NO329206B1 - Granulering og preparat med hoyt legemiddelinnhold, fremgangsmate for fremstilling derav og farmasoytisk preparat. - Google Patents
Granulering og preparat med hoyt legemiddelinnhold, fremgangsmate for fremstilling derav og farmasoytisk preparat. Download PDFInfo
- Publication number
- NO329206B1 NO329206B1 NO20002526A NO20002526A NO329206B1 NO 329206 B1 NO329206 B1 NO 329206B1 NO 20002526 A NO20002526 A NO 20002526A NO 20002526 A NO20002526 A NO 20002526A NO 329206 B1 NO329206 B1 NO 329206B1
- Authority
- NO
- Norway
- Prior art keywords
- drug content
- preparation
- high drug
- methylene
- methyl
- Prior art date
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Classifications
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- A—HUMAN NECESSITIES
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- A61K9/00—Medicinal preparations characterised by special physical form
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- A61K9/1682—Processes
- A61K9/1694—Processes resulting in granules or microspheres of the matrix type containing more than 5% of excipient
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- A—HUMAN NECESSITIES
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1682—Processes
- A61K9/1688—Processes resulting in pure drug agglomerate optionally containing up to 5% of excipient
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hospice & Palliative Care (AREA)
- Urology & Nephrology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US6591897P | 1997-11-17 | 1997-11-17 | |
| PCT/US1998/024502 WO1999025321A1 (en) | 1997-11-17 | 1998-11-17 | High drug load immediate and modified release oral dosage formulations and processes for their manufacture |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO20002526D0 NO20002526D0 (no) | 2000-05-16 |
| NO20002526L NO20002526L (no) | 2000-05-16 |
| NO329206B1 true NO329206B1 (no) | 2010-09-13 |
Family
ID=22066009
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20002526A NO329206B1 (no) | 1997-11-17 | 2000-05-16 | Granulering og preparat med hoyt legemiddelinnhold, fremgangsmate for fremstilling derav og farmasoytisk preparat. |
Country Status (14)
| Country | Link |
|---|---|
| EP (1) | EP1033974B1 (ja) |
| JP (1) | JP4880118B2 (ja) |
| KR (1) | KR100597922B1 (ja) |
| CN (1) | CN1285739A (ja) |
| AU (1) | AU750611B2 (ja) |
| BR (1) | BR9814877A (ja) |
| CA (1) | CA2310028C (ja) |
| HU (1) | HUP0004407A3 (ja) |
| IL (1) | IL136142A0 (ja) |
| NO (1) | NO329206B1 (ja) |
| NZ (1) | NZ504565A (ja) |
| PL (1) | PL340587A1 (ja) |
| TR (1) | TR200001412T2 (ja) |
| WO (1) | WO1999025321A1 (ja) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL140905A0 (en) * | 1998-07-20 | 2002-02-10 | Smithkline Beecham Corp | Bioenhanced formulations comprising eprosartan in oral solid dosage form |
| EP1242057A2 (en) | 1999-11-02 | 2002-09-25 | DepoMed, Inc. | Pharmacological inducement of the fed mode for enhanced drug administration to the stomach |
| GB0209265D0 (en) | 2002-04-23 | 2002-06-05 | Novartis Ag | Organic compounds |
| GB0228878D0 (en) * | 2002-06-21 | 2003-01-15 | Unilever Plc | Hair conditioning composition |
| JP3874419B2 (ja) | 2003-01-31 | 2007-01-31 | 三共株式会社 | 動脈硬化及び高血圧症の予防及び治療のための医薬 |
| AU2007249399A1 (en) * | 2006-05-09 | 2007-11-22 | Braincells, Inc. | Neurogenesis by modulating angiotensin |
