IL113672A - 9-phenyl-5,6-dihydro-4H-imidazo(2',1':2,3)imidazo-(4,5,1-ij)quinoline and 8-phenyl-4,5-dihydroimidazo-(1,2-a)pyrrolo(1,2,3-cd)benzimidazole derivatives their preparation and pharmaceutical compositions containing them - Google Patents

9-phenyl-5,6-dihydro-4H-imidazo(2',1':2,3)imidazo-(4,5,1-ij)quinoline and 8-phenyl-4,5-dihydroimidazo-(1,2-a)pyrrolo(1,2,3-cd)benzimidazole derivatives their preparation and pharmaceutical compositions containing them

Info

Publication number
IL113672A
IL113672A IL11367295A IL11367295A IL113672A IL 113672 A IL113672 A IL 113672A IL 11367295 A IL11367295 A IL 11367295A IL 11367295 A IL11367295 A IL 11367295A IL 113672 A IL113672 A IL 113672A
Authority
IL
Israel
Prior art keywords
imidazo
phenyl
dihydroimidazo
pyrrolo
quinoline
Prior art date
Application number
IL11367295A
Other languages
English (en)
Other versions
IL113672A0 (en
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Publication of IL113672A0 publication Critical patent/IL113672A0/xx
Publication of IL113672A publication Critical patent/IL113672A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/16—Peri-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/16—Peri-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL11367295A 1994-05-10 1995-05-09 9-phenyl-5,6-dihydro-4H-imidazo(2',1':2,3)imidazo-(4,5,1-ij)quinoline and 8-phenyl-4,5-dihydroimidazo-(1,2-a)pyrrolo(1,2,3-cd)benzimidazole derivatives their preparation and pharmaceutical compositions containing them IL113672A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9405715A FR2719843B1 (fr) 1994-05-10 1994-05-10 Dérivés de 5,6-dihydro-4h-imidazo [2',1':2,3] imidazo-[4,5,1-ij] quinoléine et de 4,5-dihydroimidazo [1,2-a] pyrrolo-[1,2,3-cd] benzimidazole, leur préparation et leur application en thérapeutique.

Publications (2)

Publication Number Publication Date
IL113672A0 IL113672A0 (en) 1995-08-31
IL113672A true IL113672A (en) 1997-11-20

Family

ID=9463058

Family Applications (1)

Application Number Title Priority Date Filing Date
IL11367295A IL113672A (en) 1994-05-10 1995-05-09 9-phenyl-5,6-dihydro-4H-imidazo(2',1':2,3)imidazo-(4,5,1-ij)quinoline and 8-phenyl-4,5-dihydroimidazo-(1,2-a)pyrrolo(1,2,3-cd)benzimidazole derivatives their preparation and pharmaceutical compositions containing them

Country Status (18)

Country Link
US (1) US5512590A (de)
EP (1) EP0682025A1 (de)
JP (1) JPH0853450A (de)
KR (1) KR950032193A (de)
CN (1) CN1115761A (de)
AU (1) AU1793595A (de)
CA (1) CA2148951A1 (de)
CZ (1) CZ119495A3 (de)
FI (1) FI952249A (de)
FR (1) FR2719843B1 (de)
HU (1) HUT72666A (de)
IL (1) IL113672A (de)
NO (1) NO951811L (de)
NZ (1) NZ272089A (de)
PL (1) PL308517A1 (de)
RU (1) RU95107157A (de)
SK (1) SK59695A3 (de)
ZA (1) ZA953750B (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0120345D0 (en) * 2001-08-21 2001-10-17 Merck Sharp & Dohme Therapeutic agents
CN100398539C (zh) * 2002-12-18 2008-07-02 马林克罗特公司 杂芳基乙酰胺的合成
AU2005262622A1 (en) * 2004-06-22 2006-01-19 Mallinckrodt Inc. Synthesis of heteroaryl acetamides from reaction mixtures having reduced water content
EP1868593A2 (de) * 2005-04-07 2007-12-26 Hythiam, Inc. Verbesserte verfahren und zusammensetzungen zur prävention von angstzuständen, substanzenmissbrauch und abhängigkeit
EP1902057B1 (de) 2005-06-14 2013-10-23 Merck Sharp & Dohme Corp. Makrocyclische heterocyclische aspartylproteaseinhibitoren
US20240101559A1 (en) * 2019-10-03 2024-03-28 Dana-Farber Cancer Institute, Inc. Tricyclic kinase inhibitors and uses thereof
US11691963B2 (en) 2020-05-06 2023-07-04 Ajax Therapeutics, Inc. 6-heteroaryloxy benzimidazoles and azabenzimidazoles as JAK2 inhibitors
TW202334139A (zh) 2021-11-09 2023-09-01 美商雅捷可斯治療公司 作為ｊａｋ２抑制劑之６－雜芳氧基苯并咪唑及氮雜苯并咪唑

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3732243A (en) * 1970-06-23 1973-05-08 Sankyo Co 2-(p-bromophenyl)-9-dimethyl-amino-propyl-9h-imidazo(1,2-a)benzimidazole
FR2568879B1 (fr) * 1984-08-07 1986-12-12 Synthelabo Imidazo(1,2-a)quinolines, leur preparation et leur application en therapeutique
FR2593817B1 (fr) * 1986-01-31 1988-04-15 Synthelabo Derives de tetrahydro-5,6,7,8 imidazo(1,2-a)pyridine, leur preparation et leur application en therapeutique
DK0480939T3 (da) * 1989-06-09 1995-07-10 Upjohn Co Heterocycliske aminer med virkning på centralnervesystemet
EP0607076A1 (de) * 1993-01-15 1994-07-20 Synthelabo 9H-Imidazo 1,2-a benzimidazolderivate mit GABA wirkung

Also Published As

Publication number Publication date
EP0682025A1 (de) 1995-11-15
FI952249A0 (fi) 1995-05-09
IL113672A0 (en) 1995-08-31
US5512590A (en) 1996-04-30
NO951811D0 (no) 1995-05-09
FR2719843A1 (fr) 1995-11-17
CZ119495A3 (en) 1995-12-13
JPH0853450A (ja) 1996-02-27
KR950032193A (ko) 1995-12-20
FI952249A (fi) 1995-11-11
PL308517A1 (en) 1995-11-13
CN1115761A (zh) 1996-01-31
CA2148951A1 (en) 1995-11-11
ZA953750B (en) 1996-04-02
NZ272089A (en) 1996-07-26
AU1793595A (en) 1995-11-16
FR2719843B1 (fr) 1996-06-07
RU95107157A (ru) 1997-03-20
NO951811L (no) 1995-11-13
SK59695A3 (en) 1995-12-06
HUT72666A (en) 1996-05-28

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