NO308508B1 - Anvendelse av levobupivacaine i enantiomert overskudd - Google Patents

Anvendelse av levobupivacaine i enantiomert overskudd

Info

Publication number
NO308508B1
NO308508B1 NO961479A NO961479A NO308508B1 NO 308508 B1 NO308508 B1 NO 308508B1 NO 961479 A NO961479 A NO 961479A NO 961479 A NO961479 A NO 961479A NO 308508 B1 NO308508 B1 NO 308508B1
Authority
NO
Norway
Prior art keywords
levobupivacaine
enantiomeric excess
enantiomeric
excess
anaesthetic
Prior art date
Application number
NO961479A
Other languages
English (en)
Norwegian (no)
Other versions
NO961479L (no
NO961479D0 (no
Inventor
Hazel Judith Bardsley
Robert William Gristwood
Original Assignee
Darwin Discovery Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26303667&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO308508(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GB939321061A external-priority patent/GB9321061D0/en
Priority claimed from GB9408014A external-priority patent/GB9408014D0/en
Application filed by Darwin Discovery Ltd filed Critical Darwin Discovery Ltd
Publication of NO961479D0 publication Critical patent/NO961479D0/no
Publication of NO961479L publication Critical patent/NO961479L/no
Publication of NO308508B1 publication Critical patent/NO308508B1/no

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P23/00Anaesthetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Neurosurgery (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Hydrogenated Pyridines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
NO961479A 1993-10-13 1996-04-12 Anvendelse av levobupivacaine i enantiomert overskudd NO308508B1 (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB939321061A GB9321061D0 (en) 1993-10-13 1993-10-13 Analgestic agent and its use
GB9408014A GB9408014D0 (en) 1994-04-22 1994-04-22 Analgesic agent and its use
PCT/GB1994/002249 WO1995010277A1 (en) 1993-10-13 1994-10-13 Analgesic agent and its use

Publications (3)

Publication Number Publication Date
NO961479D0 NO961479D0 (no) 1996-04-12
NO961479L NO961479L (no) 1996-06-11
NO308508B1 true NO308508B1 (no) 2000-09-25

Family

ID=26303667

Family Applications (1)

Application Number Title Priority Date Filing Date
NO961479A NO308508B1 (no) 1993-10-13 1996-04-12 Anvendelse av levobupivacaine i enantiomert overskudd

Country Status (15)

