NO322752B1 - Polymorfismer av N-metyl-N-(3{3-[2-tienylkarbonyl]pyrazol-[1,5-alfa]-pyrimidin-7-yl}fenyl)acetamid og blandinger og fremgangsmater relatert dertil - Google Patents
Polymorfismer av N-metyl-N-(3{3-[2-tienylkarbonyl]pyrazol-[1,5-alfa]-pyrimidin-7-yl}fenyl)acetamid og blandinger og fremgangsmater relatert dertil Download PDFInfo
- Publication number
- NO322752B1 NO322752B1 NO20021041A NO20021041A NO322752B1 NO 322752 B1 NO322752 B1 NO 322752B1 NO 20021041 A NO20021041 A NO 20021041A NO 20021041 A NO20021041 A NO 20021041A NO 322752 B1 NO322752 B1 NO 322752B1
- Authority
- NO
- Norway
- Prior art keywords
- polymorphic form
- phenyl
- acetamide
- methyl
- pyrimidin
- Prior art date
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- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicinal Preparation (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US38952499A | 1999-09-02 | 1999-09-02 | |
| US42162099A | 1999-10-19 | 1999-10-19 | |
| PCT/US2000/024051 WO2001015700A1 (en) | 1999-09-02 | 2000-09-01 | POLYMORPHS OF N-METHYL-N-(3-{3-[2-THIENYLCARBONYL]-PYRAZOL-[1,5-α]-PYRIMIDIN -7-YL }PHENYL )ACETAMIDE AND COMPOSITIONS AND METHODS RELATED THERETO |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO20021041D0 NO20021041D0 (no) | 2002-03-01 |
| NO20021041L NO20021041L (no) | 2002-04-03 |
| NO322752B1 true NO322752B1 (no) | 2006-12-04 |
Family
ID=27012737
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20021041A NO322752B1 (no) | 1999-09-02 | 2002-03-01 | Polymorfismer av N-metyl-N-(3{3-[2-tienylkarbonyl]pyrazol-[1,5-alfa]-pyrimidin-7-yl}fenyl)acetamid og blandinger og fremgangsmater relatert dertil |
Country Status (26)
| Country | Link |
|---|---|
| EP (2) | EP1477169A1 (pl) |
| JP (1) | JP4592241B2 (pl) |
| KR (1) | KR20020035585A (pl) |
| CN (2) | CN1198824C (pl) |
| AP (1) | AP1631A (pl) |
| AT (1) | ATE269082T1 (pl) |
| AU (2) | AU769856B2 (pl) |
| BR (1) | BR0014459A (pl) |
| CA (1) | CA2382588C (pl) |
| CZ (1) | CZ2002783A3 (pl) |
| DE (1) | DE60011638T2 (pl) |
| DK (1) | DK1214075T3 (pl) |
| EA (1) | EA004706B1 (pl) |
| ES (1) | ES2222920T3 (pl) |
| HK (1) | HK1047407B (pl) |
| HU (1) | HUP0202698A3 (pl) |
| IL (2) | IL148242A0 (pl) |
| MX (1) | MXPA02002314A (pl) |
| NO (1) | NO322752B1 (pl) |
| NZ (1) | NZ517298A (pl) |
| OA (1) | OA12200A (pl) |
| PL (1) | PL353362A1 (pl) |
| PT (1) | PT1214075E (pl) |
| SK (1) | SK2782002A3 (pl) |
| TR (1) | TR200200534T2 (pl) |
| WO (1) | WO2001015700A1 (pl) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE343581T1 (de) * | 2002-08-26 | 2006-11-15 | Neurocrine Biosciences Inc | Polymorph von n-methyl-n-(3- 3- 2-[thienylcarbonylö-pyrazol-[1,5-alphaö-pyrimidin- - yl phenyl)acetamid und zusammensetzungen sowie verfahren hierzu |
| WO2004110454A1 (ja) * | 2003-06-13 | 2004-12-23 | Ishihara Sangyo Kaisha, Ltd. | アデノシンＡ2ａ受容体アゴニストの投与が必要な疾患を治療又は予防するための組成物 |
| US7371906B2 (en) * | 2004-08-24 | 2008-05-13 | Eastman Kodak Company | Process for photo-oxidative stability improvements |
| EP1956021A1 (en) * | 2006-10-11 | 2008-08-13 | Ferrer Internacional, S.A. | Process for the manufacture of a crystalline pyrazolo[1,5-a]pyrimidine compound |
| EP1918290A1 (en) * | 2006-10-11 | 2008-05-07 | Ferrer Internacional, S.A. | Polymorph B of N-{2-Fluoro-5-[3-(thiophene-2-carbonyl)-pyrazolo[1,5-a] pyrimidin-7-yl]-phenyl}-N-methyl-acetamide |
| CN101177427B (zh) * | 2006-11-09 | 2011-07-20 | 中国人民解放军军事医学科学院放射与辐射医学研究所 | 一种用于催眠的化合物的多晶型α和溶剂化物,其制备方法及含该物质的组合物 |
