NO951811L - Kinolin- og benzimidazolderivater, deres fremstilling og anvendelse - Google Patents

Kinolin- og benzimidazolderivater, deres fremstilling og anvendelse

Info

Publication number
NO951811L
NO951811L NO951811A NO951811A NO951811L NO 951811 L NO951811 L NO 951811L NO 951811 A NO951811 A NO 951811A NO 951811 A NO951811 A NO 951811A NO 951811 L NO951811 L NO 951811L
Authority
NO
Norway
Prior art keywords
quinoline
preparation
benzimidazole derivatives
group
general formula
Prior art date
Application number
NO951811A
Other languages
English (en)
Norwegian (no)
Other versions
NO951811D0 (no
Inventor
George Pascal
Mireille Sevrin
Michel Peynot
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Publication of NO951811D0 publication Critical patent/NO951811D0/no
Publication of NO951811L publication Critical patent/NO951811L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/16Peri-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/16Peri-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
NO951811A 1994-05-10 1995-05-09 Kinolin- og benzimidazolderivater, deres fremstilling og anvendelse NO951811L (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9405715A FR2719843B1 (fr) 1994-05-10 1994-05-10 Dérivés de 5,6-dihydro-4h-imidazo [2',1':2,3] imidazo-[4,5,1-ij] quinoléine et de 4,5-dihydroimidazo [1,2-a] pyrrolo-[1,2,3-cd] benzimidazole, leur préparation et leur application en thérapeutique.

Publications (2)

Publication Number Publication Date
NO951811D0 NO951811D0 (no) 1995-05-09
NO951811L true NO951811L (no) 1995-11-13

Family

ID=9463058

Family Applications (1)

Application Number Title Priority Date Filing Date
NO951811A NO951811L (no) 1994-05-10 1995-05-09 Kinolin- og benzimidazolderivater, deres fremstilling og anvendelse

Country Status (18)

Country Link
US (1) US5512590A (de)
EP (1) EP0682025A1 (de)
JP (1) JPH0853450A (de)
KR (1) KR950032193A (de)
CN (1) CN1115761A (de)
AU (1) AU1793595A (de)
CA (1) CA2148951A1 (de)
CZ (1) CZ119495A3 (de)
FI (1) FI952249A (de)
FR (1) FR2719843B1 (de)
HU (1) HUT72666A (de)
IL (1) IL113672A (de)
NO (1) NO951811L (de)
NZ (1) NZ272089A (de)
PL (1) PL308517A1 (de)
RU (1) RU95107157A (de)
SK (1) SK59695A3 (de)
ZA (1) ZA953750B (de)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0120345D0 (en) * 2001-08-21 2001-10-17 Merck Sharp & Dohme Therapeutic agents
AU2003297153B2 (en) * 2002-12-18 2010-06-10 Mallinckrodt Inc. Synthesis of heteroaryl acetamides
CA2571491A1 (en) * 2004-06-22 2006-01-19 Mallinckrodt, Inc. Synthesis of heteroaryl acetamides from reaction mixtures having reduced water content
AU2006235318A1 (en) * 2005-04-07 2006-10-19 Hythiam, Inc. Improved methods of and compositions for the prevention of anxiety, substance abuse, and dependence
PE20070078A1 (es) 2005-06-14 2007-03-08 Schering Corp Compuestos heterociclicos macrociclicos como inhibidores de aspartil proteasa
AU2020357983A1 (en) * 2019-10-03 2022-04-21 Dana-Farber Cancer Institute, Inc. Tricyclic kinase inhibitors and uses thereof
AU2021267373A1 (en) 2020-05-06 2022-12-08 Ajax Therapeutics, Inc. 6-heteroaryloxy benzimidazoles and azabenzimidazoles as JAK2 inhibitors
WO2022140527A1 (en) 2020-12-23 2022-06-30 Ajax Therapeutics, Inc. 6-heteroaryloxy benzimidazoles and azabenzimidazoles as jak2 inhibitors
TW202334139A (zh) 2021-11-09 2023-09-01 美商雅捷可斯治療公司 作為jak2抑制劑之6-雜芳氧基苯并咪唑及氮雜苯并咪唑

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3732243A (en) * 1970-06-23 1973-05-08 Sankyo Co 2-(p-bromophenyl)-9-dimethyl-amino-propyl-9h-imidazo(1,2-a)benzimidazole
FR2568879B1 (fr) * 1984-08-07 1986-12-12 Synthelabo Imidazo(1,2-a)quinolines, leur preparation et leur application en therapeutique
FR2593817B1 (fr) * 1986-01-31 1988-04-15 Synthelabo Derives de tetrahydro-5,6,7,8 imidazo(1,2-a)pyridine, leur preparation et leur application en therapeutique
DK0480939T3 (da) * 1989-06-09 1995-07-10 Upjohn Co Heterocycliske aminer med virkning på centralnervesystemet
EP0607076A1 (de) * 1993-01-15 1994-07-20 Synthelabo 9H-Imidazo 1,2-a benzimidazolderivate mit GABA wirkung

Also Published As

Publication number Publication date
AU1793595A (en) 1995-11-16
KR950032193A (ko) 1995-12-20
NZ272089A (en) 1996-07-26
IL113672A0 (en) 1995-08-31
FI952249A0 (fi) 1995-05-09
CZ119495A3 (en) 1995-12-13
FR2719843A1 (fr) 1995-11-17
RU95107157A (ru) 1997-03-20
JPH0853450A (ja) 1996-02-27
CA2148951A1 (en) 1995-11-11
FI952249A (fi) 1995-11-11
NO951811D0 (no) 1995-05-09
ZA953750B (en) 1996-04-02
US5512590A (en) 1996-04-30
EP0682025A1 (de) 1995-11-15
IL113672A (en) 1997-11-20
FR2719843B1 (fr) 1996-06-07
SK59695A3 (en) 1995-12-06
CN1115761A (zh) 1996-01-31
HUT72666A (en) 1996-05-28
PL308517A1 (en) 1995-11-13

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