductive Health (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
NO980129A 1995-07-13 1998-01-12 Heterocyklylkarboksamid-derivater og deres anvendelse som terapautiske midler NO980129D0 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9514380.6A GB9514380D0 (en) 1995-07-13 1995-07-13 Therapeutic agents
PCT/EP1996/002890 WO1997003071A1 (en) 1995-07-13 1996-07-02 Heterocyclylcarboxamide derivatives and their use as therapeutic agents

Publications (2)

Publication Number Publication Date
NO980129L NO980129L (no) 1998-01-12
NO980129D0 true NO980129D0 (no) 1998-01-12

Family

ID=10777626

Family Applications (1)

Application Number Title Priority Date Filing Date
NO980129A NO980129D0 (no) 1995-07-13 1998-01-12 Heterocyklylkarboksamid-derivater og deres anvendelse som terapautiske midler

Country Status (26)

Country Link
US (1) US5935973A (pt)
EP (1) EP0839145B1 (pt)
JP (1) JPH11508599A (pt)
KR (1) KR19990028918A (pt)
CN (1) CN1071755C (pt)
AT (1) ATE253573T1 (pt)
AU (1) AU708890B2 (pt)
BG (1) BG62771B1 (pt)
BR (1) BR9609506A (pt)
CA (1) CA2223472A1 (pt)
CZ (1) CZ388497A3 (pt)
DE (1) DE69630604T2 (pt)
GB (1) GB9514380D0 (pt)
HR (1) HRP960348A2 (pt)
HU (1) HUP9901485A3 (pt)
IL (1) IL122540A (pt)
MX (1) MX9800084A (pt)
NO (1) NO980129D0 (pt)
NZ (1) NZ313164A (pt)
PL (1) PL324529A1 (pt)
RU (1) RU2169147C2 (pt)
SK (1) SK2498A3 (pt)
TR (1) TR199800041T1 (pt)
TW (1) TW454006B (pt)
WO (1) WO1997003071A1 (pt)
ZA (1) ZA965921B (pt)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9811879D0 (en) * 1998-06-03 1998-07-29 Knoll Ag Therapeutic agents
GB9915616D0 (en) * 1999-07-05 1999-09-01 Knoll Ag Therapeutic agents
UA73981C2 (en) * 2000-03-10 2005-10-17 Merck Patent Gmbh (r)-(-)-2-[5-(4-fluorophenyl)-3-pyridylmethylaminomethyl]-chromane for treatment of extrapyramidal movement disorders (variants), pharmaceutical composition and kit
AU4890301A (en) 2000-04-17 2001-10-30 Dong Wha Pharmaceutical Industrial Co., Ltd. 6-methylnicotinamide derivatives as antiviral agents
RU2283648C2 (ru) * 2000-11-14 2006-09-20 Мерк Патент Гмбх Новое применение комбинированных селективных антагонистов допаминового рецептора d2 и агонистов рецептора 5-нт 1a
GB0112836D0 (en) 2001-05-25 2001-07-18 Smithkline Beecham Plc Medicaments
US8106074B2 (en) 2001-07-13 2012-01-31 Pierre Fabre Medicament Pyridin-2-yl-methylamine derivatives for treating opiate dependence
SI1408964T1 (sl) 2001-07-26 2007-06-30 Merck Patent Gmbh Uporaba 2- 5-(4-fluorofenil)-3-piridilmetil-aminometil -kromana in njegovih fizioloĺ ko sprejemljivih soli
KR101204247B1 (ko) 2003-07-22 2012-11-22 아스텍스 테라퓨틱스 리미티드 3,4-이치환된 1h-피라졸 화합물 및 그의 시클린 의존성키나제 (cdk) 및 글리코겐 합성효소 키나제-3(gsk-3) 조정제로서 용도
EP1720874A4 (en) * 2004-02-24 2010-03-03 Bioaxone Therapeutique Inc SUBSTITUTED PIPERIDINE DERIVATIVES IN POSITION 4
JP4604583B2 (ja) * 2004-07-20 2011-01-05 ダイソー株式会社 1−アミド−3−(2−ヒドロキシフェノキシ)−2−プロパノール誘導体、ならびに2−アミドメチル−1,4−ベンゾジオキサン誘導体の製造法
US20080161251A1 (en) 2005-01-21 2008-07-03 Astex Therapeutics Limited Pharmaceutical Compounds
JP5475235B2 (ja) 2005-01-21 2014-04-16 アステックス・セラピューティクス・リミテッド 医薬化合物
TWI457122B (zh) 2007-07-20 2014-10-21 Orion Corp 作為用於治療周邊和中央神經系統疾病之alpha2C拮抗劑的2,3-二氫苯並[1,4]戴奧辛-2-基甲基衍生物
US8524766B2 (en) * 2008-04-29 2013-09-03 Nsab, Filial Af Neurosearch Sweden Ab, Sverige Modulators of dopamine neurotransmission
US9238666B2 (en) * 2012-06-11 2016-01-19 Bristol-Myers Squibb Company Phosphoramidic acid prodrugs of 5-[5-phenyl-4-(pyridin-2-ylmethylamino)quinazolin-2-yl] pyridine-3-sulfonamide

