NO333193B1 - Polyamidnukleinsyrederivater, anvendelse derav, midler inneholdende PNAderivatet og fremgangsmater for deres fremstilling. - Google Patents
Polyamidnukleinsyrederivater, anvendelse derav, midler inneholdende PNAderivatet og fremgangsmater for deres fremstilling. Download PDFInfo
- Publication number
- NO333193B1 NO333193B1 NO20024959A NO20024959A NO333193B1 NO 333193 B1 NO333193 B1 NO 333193B1 NO 20024959 A NO20024959 A NO 20024959A NO 20024959 A NO20024959 A NO 20024959A NO 333193 B1 NO333193 B1 NO 333193B1
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- Prior art keywords
- pna
- equal
- pna derivative
- derivative according
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- UEZVMMHDMIWARA-UHFFFAOYSA-M phosphonate Chemical compound [O-]P(=O)=O UEZVMMHDMIWARA-UHFFFAOYSA-M 0.000 description 1
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- 230000004962 physiological condition Effects 0.000 description 1
- 239000006187 pill Substances 0.000 description 1
- IUGYQRQAERSCNH-UHFFFAOYSA-N pivalic acid Chemical compound CC(C)(C)C(O)=O IUGYQRQAERSCNH-UHFFFAOYSA-N 0.000 description 1
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- 210000002966 serum Anatomy 0.000 description 1
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- 239000011734 sodium Substances 0.000 description 1
- 229910052708 sodium Inorganic materials 0.000 description 1
- AJPJDKMHJJGVTQ-UHFFFAOYSA-M sodium dihydrogen phosphate Chemical compound [Na+].OP(O)([O-])=O AJPJDKMHJJGVTQ-UHFFFAOYSA-M 0.000 description 1
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- 125000005931 tert-butyloxycarbonyl group Chemical group [H]C([H])([H])C(OC(*)=O)(C([H])([H])[H])C([H])([H])[H] 0.000 description 1
- WHRNULOCNSKMGB-UHFFFAOYSA-N tetrahydrofuran thf Chemical compound C1CCOC1.C1CCOC1 WHRNULOCNSKMGB-UHFFFAOYSA-N 0.000 description 1
- ZRKFYGHZFMAOKI-QMGMOQQFSA-N tgfbeta Chemical compound C([C@H](NC(=O)[C@H](C(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](N)CCSC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CC=1C=CC=CC=1)C(=O)N[C@@H](C)C(=O)N1[C@@H](CCC1)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CC=1C=CC=CC=1)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N1[C@@H](CCC1)C(=O)N1[C@@H](CCC1)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(O)=O)C1=CC=C(O)C=C1 ZRKFYGHZFMAOKI-QMGMOQQFSA-N 0.000 description 1
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H21/00—Compounds containing two or more mononucleotide units having separate phosphate or polyphosphate groups linked by saccharide radicals of nucleoside groups, e.g. nucleic acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/001—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof by chemical synthesis
- C07K14/003—Peptide-nucleic acids (PNAs)
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
- Y10T—TECHNICAL SUBJECTS COVERED BY FORMER US CLASSIFICATION
- Y10T436/00—Chemistry: analytical and immunological testing
- Y10T436/14—Heterocyclic carbon compound [i.e., O, S, N, Se, Te, as only ring hetero atom]
- Y10T436/142222—Hetero-O [e.g., ascorbic acid, etc.]
- Y10T436/143333—Saccharide [e.g., DNA, etc.]
