NO20092342L - Azaspiroderivativater - Google Patents
AzaspiroderivativaterInfo
- Publication number
- NO20092342L NO20092342L NO20092342A NO20092342A NO20092342L NO 20092342 L NO20092342 L NO 20092342L NO 20092342 A NO20092342 A NO 20092342A NO 20092342 A NO20092342 A NO 20092342A NO 20092342 L NO20092342 L NO 20092342L
- Authority
- NO
- Norway
- Prior art keywords
- present
- relates
- compounds
- azaspiroderivativater
- azaspiropiperidine
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
- C07D491/20—Spiro-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/438—The ring being spiro-condensed with carbocyclic or heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biomedical Technology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Urology & Nephrology (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Vascular Medicine (AREA)
- Gastroenterology & Hepatology (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP06127334 | 2006-12-29 | ||
PCT/EP2007/064183 WO2008080844A1 (fr) | 2006-12-29 | 2007-12-19 | Dérivés azaspiro |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20092342L true NO20092342L (no) | 2009-07-02 |
Family
ID=39201403
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20092342A NO20092342L (no) | 2006-12-29 | 2009-06-18 | Azaspiroderivativater |
Country Status (22)
Country | Link |
---|---|
US (3) | US8044202B2 (fr) |
EP (1) | EP2125827B1 (fr) |
JP (1) | JP2010514727A (fr) |
KR (1) | KR101129861B1 (fr) |
CN (1) | CN101589046B (fr) |
AR (1) | AR064547A1 (fr) |
AT (1) | ATE486877T1 (fr) |
AU (1) | AU2007341379B2 (fr) |
BR (1) | BRPI0720827A2 (fr) |
CA (1) | CA2674154A1 (fr) |
CL (1) | CL2007003832A1 (fr) |
DE (1) | DE602007010359D1 (fr) |
DK (1) | DK2125827T3 (fr) |
ES (1) | ES2351949T3 (fr) |
MX (1) | MX2009006921A (fr) |
NO (1) | NO20092342L (fr) |
PE (1) | PE20081844A1 (fr) |
PL (1) | PL2125827T3 (fr) |
PT (1) | PT2125827E (fr) |
RU (1) | RU2009124419A (fr) |
TW (1) | TW200835483A (fr) |
WO (1) | WO2008080844A1 (fr) |
Families Citing this family (20)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
RU2009119394A (ru) * | 2006-12-07 | 2011-01-20 | Ф. Хоффманн-Ля Рош Аг (Ch) | Производные спиро-пиперидина в качестве антагонистов рецептора v1a |
CA2673307A1 (fr) * | 2006-12-22 | 2008-07-03 | F. Hoffman-La Roche Ag | Derives de spiropiperidine |
ME01838B (me) | 2009-06-29 | 2014-12-20 | Lncyte Holdings Corp | Pirimidinoni kao inhibitori pi3k |
AR078948A1 (es) * | 2009-11-30 | 2011-12-14 | Lilly Co Eli | Compuestos de espiropiperidina, composicion farmaceutica que lo comprenden y su uso para preparar un medicamento util para tratar la diabetes |
WO2011075643A1 (fr) * | 2009-12-18 | 2011-06-23 | Incyte Corporation | Dérivés condensés d'hétéroaryles substitués à titre d'inhibiteurs de pi3k |
WO2011075630A1 (fr) * | 2009-12-18 | 2011-06-23 | Incyte Corporation | Dérivés substitués d'aryles et d'hétéroaryles fusionnés au titre d'inhibiteurs de pi3k |
AR081823A1 (es) | 2010-04-14 | 2012-10-24 | Incyte Corp | DERIVADOS FUSIONADOS COMO INHIBIDORES DE PI3Kd |
US9062055B2 (en) | 2010-06-21 | 2015-06-23 | Incyte Corporation | Fused pyrrole derivatives as PI3K inhibitors |
AR084366A1 (es) | 2010-12-20 | 2013-05-08 | Incyte Corp | N-(1-(fenil sustituido)etil)-9h-purin-6-aminas como inhibidores de pi3k |
US9108984B2 (en) | 2011-03-14 | 2015-08-18 | Incyte Corporation | Substituted diamino-pyrimidine and diamino-pyridine derivatives as PI3K inhibitors |
US9126948B2 (en) | 2011-03-25 | 2015-09-08 | Incyte Holdings Corporation | Pyrimidine-4,6-diamine derivatives as PI3K inhibitors |
