NO327296B1 - Ny medisinsk anvendelse av 4α-acetoksy-2α-benzoyloksy-5β,20-epoksy-1β-hydroksy-7β,10β-dimetoksy-9-okso-11-taxen-13α-yl(2R,3S)-3-tert-butoksykarbonylamino-2-hydroksy-3-fenylpropionat. - Google Patents
Ny medisinsk anvendelse av 4α-acetoksy-2α-benzoyloksy-5β,20-epoksy-1β-hydroksy-7β,10β-dimetoksy-9-okso-11-taxen-13α-yl(2R,3S)-3-tert-butoksykarbonylamino-2-hydroksy-3-fenylpropionat. Download PDFInfo
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- NO327296B1 NO327296B1 NO20010654A NO20010654A NO327296B1 NO 327296 B1 NO327296 B1 NO 327296B1 NO 20010654 A NO20010654 A NO 20010654A NO 20010654 A NO20010654 A NO 20010654A NO 327296 B1 NO327296 B1 NO 327296B1
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Classifications
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- A61K31/00—Medicinal preparations containing organic active ingredients
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/19—Cytokines; Lymphokines; Interferons
- A61K38/191—Tumor necrosis factors [TNF], e.g. lymphotoxin [LT], i.e. TNF-beta
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/19—Cytokines; Lymphokines; Interferons
- A61K38/20—Interleukins [IL]
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/19—Cytokines; Lymphokines; Interferons
- A61K38/21—Interferons [IFN]
- A61K38/212—IFN-alpha
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/19—Cytokines; Lymphokines; Interferons
- A61K38/21—Interferons [IFN]
- A61K38/215—IFN-beta
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
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- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Immunology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Zoology (AREA)
- Gastroenterology & Hepatology (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Epoxy Compounds (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP98115401A EP0982027A1 (en) | 1998-08-17 | 1998-08-17 | Taxoid derivatives for treating abnormal cell proliferation of the brain |
| US9958198P | 1998-09-08 | 1998-09-08 | |
| PCT/EP1999/006291 WO2000009120A1 (en) | 1998-08-17 | 1999-08-13 | New use of taxoid derivatives |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO20010654D0 NO20010654D0 (no) | 2001-02-07 |
| NO20010654L NO20010654L (no) | 2001-02-07 |
| NO327296B1 true NO327296B1 (no) | 2009-06-02 |
Family
ID=26149540
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20010654A NO327296B1 (no) | 1998-08-17 | 2001-02-07 | Ny medisinsk anvendelse av 4α-acetoksy-2α-benzoyloksy-5β,20-epoksy-1β-hydroksy-7β,10β-dimetoksy-9-okso-11-taxen-13α-yl(2R,3S)-3-tert-butoksykarbonylamino-2-hydroksy-3-fenylpropionat. |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US6346543B1 (et) |
| EP (1) | EP1109547A1 (et) |
| JP (1) | JP5354762B2 (et) |
| KR (1) | KR100710533B1 (et) |
| AU (1) | AU766168B2 (et) |
| BG (1) | BG65365B1 (et) |
| CA (1) | CA2340921C (et) |
| CZ (1) | CZ293959B6 (et) |
| EE (1) | EE04903B1 (et) |
| HU (1) | HU230235B1 (et) |
| ID (1) | ID27545A (et) |
| IL (1) | IL141238A0 (et) |
| ME (1) | ME00533B (et) |
| NO (1) | NO327296B1 (et) |
| NZ (1) | NZ509965A (et) |
| RS (1) | RS52011B (et) |
| SK (1) | SK285212B6 (et) |
| TR (1) | TR200100557T2 (et) |
| WO (1) | WO2000009120A1 (et) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2686899B1 (fr) * | 1992-01-31 | 1995-09-01 | Rhone Poulenc Rorer Sa | Nouveaux polypeptides biologiquement actifs, leur preparation et compositions pharmaceutiques les contenant. |
| EP1020188A1 (en) * | 1999-01-13 | 2000-07-19 | Aventis Pharma S.A. | New use of taxoid derivatives |
| CA2405557C (en) * | 2000-04-12 | 2013-09-24 | Human Genome Sciences, Inc. | Albumin fusion proteins |
| WO2002097038A2 (en) * | 2001-05-25 | 2002-12-05 | Human Genome Sciences, Inc. | Chemokine beta-1 fusion proteins |
| ES2545090T3 (es) * | 2001-12-21 | 2015-09-08 | Human Genome Sciences, Inc. | Proteínas de fusión de albúmina y GCSF |
| WO2003059934A2 (en) * | 2001-12-21 | 2003-07-24 | Human Genome Sciences, Inc. | Albumin fusion proteins |
| FR2859996B1 (fr) * | 2003-09-19 | 2006-02-03 | Aventis Pharma Sa | Solvat acetonique du dimethoxy docetaxel et son procede de preparation |
| FR2926551A1 (fr) * | 2008-01-17 | 2009-07-24 | Aventis Pharma Sa | Formes cristallines du dimethoxy docetaxel et leurs procedes de preparation |
