NO942919L - Fenylalaninanaloger av bombesin - Google Patents

Fenylalaninanaloger av bombesin

Info

Publication number
NO942919L
NO942919L NO942919A NO942919A NO942919L NO 942919 L NO942919 L NO 942919L NO 942919 A NO942919 A NO 942919A NO 942919 A NO942919 A NO 942919A NO 942919 L NO942919 L NO 942919L
Authority
NO
Norway
Prior art keywords
bombesin
derivatives
phenylalanine analogues
tests
antagonizing
Prior art date
Application number
NO942919A
Other languages
English (en)
Norwegian (no)
Other versions
NO942919D0 (es
Inventor
Judson Vincent Edwards
Bradford Otto Fanger
Original Assignee
Merrell Dow Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merrell Dow Pharma filed Critical Merrell Dow Pharma
Publication of NO942919L publication Critical patent/NO942919L/no
Publication of NO942919D0 publication Critical patent/NO942919D0/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/08—Linear peptides containing only normal peptide links having 12 to 20 amino acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/57572—Gastrin releasing peptide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/02—Peptides of undefined number of amino acids; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/08—Linear peptides containing only normal peptide links having 12 to 20 amino acids
    • C07K7/086—Bombesin; Related peptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
NO942919A 1992-02-07 1994-08-05 Fenylalaninanaloger av bombesin NO942919L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US83383492A 1992-02-07 1992-02-07
PCT/US1993/000183 WO1993016105A1 (en) 1992-02-07 1993-01-07 Phenylalanine analogs of bombesin

Publications (2)

Publication Number Publication Date
NO942919L true NO942919L (no) 1994-08-05
NO942919D0 NO942919D0 (es) 1994-08-05

Family

ID=25265391

Family Applications (1)

Application Number Title Priority Date Filing Date
NO942919A NO942919L (no) 1992-02-07 1994-08-05 Fenylalaninanaloger av bombesin

Country Status (14)

Country Link
US (1) US5428018A (es)
EP (1) EP0626973A1 (es)
JP (1) JPH07505865A (es)
KR (1) KR950700325A (es)
AU (1) AU668909B2 (es)
CA (1) CA2129032A1 (es)
FI (1) FI943638A0 (es)
HU (1) HUT71585A (es)
IL (1) IL104621A0 (es)
MX (1) MX9300602A (es)
NO (1) NO942919L (es)
NZ (1) NZ246815A (es)
WO (1) WO1993016105A1 (es)
ZA (1) ZA93716B (es)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5723578A (en) * 1987-09-24 1998-03-03 The Administrators Of Tulane Educational Fund Peptide analogs of bombesin
US5877277A (en) 1987-09-24 1999-03-02 Biomeasure, Inc. Octapeptide bombesin analogs
US7078413B2 (en) 1996-04-19 2006-07-18 Wisconsin Alumni Research Foundation Compositions and methods of use for a bombesin peptide
UA65549C2 (uk) 1996-11-05 2004-04-15 Елі Ліллі Енд Компані Спосіб регулювання ожиріння шляхом периферійного введення аналогів та похідних glp-1 (варіанти) та фармацевтична композиція
EP0977579B1 (en) * 1997-04-22 2009-03-11 Curator Of The University Of Missouri Gastrin receptor-avid peptide conjugates
US8420050B2 (en) * 2003-01-13 2013-04-16 Bracco Imaging S.P.A. Gastrin releasing peptide compounds
US7226577B2 (en) 2003-01-13 2007-06-05 Bracco Imaging, S. P. A. Gastrin releasing peptide compounds
US7850947B2 (en) 2003-01-13 2010-12-14 Bracco Imaging S.P.A. Gastrin releasing peptide compounds
WO2004062574A2 (en) * 2003-01-13 2004-07-29 Bracco Imaging S.P.A. Improved linkers for radiopharmaceutical compounds
US7922998B2 (en) * 2003-01-13 2011-04-12 Bracco Imaging S.P.A. Gastrin releasing peptide compounds
US20060239923A1 (en) * 2003-01-13 2006-10-26 Bracco Imaging S.P.A. Gastrin releasing peptide compounds
US7611692B2 (en) 2003-01-13 2009-11-03 Bracco Imaging S.P.A. Gastrin releasing peptide compounds
WO2014052471A1 (en) 2012-09-25 2014-04-03 Biosynthema Inc. Grpr-antagonists for detection, diagnosis and treatment of grpr-positive cancer

