NO313535B1 - Anvendelse av duloksetin for fremstilling av et farmasöytisk preparat for behandling av urininkontinens - Google Patents
Anvendelse av duloksetin for fremstilling av et farmasöytisk preparat for behandling av urininkontinens Download PDFInfo
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- NO313535B1 NO313535B1 NO19944456A NO944456A NO313535B1 NO 313535 B1 NO313535 B1 NO 313535B1 NO 19944456 A NO19944456 A NO 19944456A NO 944456 A NO944456 A NO 944456A NO 313535 B1 NO313535 B1 NO 313535B1
- Authority
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- Norway
- Prior art keywords
- bladder
- duloxetine
- incontinence
- activity
- mixture
- Prior art date
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- A61K31/341—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide not condensed with another ring, e.g. ranitidine, furosemide, bufetolol, muscarine
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Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
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- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
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- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Urology & Nephrology (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Saccharide Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Furan Compounds (AREA)
- Pyridine Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- External Artificial Organs (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US15812193A | 1993-11-24 | 1993-11-24 |
Publications (3)
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| NO944456D0 NO944456D0 (no) | 1994-11-21 |
| NO944456L NO944456L (no) | 1995-05-26 |
| NO313535B1 true NO313535B1 (no) | 2002-10-21 |
Family
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| Application Number | Title | Priority Date | Filing Date |
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| NO19944456A NO313535B1 (no) | 1993-11-24 | 1994-11-21 | Anvendelse av duloksetin for fremstilling av et farmasöytisk preparat for behandling av urininkontinens |
| NO2005004C NO2005004I1 (no) | 1993-11-24 | 2005-02-09 | Duloksetin og dets farmasøytisk akseptable syreaddisjonssalter, spesielt duloksetin hydroklorid |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
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| NO2005004C NO2005004I1 (no) | 1993-11-24 | 2005-02-09 | Duloksetin og dets farmasøytisk akseptable syreaddisjonssalter, spesielt duloksetin hydroklorid |
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| EP (1) | EP0654264B1 (ru) |
| JP (1) | JP3681009B2 (ru) |
| KR (1) | KR100347277B1 (ru) |
| CN (1) | CN1099284C (ru) |
| AT (1) | ATE201594T1 (ru) |
| AU (1) | AU679269B2 (ru) |
| CA (1) | CA2136120C (ru) |
| CY (2) | CY2245B1 (ru) |
| CZ (1) | CZ289069B6 (ru) |
| DE (2) | DE122005000005I2 (ru) |
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| HK (1) | HK1013799A1 (ru) |
| HU (1) | HU218920B (ru) |
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| PH (1) | PH30741A (ru) |
| PT (1) | PT654264E (ru) |
| RU (1) | RU2152786C2 (ru) |
| SI (1) | SI0654264T1 (ru) |
| TW (1) | TW344661B (ru) |
| UA (1) | UA32429C2 (ru) |
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Families Citing this family (44)
| Publication number | Priority date | Publication date | Assignee | Title |
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| US5506270A (en) * | 1995-01-30 | 1996-04-09 | American Home Products Corporation | Venlafaxine in the treatment of hypothalamic amenorrhea in non-depressed women |
| HUP9902884A3 (en) * | 1996-03-11 | 2000-12-28 | Lilly Co Eli | Use of duloxetine for treating or preventing interstitial cystitis |
| EP1331003B1 (en) * | 1996-03-25 | 2015-08-26 | Wyeth LLC | Extended release formulation containing venlafaxine |