ES2464598T3 (es) | 2011-07-22 | 2014-06-03 | Université Joseph Fourier | Nuevos derivados bis-indólicos, procedimiento para su preparación, y sus utilizaciones como fármaco |
EA033646B1 (ru) | 2011-09-02 | 2019-11-13 | Incyte Holdings Corp | Гетероциклиламины как ингибиторы pi3k |
CN102568615B (zh) * | 2011-12-13 | 2013-05-22 | 华中科技大学 | 一种小型精密调平装置 |
AR090548A1 (es) | 2012-04-02 | 2014-11-19 | Incyte Corp | Azaheterociclobencilaminas biciclicas como inhibidores de pi3k |
WO2015191677A1 (fr) | 2014-06-11 | 2015-12-17 | Incyte Corporation | Dérivés d'hétéroarylaminoalkylphényle bicycliques à titre d'inhibiteurs de pi3k |
WO2016138363A1 (fr) | 2015-02-27 | 2016-09-01 | Incyte Corporation | Sels d'un inhibiteur de pi3k et procédés de préparation de ces sels |
US9732097B2 (en) | 2015-05-11 | 2017-08-15 | Incyte Corporation | Process for the synthesis of a phosphoinositide 3-kinase inhibitor |
US9988401B2 (en) | 2015-05-11 | 2018-06-05 | Incyte Corporation | Crystalline forms of a PI3K inhibitor |
AR120324A1 (es) | 2019-10-29 | 2022-02-09 | Biogen Ma Inc | Inhibidores de o-glucoproteína-2-acetamido-2-deoxi-3-d-glucopiranosidasa espirocíclica |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2761992B1 (fr) * | 1997-04-09 | 1999-06-11 | Hoechst Marion Roussel Inc | Nouveaux steroides 4-halogenes, leur procede et intermediaires de preparation, leur application comme medicaments et les compositions pharmaceutiques les renfermant |
TWI279402B (en) | 1999-08-20 | 2007-04-21 | Banyu Pharma Co Ltd | Spiro compounds having NPY antagonistic activities and agents containing the same |
GB0003397D0 (en) | 2000-02-14 | 2000-04-05 | Merck Sharp & Dohme | Therapeutic agents |
EP1701959A1 (fr) * | 2003-12-22 | 2006-09-20 | Pfizer Limited | Dérivés de triazole comme antagonistes de vasopréssine |
GB0400700D0 (en) * | 2004-01-13 | 2004-02-18 | Pfizer Ltd | Compounds useful in therapy |
GB0504556D0 (en) * | 2005-03-04 | 2005-04-13 | Pfizer Ltd | Novel pharmaceuticals |
-
2007
- 2007-12-19 CN CN2007800479989A patent/CN101589046B/zh not_active Expired - Fee Related
- 2007-12-19 ES ES07857806T patent/ES2351949T3/es active Active
- 2007-12-19 AT AT07857806T patent/ATE486877T1/de active
- 2007-12-19 BR BRPI0720827-8A patent/BRPI0720827A2/pt not_active IP Right Cessation
- 2007-12-19 MX MX2009006921A patent/MX2009006921A/es active IP Right Grant
- 2007-12-19 DE DE602007010359T patent/DE602007010359D1/de active Active
- 2007-12-19 KR KR1020097015840A patent/KR101129861B1/ko not_active IP Right Cessation
- 2007-12-19 AU AU2007341379A patent/AU2007341379B2/en not_active Expired - Fee Related
- 2007-12-19 PL PL07857806T patent/PL2125827T3/pl unknown
- 2007-12-19 EP EP07857806A patent/EP2125827B1/fr not_active Not-in-force
- 2007-12-19 JP JP2009543443A patent/JP2010514727A/ja active Pending
- 2007-12-19 CA CA002674154A patent/CA2674154A1/fr not_active Abandoned
- 2007-12-19 PT PT07857806T patent/PT2125827E/pt unknown
- 2007-12-19 WO PCT/EP2007/064183 patent/WO2008080844A1/fr active Application Filing
- 2007-12-19 DK DK07857806.9T patent/DK2125827T3/da active
- 2007-12-19 RU RU2009124419/04A patent/RU2009124419A/ru not_active Application Discontinuation
- 2007-12-20 US US11/960,799 patent/US8044202B2/en not_active Expired - Fee Related
- 2007-12-20 US US11/960,823 patent/US8039624B2/en not_active Expired - Fee Related
- 2007-12-20 US US11/960,779 patent/US8034937B2/en not_active Expired - Fee Related
- 2007-12-26 TW TW096150410A patent/TW200835483A/zh unknown
- 2007-12-27 CL CL200703832A patent/CL2007003832A1/es unknown
- 2007-12-27 AR ARP070105915A patent/AR064547A1/es not_active Application Discontinuation