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Virology (AREA)
- Engineering & Computer Science (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Pulmonology (AREA)
- Genetics & Genomics (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Dermatology (AREA)
- Gastroenterology & Hepatology (AREA)
- Biophysics (AREA)
- Tropical Medicine & Parasitology (AREA)
- AIDS & HIV (AREA)
- Biotechnology (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Polyamides (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Investigating Or Analysing Biological Materials (AREA)
- Investigating Or Analysing Materials By The Use Of Chemical Reactions (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10019135A DE10019135A1 (de) | 2000-04-18 | 2000-04-18 | Polyamidnukleinsäure-Derivate, Mittel und Verfahren zu ihrer Herstellung |
PCT/EP2001/004030 WO2001079216A2 (fr) | 2000-04-18 | 2001-04-07 | Derives d"acide nucleique polyamide, agents et procedes permettant de les preparer |
Publications (3)
Publication Number | Publication Date |
---|---|
NO20024959L NO20024959L (no) | 2002-10-15 |
NO20024959D0 NO20024959D0 (no) | 2002-10-15 |
NO333193B1 true NO333193B1 (no) | 2013-04-02 |
Family
ID=7639143
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20024959A NO333193B1 (no) | 2000-04-18 | 2002-10-15 | Polyamidnukleinsyrederivater, anvendelse derav, midler inneholdende PNAderivatet og fremgangsmater for deres fremstilling. |
Country Status (21)
Country | Link |
---|---|
US (5) | US6905820B2 (fr) |
EP (1) | EP1276760B1 (fr) |
JP (1) | JP4908714B2 (fr) |
KR (1) | KR100842723B1 (fr) |
AR (1) | AR032153A1 (fr) |
AT (1) | ATE344276T1 (fr) |
AU (1) | AU5479501A (fr) |
BR (1) | BR0110110A (fr) |
CA (1) | CA2406169C (fr) |
CY (1) | CY1105958T1 (fr) |
DE (2) | DE10019135A1 (fr) |
DK (1) | DK1276760T3 (fr) |
ES (1) | ES2275677T3 (fr) |
IL (2) | IL152288A0 (fr) |
MX (1) | MXPA02009953A (fr) |
NO (1) | NO333193B1 (fr) |
NZ (1) | NZ521988A (fr) |
PT (1) | PT1276760E (fr) |
TW (1) | TWI298328B (fr) |
WO (1) | WO2001079216A2 (fr) |
ZA (1) | ZA200208344B (fr) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20030165888A1 (en) * | 2001-07-18 | 2003-09-04 | Brown Bob D. | Oligonucleotide probes and primers comprising universal bases for diagnostic purposes |
US6518017B1 (en) * | 1997-10-02 | 2003-02-11 | Oasis Biosciences Incorporated | Combinatorial antisense library |
WO2000061807A1 (fr) * | 1999-04-08 | 2000-10-19 | Oasis Biosciences, Inc. | Paires d'amorces d'amplification et de sequençage et leur emploi |
DE10019135A1 (de) * | 2000-04-18 | 2001-10-31 | Aventis Pharma Gmbh | Polyamidnukleinsäure-Derivate, Mittel und Verfahren zu ihrer Herstellung |
TWI286849B (en) * | 2003-03-25 | 2007-09-11 | Nichia Corp | Positive electrode active material for nonaqueous electrolyte secondary battery and nonaqueous electrolyte secondary battery |
US20100143937A1 (en) * | 2007-05-31 | 2010-06-10 | Sanofi-Aventis | ASSAY METHODS FOR IDENTIFYING AGENTS THAT MODIFY THE ACTIVITY OF NAPE-PLD OR Abh4 |
WO2009044403A2 (fr) * | 2007-10-05 | 2009-04-09 | Juvenis Ltd. | Compositions polymères biodégradables injectables pour la réparation et l'augmentation des tissus mous |
US20090276855A1 (en) * | 2008-04-30 | 2009-11-05 | Nokia Corporation | Method, apparatus, and computer program product that provide for presentation of event items |
US20090276700A1 (en) * | 2008-04-30 | 2009-11-05 | Nokia Corporation | Method, apparatus, and computer program product for determining user status indicators |
US20090276436A1 (en) * | 2008-04-30 | 2009-11-05 | Nokia Corporation | Method, apparatus, and computer program product for providing service invitations |
US20090276412A1 (en) * | 2008-04-30 | 2009-11-05 | Nokia Corporation | Method, apparatus, and computer program product for providing usage analysis |
US20090292762A1 (en) * | 2008-05-20 | 2009-11-26 | Nokia Corporation | Method, Apparatus, and Computer Program Product for Publishing Content |
US20090327434A1 (en) * | 2008-06-30 | 2009-12-31 | Nokia Corporation | Method, Apparatus, and Computer Program Product for Anonymous Polling |
JP5990987B2 (ja) * | 2012-04-11 | 2016-09-14 | 株式会社Ihi | 微生物固定方法、および微生物検出方法 |
JP2015172904A (ja) * | 2014-03-12 | 2015-10-01 | 株式会社東芝 | Ldo型電圧レギュレータ、及び、受電装置 |
EP3250197A1 (fr) * | 2015-01-27 | 2017-12-06 | Indicator Systems International, Inc. | Conjugués polymères de fluorescéine |