| WO2010109480A2 (en) * | 2009-03-24 | 2010-09-30 | Glenmark Generics Limited | Processes for the preparation of indiplon and intermediates thereof |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4654347A (en) * | 1983-06-23 | 1987-03-31 | American Cyanamid Company | Aryl and heteroaryl[[7-(3-disubstituted amino)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]methanones |
| NZ208554A (en) * | 1983-06-23 | 1987-06-30 | American Cyanamid Co | (aryl and heteroaryl)-(7-(aryl and heteroaryl)-pyrazolo (1,5-a) pyrimidin-3-yl)-methanone derivatives and pharmaceutical compositions |
| US4521422A (en) * | 1983-06-23 | 1985-06-04 | American Cyanamid Company | Aryl and heteroaryl[7-(aryl and heteroaryl)pyrazolo[1,5-a]pyrimidin-3-yl]methanones |
| US4626538A (en) * | 1983-06-23 | 1986-12-02 | American Cyanamid Company | [7-(3-disubstituted amino)phenyl]pyrazolo[1,5-a]pyrimidines |
| DE19975048I2 (de) * | 1985-05-13 | 2001-06-13 | American Cyanamid Co | 7-(3-Disubstituierte Amino)phenyl pyrazolo 1,5-a -pyrimidine |
| US5421422A (en) * | 1993-11-19 | 1995-06-06 | Boretec Inc | Roller cutter mount for tunneling machine |
-
2000
- 2000-09-01 DE DE60011638T patent/DE60011638T2/de not_active Expired - Lifetime
- 2000-09-01 JP JP2001519914A patent/JP4592241B2/ja not_active Expired - Lifetime
- 2000-09-01 TR TR2002/00534T patent/TR200200534T2/xx unknown
- 2000-09-01 AT AT00957941T patent/ATE269082T1/de active
- 2000-09-01 IL IL14824200A patent/IL148242A0/xx active IP Right Grant
- 2000-09-01 EP EP04013998A patent/EP1477169A1/en not_active Withdrawn
- 2000-09-01 AU AU69491/00A patent/AU769856B2/en not_active Ceased
- 2000-09-01 SK SK278-2002A patent/SK2782002A3/sk unknown
- 2000-09-01 NZ NZ517298A patent/NZ517298A/en not_active IP Right Cessation
- 2000-09-01 WO PCT/US2000/024051 patent/WO2001015700A1/en not_active Ceased
- 2000-09-01 MX MXPA02002314A patent/MXPA02002314A/es active IP Right Grant
- 2000-09-01 AP APAP/P/2002/002428A patent/AP1631A/en active
- 2000-09-01 KR KR1020027002829A patent/KR20020035585A/ko not_active Ceased
- 2000-09-01 CA CA002382588A patent/CA2382588C/en not_active Expired - Fee Related
- 2000-09-01 EP EP00957941A patent/EP1214075B1/en not_active Expired - Lifetime
- 2000-09-01 CN CNB008131589A patent/CN1198824C/zh not_active Expired - Fee Related
- 2000-09-01 CN CNB2005100545485A patent/CN1331865C/zh not_active Expired - Fee Related
- 2000-09-01 PT PT00957941T patent/PT1214075E/pt unknown
- 2000-09-01 BR BR0014459-2A patent/BR0014459A/pt not_active Application Discontinuation
- 2000-09-01 HU HU0202698A patent/HUP0202698A3/hu unknown
- 2000-09-01 HK HK02109094.4A patent/HK1047407B/en not_active IP Right Cessation
- 2000-09-01 PL PL00353362A patent/PL353362A1/pl not_active Application Discontinuation
- 2000-09-01 CZ CZ2002783A patent/CZ2002783A3/cs unknown
- 2000-09-01 OA OA1200200057A patent/OA12200A/en unknown
- 2000-09-01 ES ES00957941T patent/ES2222920T3/es not_active Expired - Lifetime
- 2000-09-01 DK DK00957941T patent/DK1214075T3/da active
- 2000-09-01 EA EA200200320A patent/EA004706B1/ru not_active IP Right Cessation
-
2002
- 2002-02-19 IL IL148242A patent/IL148242A/en not_active IP Right Cessation
- 2002-03-01 NO NO20021041A patent/NO322752B1/no not_active IP Right Cessation
-
2004
- 2004-03-31 AU AU2004201356A patent/AU2004201356A1/en not_active Abandoned
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| Date | Code | Title | Description |
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| MM1K | Lapsed by not paying the annual fees |