-
2008
- 2008-01-02 PE PE2008000047A patent/PE20081844A1/es not_active Application Discontinuation
-
2009
- 2009-06-18 NO NO20092342A patent/NO20092342L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
EP2125827A1 (fr) | 2009-12-02 |
US8034937B2 (en) | 2011-10-11 |
ES2351949T3 (es) | 2011-02-14 |
WO2008080844A1 (fr) | 2008-07-10 |
PT2125827E (pt) | 2010-11-22 |
JP2010514727A (ja) | 2010-05-06 |
RU2009124419A (ru) | 2011-02-10 |
US8039624B2 (en) | 2011-10-18 |
AU2007341379B2 (en) | 2012-05-24 |
AU2007341379A1 (en) | 2008-07-10 |
CN101589046A (zh) | 2009-11-25 |
WO2008080844A9 (fr) | 2009-10-08 |
BRPI0720827A2 (pt) | 2014-03-04 |
US20080281103A1 (en) | 2008-11-13 |
US20080161332A1 (en) | 2008-07-03 |
MX2009006921A (es) | 2009-07-06 |
CL2007003832A1 (es) | 2008-07-25 |
AR064547A1 (es) | 2009-04-08 |
DK2125827T3 (da) | 2010-12-20 |
ATE486877T1 (de) | 2010-11-15 |
CA2674154A1 (fr) | 2008-07-10 |
US8044202B2 (en) | 2011-10-25 |
KR20090094172A (ko) | 2009-09-03 |
PL2125827T3 (pl) | 2011-04-29 |
TW200835483A (en) | 2008-09-01 |
DE602007010359D1 (de) | 2010-12-16 |
US20080161333A1 (en) | 2008-07-03 |
CN101589046B (zh) | 2011-09-21 |
EP2125827B1 (fr) | 2010-11-03 |
PE20081844A1 (es) | 2009-01-26 |
KR101129861B1 (ko) | 2012-04-24 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
NO20092342L (no) | Azaspiroderivativater | |
NO20074592L (no) | Acetylenyl-pyrazolo-pyrimidinderivater som mGluR2-antagonister | |
NO20091766L (no) | Spiro-piperidinderivater | |
NO20073876L (no) | Pyrazolopyrimidinderivater som mGluR2-antagonister | |
NO20074258L (no) | Pyridin-2-karboksamidderivater som MGLUR5 antagonister | |
NO20060324L (no) | [1,8]Naftyridin-2-oner og relaterte forbindelser for behandling av Schizofreni | |
NO20073719L (no) | Kjemiske forbindelser | |
NO20070199L (no) | Substituerte kinazoloner som anti-kreftmidler | |
NO20063469L (no) | Polyeheterosykliske forbindelser og deres anvendelse som metabotrofe glutamat reseptorantagonister | |
NO20070489L (no) | 3-aminocyklopentankarboksamider som modulatorer av kjemokinreseptorer. | |
NO20084363L (no) | 2-Substituerte 4-benzylftalazinonderivater som histamin H1- og H3-antagonister | |
NO20072784L (no) | Pyridenkarboksamidderivater for anvendelse som anticancer midler | |
NO20085100L (no) | Nye forbindelser | |
NO20084845L (no) | 2-pyrazinonderivater for behandling av sykdom eller tilstander der inhibiering av neutrofil elastaseaktivitetet er gunstig | |
EA200801184A1 (ru) | Производные пипередин-4-ил-пиридазин-3-иламина как быстро диссоциирующие антагонисты рецептора дофамина 2 | |
NO20065456L (no) | Substituerte morfolinforbindelser for behandling av sykdommer i sentralnervesystemet | |
NO20063761L (no) | Sulfonamidderivater for behandling av sykdommer | |
NO20084872L (no) | 2-pyridonderivater for behandling av sykdom eller tilstander der inhibering av neutrofil elastaseaktivitet er gunstig | |
NO20076195L (no) | Nye 2-azetidinonderivater for behandling av hyperlipidemiske sykdommer | |
NO20076197L (no) | Nye 2-azetidinonderivater anvendbare i behandling av hyperlipidemiske tilstander | |
NO20082709L (no) | Kjemiske forbindelser | |
NO20090327L (no) | Nye forbindelser 384 | |
NO20090266L (no) | Piperazinylderivater anvendelige i behandlingen av GPR38 receptormedierte sykdommer | |
MX2009007411A (es) | Derivados de espiropiperidina-glicinamida. | |
NO20092689L (no) | Quinuclidinolderivater som muskarin reseptorantagonister |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FC2A | Withdrawal, rejection or dismissal of laid open patent application |