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1592552A (en) * 1976-12-10 1981-07-08 Inst Nat Sante Rech Med Pseudopeptides used as medicaments
US4631270A (en) * 1978-11-20 1986-12-23 Research Corporation Therapeutically useful pseudopeptides, compositions containing the same and methods of preparation and use
EP0076557B1 (en) * 1981-06-22 1985-11-13 Imperial Chemical Industries Plc Peptides and pseudopeptides in which the n terminus bears two substituents
US4871717A (en) * 1987-01-07 1989-10-03 Administrators Of The Tulane Educational Fund Peptides
JP2795449B2 (ja) * 1987-09-24 1998-09-10 ジ・アドミニストレーターズ・オブ・ザ・ツーレイン・エデュケイショナル・ファンド 治療用ペプチド
US5047502A (en) * 1987-10-23 1991-09-10 Merck And Co., Inc. Gastrin releasing peptide antagonist
EP0313158A3 (en) * 1987-10-23 1990-08-22 Merck & Co. Inc. Gastrin releasing peptide antagonist
AU618029B2 (en) * 1987-11-02 1991-12-12 Imperial Chemical Industries Plc Polypeptide compounds
GB8806644D0 (en) * 1988-03-21 1988-04-20 Imp Cancer Res Tech Neuropeptide antagonists
GB8808768D0 (en) * 1988-04-14 1988-05-18 Erba Carlo Spa Peptide ligands for bombesin receptors
GB8813356D0 (en) * 1988-06-06 1988-07-13 Ici Plc Polypeptide compounds
GR1000608B (el) * 1988-07-21 1992-08-31 Erba Carlo Spa Μεθοδος για την παρασκευη ανταγωνιστων bombesin.
JP2919889B2 (ja) * 1988-10-14 1999-07-19 アドミニストレイターズ オブ ザ テューレイン エデュケイショナル ファンド 治療用ペプチド
US5028692A (en) * 1989-04-25 1991-07-02 Merck & Co., Inc. Gastrin releasing peptide antagonist
KR920701242A (ko) * 1989-11-06 1992-08-11 원본미기재 환원된 비가역성 봄베신 길항제
CA2030212A1 (en) * 1989-11-22 1991-05-23 Judson V. Edwards Peptides
WO1991017181A1 (en) * 1990-05-09 1991-11-14 The Administrators Of The Tulane Educational Fund Cyclized and linear therapeutic peptides
ZA915740B (en) * 1990-07-26 1992-05-27 Merrell Dow Pharma Peptides
US5244883A (en) * 1990-11-29 1993-09-14 The Administrators Of The Tulane Educational Fund Nonapeptide bombesin antagonists

Also Published As

Publication number Publication date
NO942919D0 (es) 1994-08-05
ZA93716B (en) 1993-09-01
EP0626973A1 (en) 1994-12-07
HU9402285D0 (en) 1994-10-28
FI943638A (fi) 1994-08-05
KR950700325A (ko) 1995-01-16
IL104621A0 (en) 1993-06-10
FI943638A0 (fi) 1994-08-05
CA2129032A1 (en) 1993-08-19
AU668909B2 (en) 1996-05-23
MX9300602A (es) 1993-08-01
US5428018A (en) 1995-06-27
AU3439993A (en) 1993-09-03
HUT71585A (en) 1995-12-28
NZ246815A (en) 1996-02-27
JPH07505865A (ja) 1995-06-29
WO1993016105A1 (en) 1993-08-19

Similar Documents

Publication Publication Date Title
NO942919L (no) Fenylalaninanaloger av bombesin
Marasco et al. Substance P binds to the formylpeptide chemotaxis receptor on the rabbit neutrophil
Konishi et al. The effects of substance P and other peptides on spinal neurons of the frog
Solomon et al. Bioactivity of cholecystokinin analogues: CCK-8 is not more potent than CCK-33
Tashjian Jr et al. Role of calcium in the thyrotropin-releasing hormone-stimulated release of prolactin from pituitary cells in culture
Civitelli et al. Parathyroid hormone-related peptide transiently increases cytosolic calcium in osteoblast-like cells: comparison with parathyroid hormone
ATE156492T1 (de) Bombesinanaloge
JP2007302682A (ja) 副甲状腺ホルモンの類似体
US5717062A (en) Cyclic analogs of PTH and PTHrP
NO20051804L (no) GHRH analoger
RU2203286C2 (ru) Аналоги паратиреоидного гормона для лечения остеопороза
WO2001054771A3 (en) Method for using potassium channel agonists for delivering a medicant to an abnormal brain region and/or a malignant tumor
Mizrahi et al. Substance P antagonists active in vitro and in vivo
Ishibashi et al. Inhibition of growth of human small cell lung cancer by bromocriptine
Vigna et al. Effects of cholecystokinin, gastrin, and related peptides on coho salmon gallbladder contraction in vitro.
Potter et al. [Pro34] neuropeptide Y selectively identifies postjunctional-mediated actions of neuropeptide Y in vivo in rats and dogs
Toouli et al. Actions of cholecystokinin-pancreozymin, secretin and gastrin on extra-hepatic biliary tract motility in vitro.
Musso et al. Renal vasodilation and microvessel adenylate cyclase stimulation by synthetic parathyroid hormone-like protein fragments
Löffler et al. Parathyrin and calcitonin stimulate cyclic AMP accumulation in cultured murine brain cells.
NO941151L (no) Lineære adhesjonsinhibitorer
Huang et al. Parathyroid hormone stimulates adenylate cyclase in rat cerebral microvessels
Liang et al. Substance P stimulation of amylase release by isolated parotid cells and inhibition of substance P induction of salivation by vasoactive peptides
Vigna Evolution of endocrine regulation of gastrointestinal function in lower vertebrates
McGillis et al. Thymosin fraction 5 (TF5) stimulates secretion of adrenocorticotropic hormone (ACTH) from cultured rat pituitaries
Regoli et al. Neurokinin A. A pharmacological study

Legal Events

Date Code Title Description
FC2A Withdrawal, rejection or dismissal of laid open patent application