NO304740B1 - 10-desacetoksytaxolderivater - Google Patents
10-desacetoksytaxolderivaterInfo
- Publication number
- NO304740B1 NO304740B1 NO934469A NO941021A NO304740B1 NO 304740 B1 NO304740 B1 NO 304740B1 NO 934469 A NO934469 A NO 934469A NO 941021 A NO941021 A NO 941021A NO 304740 B1 NO304740 B1 NO 304740B1
- Authority
- NO
- Norway
- Prior art keywords
- opt
- aryl
- protected
- alkyl
- desacetoksytaxolderivater
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
- C07D407/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
- C07D407/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
- C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/003—Compounds containing elements of Groups 4 or 14 of the Periodic Table without C-Metal linkages
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
- C07F7/1804—Compounds having Si-O-C linkages
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Epoxy Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
- Saccharide Compounds (AREA)
- Signal Processing For Digital Recording And Reproducing (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Water Treatment By Electricity Or Magnetism (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Polysaccharides And Polysaccharide Derivatives (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US76380591A | 1991-09-23 | 1991-09-23 | |
| US90040892A | 1992-06-18 | 1992-06-18 | |
| PCT/US1992/007935 WO1993006093A1 (en) | 1991-09-23 | 1992-09-22 | 10-desacetoxytaxol derivatives |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO941021D0 NO941021D0 (no) | 1994-03-22 |
| NO941021L NO941021L (no) | 1994-05-20 |
| NO304740B1 true NO304740B1 (no) | 1999-02-08 |
Family
ID=27117344
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO934469A NO304740B1 (no) | 1991-09-23 | 1994-03-22 | 10-desacetoksytaxolderivater |
Country Status (15)
| Country | Link |
|---|---|
| EP (1) | EP0642503B1 (cs) |
| JP (1) | JP3304088B2 (cs) |
| KR (1) | KR100239201B1 (cs) |
| AT (1) | ATE187170T1 (cs) |
| AU (1) | AU663732B2 (cs) |
| CA (1) | CA2119363C (cs) |
| CZ (1) | CZ287609B6 (cs) |
| DE (1) | DE69230379T2 (cs) |
| DK (1) | DK0642503T3 (cs) |
| ES (1) | ES2141727T3 (cs) |
| FI (1) | FI112479B (cs) |
| HU (1) | HU225474B1 (cs) |
| NO (1) | NO304740B1 (cs) |
| UA (1) | UA39860C2 (cs) |
| WO (1) | WO1993006093A1 (cs) |
Families Citing this family (28)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5998656A (en) | 1991-09-23 | 1999-12-07 | Florida State University | C10 tricyclic taxanes |
| US5294637A (en) * | 1992-07-01 | 1994-03-15 | Bristol-Myers Squibb Company | Fluoro taxols |
| NZ248017A (en) * | 1992-07-01 | 1994-12-22 | Bristol Myers Squibb Co | 7-fluoro-taxol derivatives, precursors and pharmaceutical compositions thereof |
| US5681714A (en) * | 1992-07-30 | 1997-10-28 | Mount Sinai Hospital Corporation | Nucleic acid encoding tek receptor tyrosine kinase |
| EP0582469A2 (en) * | 1992-08-06 | 1994-02-09 | Wisconsin Alumni Research Foundation | Process for preparing taxol-type compound from beta-lactam precursors |
| CA2100808A1 (en) * | 1992-10-01 | 1994-04-02 | Vittorio Farina | Deoxy paclitaxels |
| US5380751A (en) * | 1992-12-04 | 1995-01-10 | Bristol-Myers Squibb Company | 6,7-modified paclitaxels |
| US5646176A (en) * | 1992-12-24 | 1997-07-08 | Bristol-Myers Squibb Company | Phosphonooxymethyl ethers of taxane derivatives |
| IL108443A0 (en) * | 1993-01-29 | 1994-04-12 | Univ Florida State | C7 taxane derivatives and pharmaceutical compositions containing them |
| ZA94128B (en) * | 1993-02-01 | 1994-08-19 | Univ New York State Res Found | Process for the preparation of taxane derivatives and betalactam intermediates therefor |
| US5703247A (en) * | 1993-03-11 | 1997-12-30 | Virginia Tech Intellectual Properties, Inc. | 2-Debenzoyl-2-acyl taxol derivatives and methods for making same |
| DE69432141T2 (de) * | 1993-03-22 | 2003-07-31 | Florida State University, Tallahassee | Taxane mit furyl-oder thienyl substituierten seitenketten |