| US6274171B1 (en) | 1996-03-25 | 2001-08-14 | American Home Products Corporation | Extended release formulation of venlafaxine hydrochloride |
| PE57198A1 (es) * | 1996-03-25 | 1998-10-10 | American Home Prod | Formula de liberacion prolongada |
| US6150396A (en) * | 1997-03-07 | 2000-11-21 | Eli Lilly And Company | Methods of treating or preventing interstitial cystitis |
| WO2000003701A1 (en) * | 1998-07-16 | 2000-01-27 | Massachusetts Institute Of Technology | Composition for treatment of stress |
| US6579899B1 (en) | 1998-07-16 | 2003-06-17 | Massachusetts Institute Of Technology | Composition for treatment of stress |
| PT1039882E (pt) * | 1998-08-27 | 2011-01-03 | Pfizer Health Ab | Formulação terapêutica para administrar tolterodina com libertação controlada |
| US6046242A (en) * | 1998-11-27 | 2000-04-04 | Basf Aktiengesellschaft | Use of aryl-substituted cyclobutylalkylamines for treating urinary incontinence |
| US6342533B1 (en) | 1998-12-01 | 2002-01-29 | Sepracor, Inc. | Derivatives of (−)-venlafaxine and methods of preparing and using the same |
| US6197828B1 (en) | 1998-12-01 | 2001-03-06 | Sepracor, Inc. | Derivatives of (+)-venlafaxine and methods of preparing and using the same |
| CA2368083A1 (en) * | 1999-04-06 | 2000-10-12 | Sepracor Inc. | Derivatives of venlafaxine and methods of preparing and using the same |
| PT1632234E (pt) * | 1999-07-01 | 2007-07-09 | Pharmacia & Upjohn Co Llc | (s,s)-reboxetina para o tratamento da síndrome de fadiga crónica |
| US7291646B2 (en) | 1999-11-24 | 2007-11-06 | Wyeth | Ethers of O-desmethyl venlafaxine |
| US6572890B2 (en) * | 2000-01-13 | 2003-06-03 | Osmotica Corp. | Osmotic device containing venlafaxine and an anti-psychotic agent |
| DE10027290C2 (de) | 2000-06-02 | 2002-07-11 | Basf Coatings Ag | Pulverklarlackdispersionen (Pulverslurry-Klarlacke) und ihre Verwendung |
| DE10059412A1 (de) | 2000-11-30 | 2002-06-13 | Gruenenthal Gmbh | Verwendung von 1-Phenyl-3-dimethylamino-propanverbindungen zur Therapie der Harninkontinenz |
| DK1360169T3 (da) | 2001-02-12 | 2007-11-26 | Wyeth Corp | Succinatsalt af O-desmethyl-venlafaxin |
| US6602911B2 (en) * | 2001-11-05 | 2003-08-05 | Cypress Bioscience, Inc. | Methods of treating fibromyalgia |
| UA77234C2 (en) * | 2001-12-05 | 2006-11-15 | Wyeth Corp | Monohydrate of venlafaxine hydrochloride and methods for its preparation (variants) |
| EP1451145A1 (en) * | 2001-12-05 | 2004-09-01 | Wyeth | Novel crystalline polymorph of venlafaxine hydrochloride and methods for the preparation thereof |
| GB0202265D0 (en) * | 2002-01-31 | 2002-03-20 | Arachnova Therapeutics Ltd | New therapeutic use |
| US6696496B2 (en) * | 2002-03-28 | 2004-02-24 | Synthon Bv | Low water-soluble venlafaxine salts |
| EP1499309A4 (en) * | 2002-04-24 | 2008-05-28 | Cypress Bioscience Inc | PREVENTION AND TREATMENT OF FUNCTIONAL SOMATIC DISEASES, INCLUDING STRESS-BASED DISEASES |
| DE10224107A1 (de) * | 2002-05-29 | 2003-12-11 | Gruenenthal Gmbh | Kombination ausgewählter Opioide mit anderen Wirkstoffen zur Therapie der Harninkontinenz |
| WO2004019892A2 (en) * | 2002-08-30 | 2004-03-11 | Watson Pharmaceuticals, Inc. | Drug delivery system for treating urinary incontinence |
| GB0221438D0 (en) * | 2002-09-16 | 2002-10-23 | Avecia Ltd | Processes and compounds |
| EP1424079A1 (en) * | 2002-11-27 | 2004-06-02 | Boehringer Ingelheim International GmbH | Combination of a beta-3-receptor agonist and of a reuptake inhibitor of serotonin and/or norepinephrine |
| US20070077301A1 (en) * | 2002-12-23 | 2007-04-05 | Meyer Glenn A | Venlafaxine osmotic device formulation |
| DE602004007225T2 (de) * | 2003-04-04 | 2008-03-06 | Dynogen Pharmaceuticals Inc., Waltham | Methode zur behandlung von erkrankungen der unteren harnwege |
| BRPI0510453A (pt) * | 2004-04-30 | 2007-10-30 | Warner Lambert Co | composto substituìdos com morfolina para o tratamento de distúrbios do sistema nervoso central |