KR102659194B1 (ko) * | 2016-07-26 | 2024-04-19 | 삼성전자주식회사 | 홀로그래픽 디스플레이 장치용 박형 백라이트 유닛 및 이를 포함하는 홀로그래픽 디스플레이 장치 |
Family Cites Families (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1995024221A1 (fr) * | 1986-08-18 | 1995-09-14 | The Dow Chemical Company | Conjugues dendrimeres bioactifs et/ou cibles |
EP0383803B1 (fr) * | 1987-10-28 | 2000-05-03 | Howard Florey Institute Of Experimental Physiology And Medicine | Conjugues d'oligonucleotide-polyamide |
DK51092D0 (da) | 1991-05-24 | 1992-04-15 | Ole Buchardt | Oligonucleotid-analoge betegnet pna, monomere synthoner og fremgangsmaade til fremstilling deraf samt anvendelser deraf |
DE4408531A1 (de) * | 1994-03-14 | 1995-09-28 | Hoechst Ag | PNA-Synthese unter Verwendung einer gegen schwache Säuren labilen Amino-Schutzgruppe |
DE4408528A1 (de) * | 1994-03-14 | 1995-09-28 | Hoechst Ag | Peptid-Oligonucleotid-Derivate, deren Herstellung und Verwendung |
PT804456E (pt) * | 1994-10-06 | 2003-01-31 | Peter Eigil Nielsen | Conjugados de acidos nucleicos dos peptidos |
DE19508923A1 (de) * | 1995-03-13 | 1996-09-19 | Hoechst Ag | Phosphonomonoesternukleinsäuren, Verfahren zu ihrer Herstellung und ihre Verwendung |
EP0739898B1 (fr) * | 1995-03-13 | 2001-09-26 | Aventis Pharma Deutschland GmbH | Phosphonomonoester acides nucléiques, leur préparation et leur utilisation |
DE19640974A1 (de) | 1996-10-04 | 1998-04-16 | Bayer Ag | Bausteine für DNA/PNA-Cooligomere |
DE19757516A1 (de) * | 1997-12-23 | 1999-06-24 | Roche Diagnostics Gmbh | Modifizierte Nukleinsäureanaloga |
US6326479B1 (en) * | 1998-01-27 | 2001-12-04 | Boston Probes, Inc. | Synthetic polymers and methods, kits or compositions for modulating the solubility of same |
US6043352A (en) * | 1998-08-07 | 2000-03-28 | Isis Pharmaceuticals, Inc. | 2'-O-Dimethylaminoethyloxyethyl-modified oligonucleotides |
DE10019135A1 (de) * | 2000-04-18 | 2001-10-31 | Aventis Pharma Gmbh | Polyamidnukleinsäure-Derivate, Mittel und Verfahren zu ihrer Herstellung |
DE10019136A1 (de) * | 2000-04-18 | 2001-10-31 | Aventis Pharma Gmbh | Polyamidnukleinsäure-Derivate, Mittel und Verfahren zu ihrer Herstellung |
-
2000
- 2000-04-18 DE DE10019135A patent/DE10019135A1/de not_active Ceased
-
2001
- 2001-04-07 PT PT01927897T patent/PT1276760E/pt unknown
- 2001-04-07 JP JP2001576814A patent/JP4908714B2/ja not_active Expired - Fee Related
- 2001-04-07 MX MXPA02009953A patent/MXPA02009953A/es active IP Right Grant
- 2001-04-07 WO PCT/EP2001/004030 patent/WO2001079216A2/fr active IP Right Grant
- 2001-04-07 DE DE50111371T patent/DE50111371D1/de not_active Expired - Lifetime
- 2001-04-07 BR BR0110110-2A patent/BR0110110A/pt not_active IP Right Cessation
- 2001-04-07 NZ NZ521988A patent/NZ521988A/xx not_active IP Right Cessation
- 2001-04-07 KR KR1020027013932A patent/KR100842723B1/ko not_active IP Right Cessation
- 2001-04-07 DK DK01927897T patent/DK1276760T3/da active
- 2001-04-07 AT AT01927897T patent/ATE344276T1/de active
- 2001-04-07 AU AU5479501A patent/AU5479501A/xx not_active Withdrawn
- 2001-04-07 ES ES01927897T patent/ES2275677T3/es not_active Expired - Lifetime
- 2001-04-07 EP EP01927897A patent/EP1276760B1/fr not_active Expired - Lifetime
- 2001-04-07 IL IL15228801A patent/IL152288A0/xx unknown
- 2001-04-07 CA CA2406169A patent/CA2406169C/fr not_active Expired - Fee Related
- 2001-04-16 AR ARP010101766A patent/AR032153A1/es unknown
- 2001-04-17 US US09/835,371 patent/US6905820B2/en not_active Expired - Fee Related
- 2001-05-16 TW TW090108986A patent/TWI298328B/zh not_active IP Right Cessation
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2002
- 2002-10-14 IL IL152288A patent/IL152288A/en not_active IP Right Cessation
- 2002-10-15 NO NO20024959A patent/NO333193B1/no not_active IP Right Cessation
- 2002-10-16 ZA ZA200208344A patent/ZA200208344B/en unknown
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2004
- 2004-06-02 US US10/858,658 patent/US20050009073A1/en not_active Abandoned
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2007
- 2007-01-29 CY CY20071100108T patent/CY1105958T1/el unknown
- 2007-09-14 US US11/855,443 patent/US7550582B2/en not_active Expired - Fee Related
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2009
- 2009-05-29 US US12/474,532 patent/US7897346B2/en not_active Expired - Fee Related
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2011
- 2011-01-24 US US13/012,266 patent/US8268560B2/en not_active Expired - Fee Related
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