| EP2331140B1 (en) | 2008-08-11 | 2018-07-04 | Nektar Therapeutics | Multi-arm polymeric alkanoate conjugates |
| WO2011051894A1 (en) | 2009-10-29 | 2011-05-05 | Aventis Pharma S.A. | Novel antitumoral use of cabazitaxel |
| US20130331443A1 (en) | 2010-12-22 | 2013-12-12 | Nektar Therapeutics | Multi-arm polymeric prodrug conjugates of taxane-based compounds |
| US10894087B2 (en) | 2010-12-22 | 2021-01-19 | Nektar Therapeutics | Multi-arm polymeric prodrug conjugates of cabazitaxel-based compounds |
| WO2013088335A1 (en) | 2011-12-13 | 2013-06-20 | Aventis Pharma S.A. | Crystalline form of cabazitaxel and process for preparing the same |
| BR112014019675A2 (pt) * | 2012-02-10 | 2017-07-11 | Aventis Pharma Sa | usos pediátricos de cabazitaxel |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MX9102128A (es) * | 1990-11-23 | 1992-07-08 | Rhone Poulenc Rorer Sa | Derivados de taxano,procedimiento para su preparacion y composicion farmaceutica que los contiene |
| FR2696459B1 (fr) | 1992-10-05 | 1994-11-25 | Rhone Poulenc Rorer Sa | Procédé de préparation de dérivés du taxane. |
| TW467896B (en) | 1993-03-19 | 2001-12-11 | Bristol Myers Squibb Co | Novel β-lactams, methods for the preparation of taxanes and sidechain-bearing taxanes |
| US5847170A (en) * | 1995-03-27 | 1998-12-08 | Rhone-Poulenc Rorer, S.A. | Taxoids, their preparation and pharmaceutical compositions containing them |
| MA23823A1 (fr) * | 1995-03-27 | 1996-10-01 | Aventis Pharma Sa | Nouveaux taxoides, leur preparation et les compositions qui les contiennent |
| US5481018A (en) | 1995-03-31 | 1996-01-02 | The Dow Chemical Company | Amino nitrile intermediate for the preparation of alanine diacetic acid |
| FR2771092B1 (fr) | 1997-11-18 | 1999-12-17 | Rhone Poulenc Rorer Sa | Procede de preparation de derives de la classe des taxoides |
-
1999
- 1999-08-11 US US09/371,838 patent/US6346543B1/en not_active Expired - Lifetime
- 1999-08-13 AU AU57419/99A patent/AU766168B2/en not_active Expired
- 1999-08-13 KR KR1020017001970A patent/KR100710533B1/ko not_active IP Right Cessation
- 1999-08-13 JP JP2000564623A patent/JP5354762B2/ja not_active Expired - Lifetime
- 1999-08-13 CA CA002340921A patent/CA2340921C/en not_active Expired - Lifetime
- 1999-08-13 TR TR2001/00557T patent/TR200100557T2/xx unknown
- 1999-08-13 HU HU0103748A patent/HU230235B1/hu unknown
- 1999-08-13 IL IL14123899A patent/IL141238A0/xx not_active IP Right Cessation
- 1999-08-13 EE EEP200100079A patent/EE04903B1/et unknown
- 1999-08-13 ME MEP-2008-893A patent/ME00533B/me unknown
- 1999-08-13 WO PCT/EP1999/006291 patent/WO2000009120A1/en not_active Application Discontinuation
- 1999-08-13 EP EP99944531A patent/EP1109547A1/en not_active Withdrawn
- 1999-08-13 RS YU7901A patent/RS52011B/sr unknown
- 1999-08-13 SK SK230-2001A patent/SK285212B6/sk not_active IP Right Cessation
- 1999-08-13 ID IDW20010379A patent/ID27545A/id unknown
- 1999-08-13 CZ CZ2001604A patent/CZ293959B6/cs not_active IP Right Cessation
- 1999-08-13 NZ NZ509965A patent/NZ509965A/en not_active IP Right Cessation
-
2001
- 2001-02-07 NO NO20010654A patent/NO327296B1/no not_active IP Right Cessation
- 2001-02-16 BG BG105264A patent/BG65365B1/bg unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ID27545A (id) | 2001-04-12 |
| CA2340921C (en) | 2009-01-06 |
| CA2340921A1 (en) | 2000-02-24 |
| HUP0103748A2 (hu) | 2002-04-29 |
| CZ2001604A3 (en) | 2001-06-13 |
| SK2302001A3 (en) | 2001-09-11 |
| WO2000009120A1 (en) | 2000-02-24 |
| BG105264A (en) | 2001-11-30 |
| AU766168B2 (en) | 2003-10-09 |
| ME00533B (me) | 2011-10-10 |
| YU7901A (sh) | 2003-12-31 |
| US6346543B1 (en) | 2002-02-12 |
| NO20010654D0 (no) | 2001-02-07 |
| EP1109547A1 (en) | 2001-06-27 |
| WO2000009120A8 (en) | 2001-04-05 |
| KR20010085396A (ko) | 2001-09-07 |
| HU230235B1 (hu) | 2015-10-28 |
| EE200100079A (et) | 2002-08-15 |
| NZ509965A (en) | 2003-09-26 |
| AU5741999A (en) | 2000-03-06 |
| CZ293959B6 (cs) | 2004-08-18 |
| JP5354762B2 (ja) | 2013-11-27 |
| EE04903B1 (et) | 2007-10-15 |
| SK285212B6 (sk) | 2006-09-07 |
| TR200100557T2 (tr) | 2001-07-23 |
| KR100710533B1 (ko) | 2007-04-23 |
| NO20010654L (no) | 2001-02-07 |
| BG65365B1 (bg) | 2008-04-30 |
| HUP0103748A3 (en) | 2003-01-28 |
| RS52011B (sr) | 2012-04-30 |
| IL141238A0 (en) | 2002-03-10 |
| JP2002522490A (ja) | 2002-07-23 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MK1K | Patent expired |