NO323076B1 - Forbindelser, preparater, nevnte forbindelser og preparater for bruk i terapi samt anvendelse av nevnte forbindelser for fremstilling av preparater til medisinsk behandling. - Google Patents
Forbindelser, preparater, nevnte forbindelser og preparater for bruk i terapi samt anvendelse av nevnte forbindelser for fremstilling av preparater til medisinsk behandling. Download PDFInfo
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- NO323076B1 NO323076B1 NO20022009A NO20022009A NO323076B1 NO 323076 B1 NO323076 B1 NO 323076B1 NO 20022009 A NO20022009 A NO 20022009A NO 20022009 A NO20022009 A NO 20022009A NO 323076 B1 NO323076 B1 NO 323076B1
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Classifications
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- C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
- C07D407/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
- C07D407/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/18—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
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- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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- Psychiatry (AREA)
- Psychology (AREA)
- Pain & Pain Management (AREA)
- Addiction (AREA)
- Epidemiology (AREA)
- Toxicology (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pyridine Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE9903997A SE9903997D0 (sv) | 1999-11-03 | 1999-11-03 | New compounds |
| PCT/SE2000/002148 WO2001032619A1 (en) | 1999-11-03 | 2000-11-01 | Positive modulators of nicotinic receptor agonists |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO20022009D0 NO20022009D0 (no) | 2002-04-26 |
| NO20022009L NO20022009L (no) | 2002-07-02 |
| NO323076B1 true NO323076B1 (no) | 2006-12-27 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20022009A NO323076B1 (no) | 1999-11-03 | 2002-04-26 | Forbindelser, preparater, nevnte forbindelser og preparater for bruk i terapi samt anvendelse av nevnte forbindelser for fremstilling av preparater til medisinsk behandling. |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US6750242B1 (https=) |
| EP (1) | EP1230216A1 (https=) |
| JP (1) | JP2003513071A (https=) |
| KR (1) | KR20020063176A (https=) |
| CN (1) | CN1239482C (https=) |
| AU (1) | AU783507B2 (https=) |
| BR (1) | BR0015195A (https=) |
| CA (1) | CA2387745A1 (https=) |
| CO (1) | CO5251458A1 (https=) |
| IL (1) | IL149098A0 (https=) |
| MX (1) | MXPA02004232A (https=) |
| NO (1) | NO323076B1 (https=) |
| NZ (2) | NZ518450A (https=) |
| SE (1) | SE9903997D0 (https=) |
| WO (1) | WO2001032619A1 (https=) |
| ZA (1) | ZA200203171B (https=) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE9903998D0 (sv) * | 1999-11-03 | 1999-11-03 | Astra Ab | New compounds |
| DE10164139A1 (de) | 2001-12-27 | 2003-07-10 | Bayer Ag | 2-Heteroarylcarbonsäureamide |
| DE10234424A1 (de) * | 2002-07-29 | 2004-02-12 | Bayer Ag | Benzothiophen-, Benzofuran- und Indolharnstoffe |
| US7244745B2 (en) | 2002-08-30 | 2007-07-17 | Memory Pharmaceuticals Corp. | Heterocyclic compounds, methods for the preparation thereof, and uses thereof |
| MXPA05003317A (es) | 2002-09-25 | 2005-07-05 | Memory Pharm Corp | Indazoles, benzotiazoles y benzoisotiazoles asi como preparacion y usos de los mismos. |
| EP1735306A2 (en) | 2004-03-25 | 2006-12-27 | Memory Pharmaceuticals Corporation | Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, and preparation and uses thereof |
| ZA200709038B (en) * | 2005-04-13 | 2009-01-28 | Neuraxon Inc | Substituted indole compounds having nos inhibitory activity |
| US20070134169A1 (en) * | 2005-12-11 | 2007-06-14 | Rabinoff Michael D | Methods for smoking cessation or alcohol cessation or other addiction cessation |
| CN101466709B (zh) * | 2006-04-13 | 2013-03-20 | 轴突公司 | 具有nos抑制活性的1,5和3,6-取代的吲哚化合物 |
| WO2009062318A1 (en) * | 2007-11-16 | 2009-05-22 | Neuraxon, Inc. | 3,5-substituted indole compounds having nos and norepinephrine reuptake inhibitory activity |
| EP2219449A4 (en) * | 2007-11-16 | 2010-10-27 | Univ Arizona State | METHOD FOR THE TREATMENT OF EXPOSURE TO DAMAGING |
| EA201000808A1 (ru) | 2007-11-16 | 2011-04-29 | Ньюраксон, Инк. | Индольные соединения и способы лечения висцеральной боли |