| NZ511762A (en) | 1993-07-19 | 2003-09-26 | Univ British Columbia | Anti-angiogenic compositions and methods of use |
| FR2711369B1 (fr) * | 1993-10-20 | 1995-11-17 | Rhone Poulenc Rorer Sa | Nouveaux taxoïdes, leur préparation et les compositions qui les contiennent. |
| FR2721024B1 (fr) * | 1994-06-09 | 1996-07-12 | Rhone Poulenc Rorer Sa | Nouveaux taxoïdes, leur préparation et les compositions pharmaceutiques qui les contiennent. |
| CA2192373A1 (en) * | 1994-06-09 | 1995-12-14 | Hirofumi Terasawa | Deacetoxytaxol derivative |
| FR2723094A1 (fr) * | 1994-07-26 | 1996-02-02 | Rhone Poulenc Rorer Sa | Nouveaux taxoides, leur preparation et les compositions pharmaceutiques qui les contiennent |
| US5840929A (en) * | 1995-04-14 | 1998-11-24 | Bristol-Myers Squibb Company | C4 methoxy ether derivatives of paclitaxel |
| AU728057B2 (en) * | 1995-09-13 | 2001-01-04 | Florida State University | Radiosensitizing taxanes and their pharmaceutical preparations |
| DE19621311A1 (de) | 1996-05-28 | 1997-12-04 | Bayer Ag | Substituierte Phenyluracile |
| US5635531A (en) * | 1996-07-08 | 1997-06-03 | Bristol-Myers Squibb Company | 3'-aminocarbonyloxy paclitaxels |
| US5773464A (en) * | 1996-09-30 | 1998-06-30 | Bristol-Myers Squibb Company | C-10 epoxy taxanes |
| US5977386A (en) * | 1996-12-24 | 1999-11-02 | Bristol-Myers Squibb Company | 6-thio-substituted paclitaxels |
| US5902822A (en) * | 1997-02-28 | 1999-05-11 | Bristol-Myers Squibb Company | 7-methylthiooxomethyl and 7-methylthiodioxomethyl paclitaxels |
| US5912264A (en) * | 1997-03-03 | 1999-06-15 | Bristol-Myers Squibb Company | 6-halo-or nitrate-substituted paclitaxels |
| US6017935A (en) * | 1997-04-24 | 2000-01-25 | Bristol-Myers Squibb Company | 7-sulfur substituted paclitaxels |
| KR101096282B1 (ko) * | 2009-04-24 | 2011-12-20 | 주식회사 삼양제넥스 | 탁산 유도체를 제조하는 방법 |
| CN108158991A (zh) | 2012-07-19 | 2018-06-15 | 富士胶片株式会社 | 含紫杉烷系活性成分的液体组合物、其制造方法及液体制剂 |
-
1992
- 1992-09-22 HU HU9400832A patent/HU225474B1/hu unknown
- 1992-09-22 KR KR1019940700948A patent/KR100239201B1/ko not_active Expired - Fee Related
- 1992-09-22 ES ES92920702T patent/ES2141727T3/es not_active Expired - Lifetime
- 1992-09-22 CA CA002119363A patent/CA2119363C/en not_active Expired - Fee Related
- 1992-09-22 AT AT92920702T patent/ATE187170T1/de not_active IP Right Cessation
- 1992-09-22 DK DK92920702T patent/DK0642503T3/da active
- 1992-09-22 JP JP50626993A patent/JP3304088B2/ja not_active Expired - Fee Related
- 1992-09-22 EP EP92920702A patent/EP0642503B1/en not_active Expired - Lifetime
- 1992-09-22 WO PCT/US1992/007935 patent/WO1993006093A1/en not_active Ceased
- 1992-09-22 CZ CZ1994661A patent/CZ287609B6/cs not_active IP Right Cessation
- 1992-09-22 DE DE69230379T patent/DE69230379T2/de not_active Expired - Fee Related
- 1992-09-22 UA UA94005360A patent/UA39860C2/uk unknown
- 1992-09-22 AU AU26926/92A patent/AU663732B2/en not_active Ceased
-
1994
- 1994-03-22 FI FI941324A patent/FI112479B/fi not_active IP Right Cessation
- 1994-03-22 NO NO934469A patent/NO304740B1/no unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP0642503A1 (en) | 1995-03-15 |
| HUT68422A (en) | 1995-04-26 |
| HU9400832D0 (en) | 1994-06-28 |
| WO1993006093A1 (en) | 1993-04-01 |
| KR100239201B1 (ko) | 2000-02-01 |
| EP0642503B1 (en) | 1999-12-01 |
| CA2119363C (en) | 2001-07-17 |
| EP0642503A4 (en) | 1994-07-07 |
| AU2692692A (en) | 1993-04-27 |
| CZ287609B6 (cs) | 2001-01-17 |
| FI941324L (fi) | 1994-03-22 |
| DE69230379D1 (de) | 2000-01-05 |
| HU225474B1 (en) | 2006-12-28 |
| DK0642503T3 (da) | 2000-05-22 |
| ES2141727T3 (es) | 2000-04-01 |
| CA2119363A1 (en) | 1993-04-01 |
| UA39860C2 (uk) | 2001-07-16 |
| CZ66194A3 (en) | 1995-07-12 |
| DE69230379T2 (de) | 2000-05-25 |
| FI941324A0 (fi) | 1994-03-22 |
| ATE187170T1 (de) | 1999-12-15 |
| FI112479B (fi) | 2003-12-15 |
| AU663732B2 (en) | 1995-10-19 |
| NO941021L (no) | 1994-05-20 |
| NO941021D0 (no) | 1994-03-22 |
| JPH07502981A (ja) | 1995-03-30 |
| JP3304088B2 (ja) | 2002-07-22 |
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