Country Link
US (1) US5708011A (de)
EP (2) EP0723445B1 (de)
JP (2) JPH09503778A (de)
KR (1) KR100365979B1 (de)
CN (1) CN1074920C (de)
AT (2) ATE210982T1 (de)
AU (1) AU694453B2 (de)
DE (2) DE69402330T2 (de)
DK (2) DK0723445T3 (de)
ES (2) ES2101578T3 (de)
GR (1) GR3023289T3 (de)
HK (1) HK1006420A1 (de)
NO (1) NO308508B1 (de)
PT (1) PT727210E (de)
WO (1) WO1995010277A1 (de)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9507677D0 (en) * 1995-04-13 1995-05-31 Chiroscience Ltd Pharmaceutical formulation and dose
GB9321061D0 (en) * 1993-10-13 1993-12-01 Chiroscience Ltd Analgestic agent and its use
MX9707875A (es) * 1995-04-13 1997-11-29 Darwin Discovery Ltd Levobupivacaina y su uso como un anestesico en mujeres embarazadas.
GB9704352D0 (en) * 1997-03-03 1997-04-23 Chiroscience Ltd Levobupivacaine and its use
GB9704351D0 (en) * 1997-03-03 1997-04-23 Chiroscience Ltd Levobupivacaine and its use
GB9704370D0 (en) * 1997-03-03 1997-04-23 Chiroscience Ltd Levobupivacaine and its use
WO1999004771A2 (en) * 1997-07-21 1999-02-04 Darwin Discovery Limited Use of levobupivacaine
CA2294921C (en) * 1997-07-22 2009-04-07 Darwin Discovery Limited Levobupivacaine and its use
ES2343767T3 (es) 1997-09-18 2010-08-09 Pacira Pharmaceuticals, Inc. Composiciones anestesicas liposomicas de liberacion sostenida.
JP4575592B2 (ja) * 1997-11-14 2010-11-04 パシラ ファーマシューティカルズ インコーポレーテッド 多小胞リポソームの製造
HU228143B1 (en) * 1997-11-19 2012-12-28 Darwin Discovery Ltd Anaesthetic formulation
JP2002520120A (ja) 1998-07-17 2002-07-09 スカイファーマ インコーポレーテッド 封入物質の制御放出のための生分解性組成物
BR0002246A (pt) * 2000-04-06 2003-04-15 Cristalia Prod Quimicos Farm Processo de obtenção dos enantiÈmeros da bupivacaìna racêmica, processo de obtenção de composições farmacêuticas a base de levobupivacaìna: composições farmacêuticas a base de levobupivacaìna formuladas nas formas básicas ou sais farmaceuticamente aceitáveis e utilização das composições farmacêuticas a base de levobupivacaìna formuladas nas formas básicas ou sais farmaceuticamente aceitáveis
WO2002096368A2 (en) * 2001-05-31 2002-12-05 Skyepharma Inc. Encapsulation of nanosuspensions in liposomes and microspheres
MXPA04004665A (es) * 2001-11-14 2004-09-10 Alza Corp Composiciones de deposito inyectable y uso de los mismos.
ATE507816T1 (de) * 2001-11-14 2011-05-15 Durect Corp Injizierbare depotzusammensetzungen und deren verwendung
US20070196415A1 (en) * 2002-11-14 2007-08-23 Guohua Chen Depot compositions with multiple drug release rate controls and uses thereof
US20040001889A1 (en) 2002-06-25 2004-01-01 Guohua Chen Short duration depot formulations
ES2321505T3 (es) * 2002-07-31 2009-06-08 Alza Corporation Composiciones de deposito de polimero multimodal inyectables y empleo de las mismas.
ATE392886T1 (de) * 2002-07-31 2008-05-15 Alza Corp Injizierbare depotzusammensetzungen und deren verwendung
US20060142234A1 (en) * 2004-12-23 2006-06-29 Guohua Chen Injectable non-aqueous suspension
WO2010065930A1 (en) * 2008-12-04 2010-06-10 The Board Of Trustees Of The Leland Stanford Junior University Methods and compositions for treating or preventing narcotic withdrawal symptoms
EP3079668A1 (de) 2013-12-09 2016-10-19 Durect Corporation Pharmazeutisch aktive wirkstoffkomplexe, polymerkomplexe und zusammensetzungen und verfahren damit
CN106214670B (zh) * 2016-07-25 2020-12-29 上海璃道医药科技有限公司 酰胺类药物的用途
JP2023515918A (ja) 2020-01-13 2023-04-17 デュレクト コーポレーション 不純物が低減された徐放性薬物送達システム及び関連の方法
US11357727B1 (en) 2021-01-22 2022-06-14 Pacira Pharmaceuticals, Inc. Manufacturing of bupivacaine multivesicular liposomes
US11033495B1 (en) 2021-01-22 2021-06-15 Pacira Pharmaceuticals, Inc. Manufacturing of bupivacaine multivesicular liposomes
US11278494B1 (en) 2021-01-22 2022-03-22 Pacira Pharmaceuticals, Inc. Manufacturing of bupivacaine multivesicular liposomes

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4695576A (en) * 1984-07-09 1987-09-22 Astra Lake Medel Aktiebolag L-N-n-propylpipecolic acid-2,6-xylidide
MX9707875A (es) * 1995-04-13 1997-11-29 Darwin Discovery Ltd Levobupivacaina y su uso como un anestesico en mujeres embarazadas.

Also Published As

Publication number Publication date
NO961479L (no) 1996-06-11
CN1133010A (zh) 1996-10-09
ES2101578T3 (es) 1997-07-01
DK0723445T3 (da) 1997-10-06
EP0723445B1 (de) 1997-03-26
HK1006420A1 (en) 1999-02-26
US5708011A (en) 1998-01-13
DE69402330D1 (de) 1997-04-30
DE69429536T2 (de) 2002-06-20
PT727210E (pt) 2002-06-28
DE69402330T2 (de) 1997-07-03
NO961479D0 (no) 1996-04-12
GR3023289T3 (en) 1997-07-30
DE69429536D1 (de) 2002-01-31
EP0727210A3 (de) 1998-03-04
ES2170179T3 (es) 2002-08-01
EP0727210B1 (de) 2001-12-19
DK0727210T3 (da) 2002-04-15
AU7859494A (en) 1995-05-04
CN1074920C (zh) 2001-11-21
JPH09503778A (ja) 1997-04-15
EP0727210A2 (de) 1996-08-21
ATE210982T1 (de) 2002-01-15
KR100365979B1 (ko) 2003-07-22
WO1995010277A1 (en) 1995-04-20
ATE150643T1 (de) 1997-04-15
AU694453B2 (en) 1998-07-23
EP0723445A1 (de) 1996-07-31
JP2006213736A (ja) 2006-08-17

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