NO861486L - PROCEDURE FOR THE PREPARATION OF FLUORED BENZYLTRIAZOL COMPOUNDS. - Google Patents

PROCEDURE FOR THE PREPARATION OF FLUORED BENZYLTRIAZOL COMPOUNDS.

Info

Publication number
NO861486L
NO861486L NO861486A NO861486A NO861486L NO 861486 L NO861486 L NO 861486L NO 861486 A NO861486 A NO 861486A NO 861486 A NO861486 A NO 861486A NO 861486 L NO861486 L NO 861486L
Authority
NO
Norway
Prior art keywords
fluored
benzyltriazol
compounds
procedure
preparation
Prior art date
Application number
NO861486A
Other languages
Norwegian (no)
Other versions
NO164295B (en
NO164295C (en
Inventor
Rene Meier
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of NO861486L publication Critical patent/NO861486L/en
Publication of NO164295B publication Critical patent/NO164295B/en
Publication of NO164295C publication Critical patent/NO164295C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C247/00Compounds containing azido groups
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C33/00Unsaturated compounds having hydroxy or O-metal groups bound to acyclic carbon atoms
    • C07C33/40Halogenated unsaturated alcohols
    • C07C33/46Halogenated unsaturated alcohols containing only six-membered aromatic rings as cyclic parts
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/041,2,3-Triazoles; Hydrogenated 1,2,3-triazoles
NO861486A 1985-04-18 1986-04-16 ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE FLUORED BENZYLTRIAZOL COMPOUNDS. NO164295C (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH166385 1985-04-18

Publications (3)

Publication Number Publication Date
NO861486L true NO861486L (en) 1986-10-20
NO164295B NO164295B (en) 1990-06-11
NO164295C NO164295C (en) 1990-09-19

Family

ID=4215715

Family Applications (1)

Application Number Title Priority Date Filing Date
NO861486A NO164295C (en) 1985-04-18 1986-04-16 ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE FLUORED BENZYLTRIAZOL COMPOUNDS.

Country Status (22)

Country Link
EP (1) EP0199262B1 (en)
JP (1) JPS61243068A (en)
KR (1) KR900008810B1 (en)
AU (1) AU599024B2 (en)
CA (1) CA1272201A (en)
CY (1) CY1751A (en)
DD (1) DD245874A5 (en)
DE (1) DE3677626D1 (en)
DK (1) DK169720B1 (en)
ES (2) ES8800176A1 (en)
FI (1) FI93544C (en)
GR (1) GR861004B (en)
HK (1) HK1494A (en)
HU (1) HU203327B (en)
IE (1) IE58472B1 (en)
IL (1) IL78510A (en)
MX (1) MX9203628A (en)
NO (1) NO164295C (en)
NZ (1) NZ215871A (en)
PH (1) PH22568A (en)
PT (1) PT82400B (en)
ZA (1) ZA862873B (en)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0151528B1 (en) * 1984-02-02 1990-07-04 Merck & Co. Inc. 5-(amino or substituted amino)-1,2,3-triazoles
AU2633897A (en) * 1996-04-19 1997-11-12 Novo Nordisk A/S Solid phase and combinatorial synthesis of substituted 1,2,3-triazoles and of arrays of substituted 1,2,3-triazoles
CN1083436C (en) * 1996-07-11 2002-04-24 诺瓦提斯公司 Process for preparing 1-substituted 4-cyano-1,2,3-triazoles
TW403740B (en) * 1997-06-10 2000-09-01 Novartis Ag Novel crystal modifications of the compound 1-(2,6-difluorobenzyl)-1H-1,2,3-triazole-4-carboxamide
TW513301B (en) * 1999-03-01 2002-12-11 Novartis Ag Pharmaceutical composition for treatment of neuropathic pain and affective and attention disorders
WO2004106329A2 (en) * 2003-06-03 2004-12-09 Dr. Reddy's Laboratories Ltd. Novel antiinfective compounds and their pharmaceutical compositions
IT1393368B1 (en) * 2009-03-23 2012-04-20 Dipharma Francis Srl METHOD FOR THE PREPARATION OF RUFINAMIDE
IT1395736B1 (en) 2009-08-04 2012-10-19 Dipharma Francis Srl CRYSTALLINE FORMS OF RUFINAMIDE
WO2011135105A1 (en) * 2010-04-30 2011-11-03 Laboratorios Lesvi, S.L. Improved process for preparing rufinamide intermediate
ITMI20110718A1 (en) 2011-04-29 2012-10-30 Dipharma Francis Srl PROCEDURE FOR PURIFICATION OF RUFINAMIDE
US20150368211A1 (en) * 2013-01-31 2015-12-24 The Johns Hopkins University Rufinamide and derivatives and their use in modulating the gating process of human voltage-gated sodium channels
US9771335B2 (en) * 2015-07-31 2017-09-26 The Johns Hopkins University Derivatives of rufinamide and their use in inhibtion of the activation of human voltage-gated sodium channels
CA3008048C (en) 2015-12-11 2023-11-14 Aarhus Universitet Rufinamide for use in the treatment of myotonia
WO2021099481A1 (en) 2019-11-20 2021-05-27 Medichem, S.A. Solid composition containing rufinamide

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1511195A (en) * 1976-10-18 1978-05-17 Ici America Inc Triazole derivatives
FI834666A (en) * 1982-12-23 1984-06-24 Ciba Geigy Ag FOERFARANDE FOER FRAMSTAELLNING AV NYA ARALKYLTRIAZOLFOERENINGAR.

Also Published As

Publication number Publication date
HK1494A (en) 1994-01-14
EP0199262B1 (en) 1991-02-27
DD245874A5 (en) 1987-05-20
ES8800176A1 (en) 1987-10-16
PT82400B (en) 1988-08-17
DK169720B1 (en) 1995-01-23
PH22568A (en) 1988-10-17
AU599024B2 (en) 1990-07-12
GR861004B (en) 1986-08-12
CY1751A (en) 1994-06-03
NO164295B (en) 1990-06-11
FI93544C (en) 1995-04-25
CA1272201A (en) 1990-07-31
EP0199262A2 (en) 1986-10-29
PT82400A (en) 1986-05-01
IL78510A0 (en) 1986-08-31
DK175686A (en) 1986-10-19
MX9203628A (en) 1992-09-01
JPH0564949B2 (en) 1993-09-16
FI861573A (en) 1986-10-19
KR900008810B1 (en) 1990-11-30
ZA862873B (en) 1986-12-30
HUT40792A (en) 1987-02-27
AU5631986A (en) 1986-10-23
KR860008152A (en) 1986-11-12
FI861573A0 (en) 1986-04-14
NZ215871A (en) 1989-01-27
ES8802501A1 (en) 1988-07-01
JPS61243068A (en) 1986-10-29
DK175686D0 (en) 1986-04-17
IE861015L (en) 1986-10-18
IL78510A (en) 1992-05-25
HU203327B (en) 1991-07-29
NO164295C (en) 1990-09-19
ES557641A0 (en) 1988-07-01
ES554024A0 (en) 1987-10-16
FI93544B (en) 1995-01-13
DE3677626D1 (en) 1991-04-04
EP0199262A3 (en) 1987-08-26
IE58472B1 (en) 1993-09-22

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