| PT2295035T (pt) * | 2007-11-06 | 2016-08-22 | Novartis Ag | Composições farmacêuticas de dupla acção com base em superestruturas de antagonista/bloqueador de receptores de angiotensina (arb) com inibidor da endopeptidase neutra (nep) |
| AR072477A1 (es) * | 2008-07-11 | 2010-09-01 | Solvay Pharm Bv | Formulacion farmaceutica de eprosartan. uso. |
| JP5476782B2 (ja) * | 2009-04-21 | 2014-04-23 | 大正製薬株式会社 | アルギニン含有錠剤の製造方法 |
| JP5446716B2 (ja) * | 2009-10-21 | 2014-03-19 | 大正製薬株式会社 | アルギニン及びカルニチン含有錠剤の製造方法 |
| TR201007508A1 (tr) * | 2010-09-14 | 2012-04-24 | Sanovel İlaç San. Ve Ti̇c. A.Ş. | Oral yolla dağılan bileşimler |
| CN104546779A (zh) * | 2013-10-14 | 2015-04-29 | 深圳海王药业有限公司 | 高药物荷载的枸橼酸西地那非片剂及其制备方法 |
| WO2019072877A1 (en) * | 2017-10-10 | 2019-04-18 | Capsugel Belgium Nv | GETTING MULTIPARTICULAR COMPOSITIONS |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5185351A (en) * | 1989-06-14 | 1993-02-09 | Smithkline Beecham Corporation | Imidazolyl-alkenoic acids useful as angiotensin II receptor antagonists |
| EP0563238B1 (en) * | 1990-12-14 | 2002-05-22 | Smithkline Beecham Corporation | Imidazolyl-alkenoic acids |
| CA2168647A1 (en) * | 1993-08-02 | 1995-02-09 | Barbara A. Sosnowski | Monogenous preparations of cytotoxic conjugates |
| ES2198564T3 (es) * | 1996-03-29 | 2004-02-01 | Smithkline Beecham Corporation | Dihidrato de eprosartan y un procedimiento para su produccion y formulacion. |
-
1998
- 1998-11-17 CA CA002310028A patent/CA2310028C/en not_active Expired - Fee Related
- 1998-11-17 AU AU15887/99A patent/AU750611B2/en not_active Ceased
- 1998-11-17 HU HU0004407A patent/HUP0004407A3/hu not_active Application Discontinuation
- 1998-11-17 BR BR9814877-0A patent/BR9814877A/pt not_active Application Discontinuation
- 1998-11-17 PL PL98340587A patent/PL340587A1/xx not_active Application Discontinuation
- 1998-11-17 EP EP98960242.0A patent/EP1033974B1/en not_active Expired - Lifetime
- 1998-11-17 KR KR1020007005316A patent/KR100597922B1/ko not_active IP Right Cessation
- 1998-11-17 TR TR2000/01412T patent/TR200001412T2/xx unknown
- 1998-11-17 IL IL13614298A patent/IL136142A0/xx not_active IP Right Cessation
- 1998-11-17 NZ NZ504565A patent/NZ504565A/xx not_active IP Right Cessation
- 1998-11-17 JP JP2000520755A patent/JP4880118B2/ja not_active Expired - Fee Related
- 1998-11-17 CN CN98813140A patent/CN1285739A/zh active Pending
- 1998-11-17 WO PCT/US1998/024502 patent/WO1999025321A1/en active IP Right Grant
-
2000
- 2000-05-16 NO NO20002526A patent/NO329206B1/no not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| KR100597922B1 (ko) | 2006-07-10 |
| KR20010032129A (ko) | 2001-04-16 |
| AU1588799A (en) | 1999-06-07 |
| CN1285739A (zh) | 2001-02-28 |
| EP1033974B1 (en) | 2014-01-22 |
| AU750611B2 (en) | 2002-07-25 |
| BR9814877A (pt) | 2000-10-03 |
| JP2001522872A (ja) | 2001-11-20 |
| CA2310028C (en) | 2008-06-10 |
| NZ504565A (en) | 2002-11-26 |
| CA2310028A1 (en) | 1999-05-27 |
| TR200001412T2 (tr) | 2000-09-21 |
| WO1999025321A1 (en) | 1999-05-27 |
| PL340587A1 (en) | 2001-02-12 |
| IL136142A0 (en) | 2001-05-20 |
| HUP0004407A3 (en) | 2002-03-28 |
| NO20002526D0 (no) | 2000-05-16 |
| JP4880118B2 (ja) | 2012-02-22 |
| HUP0004407A1 (hu) | 2002-02-28 |
| NO20002526L (no) | 2000-05-16 |
| EP1033974A1 (en) | 2000-09-13 |
| EP1033974A4 (en) | 2007-05-02 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM1K | Lapsed by not paying the annual fees |