| EP2248524A3 (en) | 2004-08-25 | 2011-03-09 | Takeda Pharmaceutical Company Limited | Preventives/remedies for stress urinary incontinence and method of screening the same |
| WO2006071868A2 (en) * | 2004-12-23 | 2006-07-06 | Teva Pharmaceutical Industries Ltd. | Process for preparing pharmaceutically acceptable salts of duloxetine and intermediates thereof |
| TW200639162A (en) | 2005-03-14 | 2006-11-16 | Teva Pharma | Pure duloxetine hydrochloride |
| WO2007038253A2 (en) | 2005-09-22 | 2007-04-05 | Teva Pharmaceutical Industries Ltd. | Dnt-maleate and methods of preparation thereof |
| US7994220B2 (en) * | 2005-09-28 | 2011-08-09 | Cypress Bioscience, Inc. | Milnacipran for the long-term treatment of fibromyalgia syndrome |
| DK1954669T3 (en) | 2005-12-01 | 2015-10-12 | Auspex Pharmaceuticals Inc | SUBSTITUTED phenethylamines a serotonergic AND / OR NOREPINEPHRINERG ACTIVITY |
| EP1957470A1 (en) | 2005-12-05 | 2008-08-20 | Wyeth | Process for selective synthesis of enantiomers of substituted 1-(2-amino-1-phenyl-ethyl)-cyclohexanols |
| WO2007067581A1 (en) * | 2005-12-05 | 2007-06-14 | Teva Pharmaceutical Industries Ltd. | 2-(n-methyl-propanamine)-3-(2-naphthol) thiophene, an impurity of duloxetine hydrochloride |
| EP1826204A1 (en) | 2006-02-28 | 2007-08-29 | Laboratorios Del Dr. Esteve, S.A. | Process for obtaining enantiomers of duloxetine precursors |
| US20080081067A1 (en) * | 2006-10-03 | 2008-04-03 | Gupta Manishkumar | Sustained release pharmaceutical compositions of venlafaxine and process for preparation thereof |
| EP3269706A1 (en) | 2007-03-15 | 2018-01-17 | Auspex Pharmaceuticals, Inc. | Deuterated o-desmethylvenlafaxine with serotoninergic and/or norepinephrinergic activity |
| CA3104701A1 (en) | 2018-07-11 | 2020-01-16 | Dignify Therapeutics, Llc | Method of treating voiding dysfunction |
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| US4314081A (en) * | 1974-01-10 | 1982-02-02 | Eli Lilly And Company | Arloxyphenylpropylamines |
| US4018895A (en) * | 1974-01-10 | 1977-04-19 | Eli Lilly And Company | Aryloxyphenylpropylamines in treating depression |
| GR75395B (ru) * | 1980-11-14 | 1984-07-13 | Lilly Co Eli | |
| IE56324B1 (en) * | 1982-12-13 | 1991-06-19 | American Home Prod | Phenethylamine derivatives and intermediates therefor |
| US4761501A (en) * | 1983-10-26 | 1988-08-02 | American Home Products Corporation | Substituted phenylacetamides |
| KR880007433A (ko) * | 1986-12-22 | 1988-08-27 | 메리 앤 터커 | 3-아릴옥시-3-치환된 프로판아민 |
| US4956388A (en) * | 1986-12-22 | 1990-09-11 | Eli Lilly And Company | 3-aryloxy-3-substituted propanamines |
| CA1329937C (en) * | 1987-04-09 | 1994-05-31 | Dennis Charles Thompson | 1-phenyl-3-naphthalenyloxypropanamines |
| SE8804003D0 (sv) * | 1988-11-04 | 1988-11-04 | Pharmacia Ab | Compounds for the treatment of urinary incontinence |
| US5250571A (en) * | 1988-11-14 | 1993-10-05 | Eli Lilly And Company | (S)-norfluoxetine in method of inhibiting serotonin uptake |
| PH30083A (en) * | 1991-02-25 | 1996-12-27 | Lilly Co Eli | Treatment of lower urinary tract disorders |
| EP0537915B1 (en) * | 1991-09-27 | 1995-07-12 | Eli Lilly And Company | N-alkyl-3-phenyl-3-(2-alkylthiophenoxy)propylamines as norepinephrine inhibitors |
| US5281624A (en) * | 1991-09-27 | 1994-01-25 | Eli Lilly And Company | N-alkyl-3-phenyl-3-(2-substituted phenoxy) propylamines and pharmaceutical use thereof |
| US5192751A (en) * | 1992-07-24 | 1993-03-09 | Eli Lilly And Company | Use of competitive NMDA receptor antagonists in the treatment of urinary incontinence |
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- 1994-11-18 CA CA002136120A patent/CA2136120C/en not_active Expired - Lifetime
- 1994-11-21 UA UA94119056A patent/UA32429C2/ru unknown
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