| US8383657B2 (en) | 2007-12-21 | 2013-02-26 | Abbott Laboratories | Thiazolylidine urea and amide derivatives and methods of use thereof |
| JP2011511800A (ja) * | 2008-02-07 | 2011-04-14 | アボット・ラボラトリーズ | 正のアロステリックな修飾物質としてのアミド誘導体およびこれらの使用方法 |
| TW201004939A (en) * | 2008-04-17 | 2010-02-01 | Glaxo Group Ltd | Novel compounds |
| EP2419420B1 (en) * | 2009-04-16 | 2013-03-13 | Proximagen Limited | Indole derivative modulators of the alpha 7 nachr |
| PE20170923A1 (es) * | 2010-05-17 | 2017-07-12 | Forum Pharmaceuticals Inc | Una forma cristalina de clorhidrato de (r)-7-cloro-n-(quinuclidin-3-il)benzo[b]tiofeno-2-carboxamida monohidratado |
| TW201245185A (en) | 2011-04-01 | 2012-11-16 | Lundbeck & Co As H | New positive allosteric modulators of nicotinic acetylcholine receptor |
| AR086791A1 (es) | 2011-07-01 | 2014-01-22 | Lundbeck & Co As H | Moduladores alostericos positivos del receptor de acetilcolina nicotinico |
| EP3461481A1 (en) | 2012-05-08 | 2019-04-03 | Forum Pharmaceuticals Inc. | Methods of maintaining, treating or improving cognitive function |
| WO2020045982A1 (ko) * | 2018-08-29 | 2020-03-05 | 숙명여자대학교산학협력단 | 치환된 인돌 유도체, 이의 제조방법 및 이를 유효성분으로 포함하는 PPARα, PPARγ 및 PPARδ 관련 질환의 예방 또는 치료용 약학적 조성물 |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2787551A (en) * | 1954-02-24 | 1957-04-02 | Eastman Kodak Co | Compositions stabilized with hydroxyindole |
| BE758766A (fr) * | 1969-11-17 | 1971-05-10 | Ici Ltd | Nouveaux derives de la morpholine et de la |
| US4704390A (en) * | 1986-02-13 | 1987-11-03 | Warner-Lambert Company | Phenyl and heterocyclic tetrahydropyridyl alkoxy-benzheterocyclic compounds as antipsychotic agents |
| IE913204A1 (en) * | 1990-09-13 | 1992-02-25 | Beecham Group Plc | Novel compounds |
| HUT69705A (en) * | 1991-11-25 | 1995-09-28 | Pfizer | Indole derivatives |
| WO1993018026A1 (en) * | 1992-03-04 | 1993-09-16 | Beecham Group Plc | Indole ureas as 5-ht1c receptor antogonists |
| US5504101A (en) * | 1994-05-06 | 1996-04-02 | Allelix Biopharmaceuticals, Inc. | 5-HT-1D receptor ligands |
| FR2722686B1 (fr) * | 1994-07-22 | 1996-08-30 | Oreal | Set, procede, dispositif et composition de teinture des fibres keratiniques |
| US5576321A (en) * | 1995-01-17 | 1996-11-19 | Eli Lilly And Company | Compounds having effects on serotonin-related systems |
-
1999
- 1999-11-03 SE SE9903997A patent/SE9903997D0/xx unknown
-
2000
- 2000-11-01 CA CA002387745A patent/CA2387745A1/en not_active Abandoned
- 2000-11-01 JP JP2001534771A patent/JP2003513071A/ja not_active Abandoned
- 2000-11-01 BR BR0015195-5A patent/BR0015195A/pt not_active IP Right Cessation
- 2000-11-01 EP EP00976500A patent/EP1230216A1/en not_active Withdrawn
- 2000-11-01 US US10/111,027 patent/US6750242B1/en not_active Expired - Fee Related
- 2000-11-01 CN CNB008154414A patent/CN1239482C/zh not_active Expired - Fee Related
- 2000-11-01 NZ NZ518450A patent/NZ518450A/en unknown
- 2000-11-01 KR KR1020027005706A patent/KR20020063176A/ko not_active Ceased
- 2000-11-01 WO PCT/SE2000/002148 patent/WO2001032619A1/en not_active Ceased
- 2000-11-01 CO CO00083175A patent/CO5251458A1/es not_active Application Discontinuation
- 2000-11-01 IL IL14909800A patent/IL149098A0/xx unknown
- 2000-11-01 NZ NZ530161A patent/NZ530161A/en unknown
- 2000-11-01 MX MXPA02004232A patent/MXPA02004232A/es unknown
- 2000-11-01 AU AU14264/01A patent/AU783507B2/en not_active Ceased
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2002
- 2002-04-22 ZA ZA200203171A patent/ZA200203171B/xx unknown
- 2002-04-26 NO NO20022009A patent/NO323076B1/no unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CA2387745A1 (en) | 2001-05-10 |
| AU1426401A (en) | 2001-05-14 |
| WO2001032619A1 (en) | 2001-05-10 |
| US6750242B1 (en) | 2004-06-15 |
| IL149098A0 (en) | 2002-11-10 |
| CN1239482C (zh) | 2006-02-01 |
| NO20022009D0 (no) | 2002-04-26 |
| ZA200203171B (en) | 2003-09-23 |
| EP1230216A1 (en) | 2002-08-14 |
| CN1387512A (zh) | 2002-12-25 |
| NZ530161A (en) | 2005-08-26 |
| AU783507B2 (en) | 2005-11-03 |
| JP2003513071A (ja) | 2003-04-08 |
| SE9903997D0 (sv) | 1999-11-03 |
| KR20020063176A (ko) | 2002-08-01 |
| CO5251458A1 (es) | 2003-02-28 |
| NO20022009L (no) | 2002-07-02 |
| MXPA02004232A (es) | 2002-10-17 |
| BR0015195A (pt) | 2002-06-18 |
| NZ518450A (en) | 2004-04-30 |
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