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8302622D0 (en) * 1983-01-31 1983-03-02 Celltech Ltd Immunoassay
EP0200960A1 (en) * 1985-05-08 1986-11-12 Abbott Laboratories Total estriol fluorescence polarization immunoassay
EP0594593A1 (en) * 1990-03-15 1994-05-04 PHARMACIA & UPJOHN COMPANY Therapeutically useful heterocyclic indole compounds
US5240943A (en) * 1991-12-19 1993-08-31 G. D. Searle & Co. Benzopyran class iii antiarrhythmic agents
GB9314758D0 (en) * 1993-07-16 1993-08-25 Wyeth John & Brother Ltd Heterocyclic derivatives
GB9318431D0 (en) * 1993-09-06 1993-10-20 Boots Co Plc Therapeutic agents
FR2724383B1 (fr) * 1994-09-13 1996-10-18 Synthelabo Derives de 2-aminopyrimidine-4-carboxamide, leur preparation et leur application en therapeutique

Also Published As

Publication number Publication date
GB9514380D0 (en) 1995-09-13
NZ313164A (en) 1999-07-29
RU2169147C2 (ru) 2001-06-20
HRP960348A2 (en) 1998-04-30
DE69630604T2 (de) 2004-09-23
NO980129L (no) 1998-01-12
BG102145A (en) 1998-11-30
IL122540A0 (en) 1998-06-15
BG62771B1 (bg) 2000-07-31
AU6517296A (en) 1997-02-10
SK2498A3 (en) 1998-09-09
US5935973A (en) 1999-08-10
TR199800041T1 (xx) 1998-05-21
ZA965921B (en) 1998-01-12
CN1071755C (zh) 2001-09-26
CZ388497A3 (cs) 1998-06-17
AU708890B2 (en) 1999-08-12
HUP9901485A3 (en) 2001-03-28
PL324529A1 (en) 1998-06-08
CN1190967A (zh) 1998-08-19
DE69630604D1 (de) 2003-12-11
JPH11508599A (ja) 1999-07-27
IL122540A (en) 2001-10-31
KR19990028918A (ko) 1999-04-15
MX9800084A (es) 1998-03-29
BR9609506A (pt) 1999-06-01
ATE253573T1 (de) 2003-11-15
CA2223472A1 (en) 1997-01-30
EP0839145B1 (en) 2003-11-05
TW454006B (en) 2001-09-11
WO1997003071A1 (en) 1997-01-30
HUP9901485A2 (en) 2000-07-28
EP0839145A1 (en) 1998-05-06

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